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Positron emission tomography studies of organophosphate chemical threats and oxime countermeasures

Neurobiology of disease, 2020-01, Vol.133, p.104455-104455, Article 104455

2020

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Development of effective PET and SPECT imaging agents for the serotonin transporter: has a twenty-year journey reached its destination?

Current topics in medicinal chemistry, 2010-10, Vol.10 (15), p.1499

2010

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The inhibition, reactivation and mechanism of VX-, sarin-, fluoro-VX and fluoro-sarin surrogates following their interaction with HuAChE and HuBuChE

Chemico-biological interactions, 2018-08, Vol.291, p.220-227

2018

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[ 11 C]Paraoxon: Radiosynthesis, Biodistribution and In Vivo Positron Emission Tomography Imaging in Rat

The Journal of pharmacology and experimental therapeutics, 2024-02, Vol.388 (2), p.333

2024

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Novel Organophosphate Ligand O‑(2-Fluoroethyl)-O‑(p‑Nitrophenyl)Methylphosphonate: Synthesis, Hydrolytic Stability and Analysis of the Inhibition and Reactivation of Cholinesterases

Chemical research in toxicology, 2016-11, Vol.29 (11), p.1810-1817

2016

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Positron emission tomography evaluation of oxime countermeasures in live rats using the tracer O‐(2‐[18F]fluoroethyl)‐O‐(p‐nitrophenyl)methylphosphonate [18F]‐VXS

Annals of the New York Academy of Sciences, 2020-11, Vol.1479 (1), p.180-195

2020

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Biological Distribution and Metabolic Profiles of Carbon-11 and Fluorine-18 Tracers of VX- and Sarin-Analogs in Sprague–Dawley Rats

Chemical research in toxicology, 2021-01, Vol.34 (1), p.63-69

2021

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Inhibition of the Vesicular Glutamate Transporter (VGLUT) with Congo Red Analogs: New Binding Insights

Neurochemical research, 2021-03, Vol.46 (3), p.494-503

2021

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Divergent synthesis of organophosphate [11C]VX- and [11C]Sarin-surrogates from a common set of starting materials

Applied radiation and isotopes, 2019-09, Vol.151, p.182-186

2019

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Tetrapeptide inhibitors of the glutamate vesicular transporter (VGLUT)

Bioorganic & medicinal chemistry letters, 2007-09, Vol.17 (18), p.5125-5128

2007

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Radiosynthesis of O‐(1‐[18F]fluoropropan‐2‐yl)‐O‐(4‐nitrophenyl)methylphosphonate: A novel PET tracer surrogate of sarin

Journal of labelled compounds & radiopharmaceuticals, 2018-12, Vol.61 (14), p.1089-1094

2018

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The development of benzo- and naphtho-fused quinoline-2,4-dicarboxylic acids as vesicular glutamate transporter (VGLUT) inhibitors reveals a possible role for neuroactive steroids

Bioorganic & medicinal chemistry letters, 2014-02, Vol.24 (3), p.850-854

2014

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An improved radiosynthesis of O‐(2‐[18F]fluoroethyl)‐O‐(p‐nitrophenyl)methylphosphonate: A first‐in‐class cholinesterase PET tracer

Journal of labelled compounds & radiopharmaceuticals, 2017-06, Vol.60 (7), p.337-342

2017

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Synthesis and anti-acetylcholinesterase properties of novel β- and γ-substituted alkoxy organophosphonates

Bioorganic & medicinal chemistry letters, 2013-04, Vol.23 (7), p.2048-2051

2013

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Radiosynthesis, ex Vivo Biodistribution, and in Vivo Positron Emission Tomography Imaging Evaluations of [11C]2-Pyridinealdoxime Methiodide ([11C]2-PAM): A First-In-Class Antidote Tracer for Organophosphate Intoxication

ACS chemical neuroscience, 2018-12, Vol.9 (12), p.3007-3014

2018

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Novel Lavendamycin Analogues as Antitumor Agents: Synthesis, in Vitro Cytotoxicity, Structure−Metabolism, and Computational Molecular Modeling Studies with NAD(P)H:Quinone Oxidoreductase 1

Journal of medicinal chemistry, 2005-12, Vol.48 (24), p.7733-7749

2005

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A Novel Fluorine-18 β‑Fluoroethoxy Organophosphate Positron Emission Tomography Imaging Tracer Targeted to Central Nervous System Acetylcholinesterase

ACS chemical neuroscience, 2014-07, Vol.5 (7), p.519-524

2014

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Lavendamycin Antitumor Agents: Structure-Based Design, Synthesis, and NAD(P)H:Quinone Oxidoreductase 1 (NQO1) Model Validation with Molecular Docking and Biological Studies

Journal of medicinal chemistry, 2008-06, Vol.51 (11), p.3104-3115

2008

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Isoxazole analogues bind the System Xc- transporter: Structure-activity relationship and pharmacophore model

Bioorganic & medicinal chemistry, 2010-01, Vol.18 (1), p.202-213

2010

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Inhibition of acetylcholinesterase by chromophore-linked fluorophosphonates

Bioorganic & medicinal chemistry letters, 2010-02, Vol.20 (3), p.1194-1197

2010

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Serotonin transporter inhibitors: synthesis and binding potency of 2′-methyl- and 3′-methyl-6-nitroquipazine

Bioorganic & medicinal chemistry letters, 2000-12, Vol.10 (23), p.2643-2646

2000

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Organic reactions at high pressure. Preparation of Wittig phosphonium salts at ambient temperature

Journal of organic chemistry, 1984-11, Vol.49 (22), p.4293-4295

1984

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Synthesis and in vitro evaluation of 2,3-dimethoxy-5-(fluoroalkyl)-substituted benzamides: high-affinity ligands for CNS dopamine D2 receptors

Journal of medicinal chemistry, 1991-05, Vol.34 (5), p.1612-1624

1991

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Synthesis of 2,3-dimethoxy-5-iodobenzoic acid

Journal of organic chemistry, 1991-08, Vol.56 (18), p.5451-5456

1991

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Positron emission tomography studies of organophosphate chemical threats and oxime countermeasures

Development of effective PET and SPECT imaging agents for the serotonin transporter: has a twenty-year journey reached its destination?

The inhibition, reactivation and mechanism of VX-, sarin-, fluoro-VX and fluoro-sarin surrogates following their interaction with HuAChE and HuBuChE

[ 11 C]Paraoxon: Radiosynthesis, Biodistribution and In Vivo Positron Emission Tomography Imaging in Rat

Novel Organophosphate Ligand O‑(2-Fluoroethyl)-O‑(p‑Nitrophenyl)Methylphosphonate: Synthesis, Hydrolytic Stability and Analysis of the Inhibition and Reactivation of Cholinesterases

Positron emission tomography evaluation of oxime countermeasures in live rats using the tracer O‐(2‐[18F]fluoroethyl)‐O‐(p‐nitrophenyl)methylphosphonate [18F]‐VXS

Biological Distribution and Metabolic Profiles of Carbon-11 and Fluorine-18 Tracers of VX- and Sarin-Analogs in Sprague–Dawley Rats

Inhibition of the Vesicular Glutamate Transporter (VGLUT) with Congo Red Analogs: New Binding Insights

Targeting Chikungunya Virus Replication by Benzoannulene Inhibitors

Divergent synthesis of organophosphate [11C]VX- and [11C]Sarin-surrogates from a common set of starting materials

Tetrapeptide inhibitors of the glutamate vesicular transporter (VGLUT)

Radiosynthesis of O‐(1‐[18F]fluoropropan‐2‐yl)‐O‐(4‐nitrophenyl)methylphosphonate: A novel PET tracer surrogate of sarin

The development of benzo- and naphtho-fused quinoline-2,4-dicarboxylic acids as vesicular glutamate transporter (VGLUT) inhibitors reveals a possible role for neuroactive steroids

An improved radiosynthesis of O‐(2‐[18F]fluoroethyl)‐O‐(p‐nitrophenyl)methylphosphonate: A first‐in‐class cholinesterase PET tracer

Synthesis and anti-acetylcholinesterase properties of novel β- and γ-substituted alkoxy organophosphonates

Radiosynthesis, ex Vivo Biodistribution, and in Vivo Positron Emission Tomography Imaging Evaluations of [11C]2-Pyridinealdoxime Methiodide ([11C]2-PAM): A First-In-Class Antidote Tracer for Organophosphate Intoxication

Novel Lavendamycin Analogues as Antitumor Agents: Synthesis, in Vitro Cytotoxicity, Structure−Metabolism, and Computational Molecular Modeling Studies with NAD(P)H:Quinone Oxidoreductase 1

A Novel Fluorine-18 β‑Fluoroethoxy Organophosphate Positron Emission Tomography Imaging Tracer Targeted to Central Nervous System Acetylcholinesterase

Lavendamycin Antitumor Agents: Structure-Based Design, Synthesis, and NAD(P)H:Quinone Oxidoreductase 1 (NQO1) Model Validation with Molecular Docking and Biological Studies

Isoxazole analogues bind the System Xc- transporter: Structure-activity relationship and pharmacophore model

Inhibition of acetylcholinesterase by chromophore-linked fluorophosphonates

Serotonin transporter inhibitors: synthesis and binding potency of 2′-methyl- and 3′-methyl-6-nitroquipazine

Organic reactions at high pressure. Preparation of Wittig phosphonium salts at ambient temperature

Synthesis and in vitro evaluation of 2,3-dimethoxy-5-(fluoroalkyl)-substituted benzamides: high-affinity ligands for CNS dopamine D2 receptors

Synthesis of 2,3-dimethoxy-5-iodobenzoic acid

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