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Structures of Kibdelomycin Bound to Staphylococcus aureus GyrB and ParE Showed a Novel U‑Shaped Binding Mode

ACS chemical biology, 2014-09, Vol.9 (9), p.2023-2031

2014

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Kibdelomycin is a bactericidal broad-spectrum aerobic antibacterial agent

Antimicrobial agents and chemotherapy, 2015-06, Vol.59 (6), p.3474-3481

2015

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Synthesis and Antibacterial Activity of Novel Pyrido[1,2,3-de][1,4]benzoxazine-6-carboxylic Acid Derivatives Carrying the 3-Cyclopropylaminomethyl-4-substituted-1-pyrrolidinyl Group as a C-10 Substituent

Journal of medicinal chemistry, 2008-06, Vol.51 (11), p.3238-3249

2008

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Stereoselective Synthesis of cis-2-Fluorocyclopropanecarboxylic Acid

Journal of organic chemistry, 2014-08, Vol.79 (15), p.7226-7231

2014

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Efficient synthesis of cyclopropylhydrazine salts

Tetrahedron letters, 2014-07, Vol.55 (30), p.4102-4104

2014

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Structure activity relationship of N-1 substituted 1,5-naphthyrid-2-one analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-9)

Bioorganic & medicinal chemistry letters, 2022-11, Vol.75, p.128808, Article 128808

2022

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Synthesis and Structure−Activity Relationship Studies of Highly Potent Novel Oxazolidinone Antibacterials

Journal of medicinal chemistry, 2008-10, Vol.51 (20), p.6558-6562

2008

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In Vitro and In Vivo Characterization of the Novel Oxabicyclooctane-Linked Bacterial Topoisomerase Inhibitor AM-8722, a Selective, Potent Inhibitor of Bacterial DNA Gyrase

Antimicrobial agents and chemotherapy, 2016-08, Vol.60 (8), p.4830-4839

2016

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Oxabicyclooctane-Linked Novel Bacterial Topoisomerase Inhibitors as Broad Spectrum Antibacterial Agents

ACS medicinal chemistry letters, 2014-05, Vol.5 (5), p.609-614

2014

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Tricyclic 1,5-naphthyridinone oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents-SAR of left-hand-side moiety (Part-2)

Bioorganic & medicinal chemistry letters, 2015-05, Vol.25 (9), p.1831-1835

2015

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Hydroxy tricyclic 1,5-naphthyridinone oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents-SAR of RHS moiety (Part-3)

Bioorganic & medicinal chemistry letters, 2015-06, Vol.25 (12), p.2473-2478

2015

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Structure activity relationship of pyridoxazinone substituted RHS analogs of oxabicyclooctane-linked 1,5-naphthyridinyl novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-6)

Bioorganic & medicinal chemistry letters, 2015-09, Vol.25 (17), p.3636-3643

2015

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Structure activity relationship of C-2 ether substituted 1,5-naphthyridine analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-5)

Bioorganic & medicinal chemistry letters, 2015-09, Vol.25 (17), p.3630-3635

2015

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Structure activity relationship of substituted 1,5-naphthyridine analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-4)

Bioorganic & medicinal chemistry letters, 2015-06, Vol.25 (11), p.2409-2415

2015

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Synthetic studies on duocarmycin. 1. Total synthesis of dl-duocarmycin A and its 2-epimer

Tetrahedron, 1994-02, Vol.50 (9), p.2793-2808

1994

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Synthetic studies on duocarmycin. 2. Synthesis and cytotoxicity of natural (+)-duocarmycin A and its three possible stereoisomers

Tetrahedron, 1994-02, Vol.50 (9), p.2809-2820

1994

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Synthesis and antitumor activity of novel cyclopropapyrroloindole(CPI) derivatives bearing methoxycarbonyl and trifluoromethyl groups

Bioorganic & medicinal chemistry letters, 1997-07, Vol.7 (13), p.1683-1688

1997

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The novel cyclopropapyrroloindole(CPI) bisalkylators bearing methoxycarbonyl and trifluoromethyl groups

Bioorganic & medicinal chemistry letters, 1998-06, Vol.8 (11), p.1387-1390

1998

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C1–C2-linker substituted 1,5-naphthyridine analogues of oxabicyclooctane-linked NBTIs as broad-spectrum antibacterial agents (part 7)

MedChemComm, 2015-01, Vol.6 (10), p.1773-1780

2015

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Synthesis and cytotoxicity of enantiomeric pairs of duocarmycin a and its 2-epimer

Bioorganic & medicinal chemistry letters, 1992-07, Vol.2 (7), p.755-758

1992

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Novel Seco Cyclopropa[c]pyrrolo[3,2-e]indole Bisalkylators Bearing a 3,3‘-Arylenebisacryloyl Group as a Linker

Journal of medicinal chemistry, 2001-04, Vol.44 (9), p.1396-1406

2001

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Novel Cyclopropapyrroloindole Derivative (AT-3510) Bearing Methoxycarbonyl and Trifluoromethyl Groups

Journal of medicinal chemistry, 1999-04, Vol.42 (8), p.1448-1458

1999

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A novel synthesis of (+)-duocarmycin SA

Tetrahedron letters, 1997-10, Vol.38 (41), p.7207-7208

1997

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Novel Seco Cyclopropa[ c ]pyrrolo[3,2- e ]indole Bisalkylators Bearing a 3,3‘-Arylenebisacryloyl Group as a Linker

Journal of medicinal chemistry, 2001-04, Vol.44 (9), p.1396-1406

2001

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Structures of Kibdelomycin Bound to Staphylococcus aureus GyrB and ParE Showed a Novel U‑Shaped Binding Mode

Kibdelomycin is a bactericidal broad-spectrum aerobic antibacterial agent

Synthesis and Antibacterial Activity of Novel Pyrido[1,2,3-de][1,4]benzoxazine-6-carboxylic Acid Derivatives Carrying the 3-Cyclopropylaminomethyl-4-substituted-1-pyrrolidinyl Group as a C-10 Substituent

Stereoselective Synthesis of cis-2-Fluorocyclopropanecarboxylic Acid

Efficient synthesis of cyclopropylhydrazine salts

Structure activity relationship of N-1 substituted 1,5-naphthyrid-2-one analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-9)

Synthesis and Structure−Activity Relationship Studies of Highly Potent Novel Oxazolidinone Antibacterials

In Vitro and In Vivo Characterization of the Novel Oxabicyclooctane-Linked Bacterial Topoisomerase Inhibitor AM-8722, a Selective, Potent Inhibitor of Bacterial DNA Gyrase

Oxabicyclooctane-Linked Novel Bacterial Topoisomerase Inhibitors as Broad Spectrum Antibacterial Agents

Tricyclic 1,5-naphthyridinone oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents-SAR of left-hand-side moiety (Part-2)

Hydroxy tricyclic 1,5-naphthyridinone oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents-SAR of RHS moiety (Part-3)

Structure activity relationship of pyridoxazinone substituted RHS analogs of oxabicyclooctane-linked 1,5-naphthyridinyl novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-6)

Structure activity relationship of C-2 ether substituted 1,5-naphthyridine analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-5)

Structure activity relationship of substituted 1,5-naphthyridine analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-4)

Synthetic studies on duocarmycin. 1. Total synthesis of dl-duocarmycin A and its 2-epimer

Synthetic studies on duocarmycin. 2. Synthesis and cytotoxicity of natural (+)-duocarmycin A and its three possible stereoisomers

Synthesis and antitumor activity of novel cyclopropapyrroloindole(CPI) derivatives bearing methoxycarbonyl and trifluoromethyl groups

The novel cyclopropapyrroloindole(CPI) bisalkylators bearing methoxycarbonyl and trifluoromethyl groups

C1–C2-linker substituted 1,5-naphthyridine analogues of oxabicyclooctane-linked NBTIs as broad-spectrum antibacterial agents (part 7)

C1-C2-linker substituted 1,5-naphthyridine analogues of oxabicyclooctane-linked NBTIs as broad-spectrum antibacterial agents (part 7)Electronic supplementary information (ESI) available: Synthetic details of compounds and intermediates. See DOI: 10.1039/c5md00297d

Synthesis and cytotoxicity of enantiomeric pairs of duocarmycin a and its 2-epimer

Novel Seco Cyclopropa[c]pyrrolo[3,2-e]indole Bisalkylators Bearing a 3,3‘-Arylenebisacryloyl Group as a Linker

Novel Cyclopropapyrroloindole Derivative (AT-3510) Bearing Methoxycarbonyl and Trifluoromethyl Groups

A novel synthesis of (+)-duocarmycin SA

Novel Seco Cyclopropa[ c ]pyrrolo[3,2- e ]indole Bisalkylators Bearing a 3,3‘-Arylenebisacryloyl Group as a Linker

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