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Pharmacological characterization of the competitive GLUK5 receptor antagonist decahydroisoquinoline LY466195 in vitro and in vivo

The Journal of pharmacology and experimental therapeutics, 2006-08, Vol.318 (2), p.772

2006

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Synthesis and Preclinical Characterization of LY3154885, a Human Dopamine D1 Receptor Positive Allosteric Modulator with an Improved Nonclinical Drug–Drug Interaction Risk Profile

Journal of medicinal chemistry, 2022-03, Vol.65 (5), p.3786-3797

2022

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GluK1 antagonists from 6-(tetrazolyl)phenyl decahydroisoquinoline derivatives: In vitro profile and in vivo analgesic efficacy

Bioorganic & medicinal chemistry letters, 2013-12, Vol.23 (23), p.6463-6466

2013

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GluK1 antagonists from 6-(carboxy)phenyl decahydroisoquinoline derivatives. SAR and evaluation of a prodrug strategy for oral efficacy in pain models

Bioorganic & medicinal chemistry letters, 2013-12, Vol.23 (23), p.6459-6462

2013

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A general method for the preparation of 2,3,5-trisubstituted-furo[3,2- b]pyridines

Tetrahedron letters, 2003-01, Vol.44 (4), p.725-728

2003

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Discovery of a Potent, Dual Serotonin and Norepinephrine Reuptake Inhibitor

ACS medicinal chemistry letters, 2013-06, Vol.4 (6), p.560-564

2013

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Novel Potent 5-HT1F Receptor Agonists: Structure−Activity Studies of a Series of Substituted N-[3-(1-Methyl-4-piperidinyl)-1H-pyrrolo[3,2-b]pyridin-5-yl]amides

Journal of medicinal chemistry, 2003-07, Vol.46 (14), p.3060-3071

2003

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Benzopyranoisoxazolidines as Chiral Auxiliaries for Asymmetric Synthesis

Angewandte Chemie (International ed.), 1995-04, Vol.34 (7), p.793-795

1995

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Substituted furo[3,2-b]pyridines: novel bioisosteres of 5-HT1F receptor agonists

Bioorganic & medicinal chemistry letters, 2004-01, Vol.14 (1), p.167-170

2004

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Substituted furo[3,2- b]pyridines: novel bioisosteres of 5-HT 1F receptor agonists

Bioorganic & medicinal chemistry letters, 2004-01, Vol.14 (1), p.167-170

2004

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Discovery of selective N-[3-(1-methyl-piperidine-4-carbonyl)-phenyl]-benzamide-based 5-HT1F receptor agonists: Evolution from bicyclic to monocyclic cores

Bioorganic & medicinal chemistry letters, 2015-10, Vol.25 (19), p.4337-4341

2015

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On the Stereochemistry of Diaryl-Substituted Cyclohexanones Formed by Michael Reactions. Trans to Cis Isomerization of Their Ketals under Basic Conditions

Journal of organic chemistry, 1998-06, Vol.63 (13), p.4359-4365

1998

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Synthesis of C1-C8 and C9-C24 fragments of (−)-discodermolide: use of asymmetric alkylation and stereoselective aldol reactions

Tetrahedron letters, 1999-07, Vol.40 (30), p.5449-5453

1999

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Benzopyranoisoxazolidines as Chiral Auxiliaries for Asymmetric Synthesis

Angewandte Chemie International Edition, 1995-04, Vol.34 (7), p.793-795

1995

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A tandem Michael-aldol reaction sequence: An undergraduate research organic experiment

Journal of chemical education, 1989-06, Vol.66 (6), p.520

1989

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The Synthesis of Naturally Occurring ()-Calyculin A

Angewandte Chemie (International ed.), 1994-03, Vol.33 (6), p.673-675

1994

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Novel potent 5-HT(1F) receptor agonists: structure-activity studies of a series of substituted N-[3-(1-methyl-4-piperidinyl)-1H-pyrrolo[3,2-b]pyridin-5-yl]amides

Journal of medicinal chemistry, 2003-07, Vol.46 (14), p.3060-3071

2003

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Novel Potent 5-HT 1F Receptor Agonists: Structure−Activity Studies of a Series of Substituted N -[3-(1-Methyl-4-piperidinyl)-1 H -pyrrolo[3,2- b ]pyridin-5-yl]amides

Journal of medicinal chemistry, 2003-07, Vol.46 (14), p.3060-3071

2003

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Use of 2-trimethylsilylethyl as a protecting group in phosphate monoester synthesis

Tetrahedron letters, 1993-12, Vol.33 (50), p.7685-7686

1993

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A General Method for the Preparation of 2,3,5-Trisubstituted-furo[3,2-b]pyridines

ChemInform, 2003-05, Vol.34 (18), p.no-no

2003

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Benzopyranoisoxazolidine als Auxiliare für die asymmetrische Synthese

Angewandte Chemie, 1995-03, Vol.107 (7), p.869-871

1995

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A Tandem Michael-Aldol Reaction Sequence

Journal of chemical education, 1989-06, Vol.66 (6), p.520

1989

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Pharmacological characterization of the competitive GLUK5 receptor antagonist decahydroisoquinoline LY466195 in vitro and in vivo

Synthesis and Preclinical Characterization of LY3154885, a Human Dopamine D1 Receptor Positive Allosteric Modulator with an Improved Nonclinical Drug–Drug Interaction Risk Profile

GluK1 antagonists from 6-(tetrazolyl)phenyl decahydroisoquinoline derivatives: In vitro profile and in vivo analgesic efficacy

GluK1 antagonists from 6-(carboxy)phenyl decahydroisoquinoline derivatives. SAR and evaluation of a prodrug strategy for oral efficacy in pain models

A general method for the preparation of 2,3,5-trisubstituted-furo[3,2- b]pyridines

Discovery of a Potent, Dual Serotonin and Norepinephrine Reuptake Inhibitor

Novel Potent 5-HT1F Receptor Agonists: Structure−Activity Studies of a Series of Substituted N-[3-(1-Methyl-4-piperidinyl)-1H-pyrrolo[3,2-b]pyridin-5-yl]amides

Benzopyranoisoxazolidines as Chiral Auxiliaries for Asymmetric Synthesis

Substituted furo[3,2-b]pyridines: novel bioisosteres of 5-HT1F receptor agonists

Substituted furo[3,2- b]pyridines: novel bioisosteres of 5-HT 1F receptor agonists

Discovery of selective N-[3-(1-methyl-piperidine-4-carbonyl)-phenyl]-benzamide-based 5-HT1F receptor agonists: Evolution from bicyclic to monocyclic cores

On the Stereochemistry of Diaryl-Substituted Cyclohexanones Formed by Michael Reactions. Trans to Cis Isomerization of Their Ketals under Basic Conditions

Ethyl (3S,4aR,6S,8aR)-6-(4-Ethoxycar- bonylimidazol-1-ylmethyl)decahydroiso- quinoline-3-carboxylic Ester: A Prodrug of a GluR5 Kainate Receptor Antagonist Active in Two Animal Models of Acute Migraine

Synthesis of C1-C8 and C9-C24 fragments of (−)-discodermolide: use of asymmetric alkylation and stereoselective aldol reactions

Benzopyranoisoxazolidines as Chiral Auxiliaries for Asymmetric Synthesis

A tandem Michael-aldol reaction sequence: An undergraduate research organic experiment

The Synthesis of Naturally Occurring ()-Calyculin A

Two prodrugs of potent and selective GluR5 kainate receptor antagonists actives in three animal models of pain : 2005 American Chemical Society Award for Computers in Chemical and Pharmaceutical Research

Novel potent 5-HT(1F) receptor agonists: structure-activity studies of a series of substituted N-[3-(1-methyl-4-piperidinyl)-1H-pyrrolo[3,2-b]pyridin-5-yl]amides

Novel Potent 5-HT 1F Receptor Agonists: Structure−Activity Studies of a Series of Substituted N -[3-(1-Methyl-4-piperidinyl)-1 H -pyrrolo[3,2- b ]pyridin-5-yl]amides

Use of 2-trimethylsilylethyl as a protecting group in phosphate monoester synthesis

Ethyl (3S, 4aR, 6S, 8aR)-6-(4-ethoxycarbonylimidazol-1-ylmethyl)decahydroisoquinoline-3-c arboxylic ester: A prodrug of a GluR5 kainate receptor antagonist active in two animal models of acute migraine

A General Method for the Preparation of 2,3,5-Trisubstituted-furo[3,2-b]pyridines

Benzopyranoisoxazolidine als Auxiliare für die asymmetrische Synthese

A Tandem Michael-Aldol Reaction Sequence

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