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The Importance of Medicinal Chemistry Knowledge in the Clinical Pharmacist’s Education

American journal of pharmaceutical education, 2018-03, Vol.82 (2), p.6083-114, Article 6083

Fernandes, João Paulo S.

2018

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Metabolite profile of Nectandra oppositifolia Nees & Mart. and assessment of antitrypanosomal activity of bioactive compounds through efficiency analyses

PloS one, 2021-02, Vol.16 (2), p.e0247334-e0247334

2021

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Piperazine amides with desirable solubility, physicochemical and drug-like properties: Synthesis and evaluation of the anti-Trypanosoma cruzi activity

Saudi pharmaceutical journal, 2023-07, Vol.31 (7), p.1265-1273

2023

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Antihistamines H1 as Potential Anthelmintic Agents against the Zoonotic Parasite Angiostrongylus cantonensis

ACS omega, 2024-07, Vol.9 (28), p.31159-31165

2024

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Synthetic Analogues of Gibbilimbol B Induce Bioenergetic Damage and Calcium Imbalance in Trypanosoma cruzi

Life (Basel, Switzerland), 2023-02, Vol.13 (3), p.663

2023

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Investigation of Structure–Activity Relationships for Benzoyl and Cinnamoyl Piperazine/Piperidine Amides as Tyrosinase Inhibitors

ACS omega, 2023-11, Vol.8 (46), p.44265-44275

2023

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Gibbilimbol analogues as antiparasitic agents—Synthesis and biological activity against Trypanosoma cruzi and Leishmania (L.) infantum

Bioorganic & medicinal chemistry letters, 2016-02, Vol.26 (4), p.1180-1183

2016

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Histamine research advancements in the second year of the COVID-19 pandemic: report of the European Histamine Research Society (EHRS)

Inflammation research, 2022-08, Vol.71 (7-8), p.995-998

2022

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Esterification of p -Coumaric Acid Improves the Control over Melanoma Cell Growth

Biomedicines, 2023-01, Vol.11 (1), p.196

2023

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Differential contribution of H3R antagonism by LINS01 compounds on memory, anxiety-like behaviour and spontaneous locomotor activity in healthy rats

Behavioural brain research, 2020-01, Vol.377, p.112230, Article 112230

2020

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Lethal action of Licarin A derivatives in Leishmania (L.) infantum: Imbalance of calcium and bioenergetic metabolism

Biochimie, 2023-05, Vol.208, p.141-150

2023

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Toward anthelmintic drug candidates for toxocariasis: Challenges and recent developments

European journal of medicinal chemistry, 2023-05, Vol.251, p.115268-115268, Article 115268

2023

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Coumaric acid derivatives as tyrosinase inhibitors: Efficacy studies through in silico, in vitro and ex vivo approaches

Bioorganic chemistry, 2020-10, Vol.103, p.104108, Article 104108

2020

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Histamine H3 receptor and cholinesterases as synergistic targets for cognitive decline: Strategies to the rational design of multitarget ligands

Chemical biology & drug design, 2021-08, Vol.98 (2), p.212-225

2021

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Multitargeting approaches to cognitive impairment: Synthesis of aryl-alkylpiperazines and assessment at cholinesterases, histamine H3 and dopamine D3 receptors

Bioorganic & medicinal chemistry, 2023-01, Vol.78, p.117132-117132, Article 117132

2023

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Novel potent vasodilating agents: Evaluation of the activity and potency of LINS01005 and derivatives in rat aorta

European journal of pharmaceutical sciences, 2020-02, Vol.143, p.105171-105171, Article 105171

2020

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Optimization of physicochemical properties is a strategy to improve drug-likeness associated with activity: Novel active and selective compounds against Trypanosoma cruzi

European journal of pharmaceutical sciences, 2022-04, Vol.171, p.106114-106114, Article 106114

2022

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Neurotoxicity Assessment of 1-[(2,3-Dihydro-1-Benzofuran-2-yl)Methyl]Piperazine (LINS01 Series) Derivatives and their Protective Effect on Cocaine-Induced Neurotoxicity Model in SH-SY5Y Cell Culture

Neurotoxicity research, 2022-12, Vol.40 (6), p.1653-1663

2022

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Bioisosteric modification on benzylidene‐carbonyl compounds improved the drug‐likeness and maintained the antifungal activity against Sporothrix brasiliensis

Chemical biology & drug design, 2022-03, Vol.99 (3), p.391-397

2022

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Coumaric acid analogues inhibit growth and melanin biosynthesis in Cryptococcus neoformans and potentialize amphotericin B antifungal activity

European journal of pharmaceutical sciences, 2020-10, Vol.153, p.105473-105473, Article 105473

2020

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Novel potent (dihydro)benzofuranyl piperazines as human histamine receptor ligands – Functional characterization and modeling studies on H3 and H4 receptors

Bioorganic & medicinal chemistry, 2021-01, Vol.30, p.115924, Article 115924

2021

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Evaluation of the histamine H3 receptor antagonists from LINS01 series as cholinesterases inhibitors: Enzymatic and modeling studies

Chemical biology & drug design, 2022-11, Vol.100 (5), p.722-729

2022

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Profiling of LINS01 compounds at human dopamine D2 and D3 receptors

Journal of chemical sciences (Bangalore, India), 2020-12, Vol.132 (1), Article 5

2020

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The Novel H4R Antagonist 1-[(5-Chloro-2,3-Dihydro-1-Benzofuran-2-Yl)Methyl]-4-Methyl-Piperazine (LINS01007) Attenuates Several Symptoms in Murine Allergic Asthma

Cellular physiology and biochemistry, 2020-11, Vol.54 (6), p.1163-1176

2020

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New alkenyl derivative from Piper malacophyllum and analogues: Antiparasitic activity against Trypanosoma cruzi and Leishmania infantum

Chemical biology & drug design, 2017-11, Vol.90 (5), p.1007-1011

2017

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The Importance of Medicinal Chemistry Knowledge in the Clinical Pharmacist’s Education

Metabolite profile of Nectandra oppositifolia Nees & Mart. and assessment of antitrypanosomal activity of bioactive compounds through efficiency analyses

Piperazine amides with desirable solubility, physicochemical and drug-like properties: Synthesis and evaluation of the anti-Trypanosoma cruzi activity

Antihistamines H1 as Potential Anthelmintic Agents against the Zoonotic Parasite Angiostrongylus cantonensis

Synthetic Analogues of Gibbilimbol B Induce Bioenergetic Damage and Calcium Imbalance in Trypanosoma cruzi

Investigation of Structure–Activity Relationships for Benzoyl and Cinnamoyl Piperazine/Piperidine Amides as Tyrosinase Inhibitors

Gibbilimbol analogues as antiparasitic agents—Synthesis and biological activity against Trypanosoma cruzi and Leishmania (L.) infantum

Histamine research advancements in the second year of the COVID-19 pandemic: report of the European Histamine Research Society (EHRS)

Esterification of p -Coumaric Acid Improves the Control over Melanoma Cell Growth

Differential contribution of H3R antagonism by LINS01 compounds on memory, anxiety-like behaviour and spontaneous locomotor activity in healthy rats

Lethal action of Licarin A derivatives in Leishmania (L.) infantum: Imbalance of calcium and bioenergetic metabolism

Toward anthelmintic drug candidates for toxocariasis: Challenges and recent developments

Coumaric acid derivatives as tyrosinase inhibitors: Efficacy studies through in silico, in vitro and ex vivo approaches

Histamine H3 receptor and cholinesterases as synergistic targets for cognitive decline: Strategies to the rational design of multitarget ligands

Multitargeting approaches to cognitive impairment: Synthesis of aryl-alkylpiperazines and assessment at cholinesterases, histamine H3 and dopamine D3 receptors

Novel potent vasodilating agents: Evaluation of the activity and potency of LINS01005 and derivatives in rat aorta

Optimization of physicochemical properties is a strategy to improve drug-likeness associated with activity: Novel active and selective compounds against Trypanosoma cruzi

Neurotoxicity Assessment of 1-[(2,3-Dihydro-1-Benzofuran-2-yl)Methyl]Piperazine (LINS01 Series) Derivatives and their Protective Effect on Cocaine-Induced Neurotoxicity Model in SH-SY5Y Cell Culture

Bioisosteric modification on benzylidene‐carbonyl compounds improved the drug‐likeness and maintained the antifungal activity against Sporothrix brasiliensis

Coumaric acid analogues inhibit growth and melanin biosynthesis in Cryptococcus neoformans and potentialize amphotericin B antifungal activity

Novel potent (dihydro)benzofuranyl piperazines as human histamine receptor ligands – Functional characterization and modeling studies on H3 and H4 receptors

Evaluation of the histamine H3 receptor antagonists from LINS01 series as cholinesterases inhibitors: Enzymatic and modeling studies

Profiling of LINS01 compounds at human dopamine D2 and D3 receptors

The Novel H4R Antagonist 1-[(5-Chloro-2,3-Dihydro-1-Benzofuran-2-Yl)Methyl]-4-Methyl-Piperazine (LINS01007) Attenuates Several Symptoms in Murine Allergic Asthma

New alkenyl derivative from Piper malacophyllum and analogues: Antiparasitic activity against Trypanosoma cruzi and Leishmania infantum

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