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Computational aptamer design for spike glycoprotein (S) (SARS CoV-2) detection with an electrochemical aptasensor

Applied microbiology and biotechnology, 2024-12, Vol.108 (1), p.259-259, Article 259

2024

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Synthesis and structure–activity relationship of new 1,5-dialkyl-1,5-benzodiazepines as cholecystokinin-2 receptor antagonists

Bioorganic & medicinal chemistry, 2011-07, Vol.19 (14), p.4257-4273

2011

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From High-Throughput Screening to Target Validation: Benzo[d]isothiazoles as Potent and Selective Agonists of Human Transient Receptor Potential Cation Channel Subfamily M Member 5 Possessing In Vivo Gastrointestinal Prokinetic Activity in Rodents

Journal of medicinal chemistry, 2021-05, Vol.64 (9), p.5931-5955

2021

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Substituted Indole-2-carboxylates as in Vivo Potent Antagonists Acting as the Strychnine-Insensitive Glycine Binding Site

Journal of medicinal chemistry, 1997-03, Vol.40 (6), p.841-850

1997

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Novel morpholine scaffolds as selective dopamine (DA) D3 receptor antagonists

Bioorganic & medicinal chemistry letters, 2016-02, Vol.26 (4), p.1329-1332

2016

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1,2,4-Triazolyl 5‑Azaspiro[2.4]heptanes: Lead Identification and Early Lead Optimization of a New Series of Potent and Selective Dopamine D3 Receptor Antagonists

Journal of medicinal chemistry, 2016-09, Vol.59 (18), p.8549-8576

2016

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1,2,4-Triazolyl octahydropyrrolo[2,3-b]pyrroles: A new series of potent and selective dopamine D3 receptor antagonists

Bioorganic & medicinal chemistry, 2016-04, Vol.24 (8), p.1619-1636

2016

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Synthesis and Pharmacological Characterization of Novel Druglike Corticotropin-Releasing Factor 1 Antagonists

Journal of medicinal chemistry, 2008-12, Vol.51 (23), p.7370-7379

2008

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Ciprofloxacin affects conformational equilibria of DNA gyrase A in the presence of magnesium ions

Journal of molecular biology, 2001-08, Vol.311 (1), p.195-203

2001

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Generation of a Focused Set of GSK Compounds Biased toward Ligand-Gated Ion-Channel Ligands

Journal of chemical information and modeling, 2006-03, Vol.46 (2), p.659-664

2006

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Dihydropyrrole[2,3-d]pyridine Derivatives as Novel Corticotropin-Releasing Factor-1 Antagonists: Mapping of the Receptor Binding Pocket by in Silico Docking Studies

Journal of medicinal chemistry, 2008-11, Vol.51 (22), p.7273-7286

2008

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Synthesis and pharmacological characterisation of 2,4-Dicarboxy-pyrroles as selective non-Competitive mGluR1 antagonists

Bioorganic & medicinal chemistry, 2003-01, Vol.11 (2), p.171-183

2003

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Synthesis and SAR of New 5-Phenyl-3-ureido-1,5-benzodiazepines as Cholecystokinin-B Receptor Antagonists

Journal of medicinal chemistry, 2000-10, Vol.43 (20), p.3596-3613

2000

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Substituted Analogues of GV150526 as Potent Glycine Binding Site Antagonists in Animal Models of Cerebral Ischemia

Journal of medicinal chemistry, 1999-09, Vol.42 (18), p.3486-3493

1999

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(E)-3-(2-(N-Phenylcarbamoyl)vinyl)pyrrole-2-carboxylic Acid Derivatives. A Novel Class of Glycine Site Antagonists

Journal of medicinal chemistry, 1998-03, Vol.41 (6), p.808-820

1998

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Cholinergic Agents Structurally Related to Furtrethonium. 2. Synthesis and Antimuscarinic Activity of a Series of N-[5-[(1'-Substituted-acetoxy)methyl]-2-furfuryl]dialkylamines

Journal of medicinal chemistry, 1994-12, Vol.37 (25), p.4278-4287

1994

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Synthesis and biological evaluation of 4-heterotribactams

Bioorganic & medicinal chemistry letters, 1995-06, Vol.5 (12), p.1235-1240

1995

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3-Methyl pyrrole-2,4-dicarboxylic acid 2-propyl ester 4-(1,2,2-trimethyl-propyl) ester: an exploration of the C-2 position. Part I

Farmaco (Società chimica italiana : 1989), 2004-03, Vol.59 (3), p.175-183

2004

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Benzoazepine derivative as potent antagonists of the glycine binding site associated to the NMDA receptor

Farmaco (Società chimica italiana : 1989), 2003-09, Vol.58 (9), p.723-738

2003

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Synthesis and SAR of New 5-Phenyl-3-ureido-1,5-benzodiazepines as Cholecystokinin-B Receptor Antagonists

Journal of medicinal chemistry, 2000-12, Vol.43 (26), p.5057-5057

2000

Volltextzugriff (PDF)

(E)-3-(2-(N-Phenylcarbamoyl)vinyl)pyrrole-2-carboxylic Acid Derivatives. A Novel Class of Glycine Site Antagonists

Journal of medicinal chemistry, 1998-03, Vol.41 (6), p.808-820

1998

Volltextzugriff (PDF)

Statistical analysis on a series of glycine antagonists

Farmaco (Società chimica italiana : 1989), 2000-03, Vol.55 (3), p.194-196

2000

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Cycloalkyl Indole-2-Carboxylates as Useful Tools for Mapping the "North-Eastern" Region of the Glycine Binding Site Associated with the NMDA Receptor

Archiv der Pharmazie (Weinheim), 1999-03, Vol.332 (3), p.73-80

1999

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A Combinatorial Approach to [1,5]Benzothiazepine Derivatives as Potential Antibacterial Agents

Journal of combinatorial chemistry, 2001-03, Vol.3 (2), p.224-228

2001

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Novel glycine antagonists as potent neuroprotective agents

Pharmacochemistry Library, 1997, Vol.28, p.81-95

1997

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Computational aptamer design for spike glycoprotein (S) (SARS CoV-2) detection with an electrochemical aptasensor

Synthesis and structure–activity relationship of new 1,5-dialkyl-1,5-benzodiazepines as cholecystokinin-2 receptor antagonists

From High-Throughput Screening to Target Validation: Benzo[d]isothiazoles as Potent and Selective Agonists of Human Transient Receptor Potential Cation Channel Subfamily M Member 5 Possessing In Vivo Gastrointestinal Prokinetic Activity in Rodents

Substituted Indole-2-carboxylates as in Vivo Potent Antagonists Acting as the Strychnine-Insensitive Glycine Binding Site

Novel morpholine scaffolds as selective dopamine (DA) D3 receptor antagonists

1,2,4-Triazolyl 5‑Azaspiro[2.4]heptanes: Lead Identification and Early Lead Optimization of a New Series of Potent and Selective Dopamine D3 Receptor Antagonists

1,2,4-Triazolyl octahydropyrrolo[2,3-b]pyrroles: A new series of potent and selective dopamine D3 receptor antagonists

Synthesis and Pharmacological Characterization of Novel Druglike Corticotropin-Releasing Factor 1 Antagonists

Ciprofloxacin affects conformational equilibria of DNA gyrase A in the presence of magnesium ions

Generation of a Focused Set of GSK Compounds Biased toward Ligand-Gated Ion-Channel Ligands

Dihydropyrrole[2,3-d]pyridine Derivatives as Novel Corticotropin-Releasing Factor-1 Antagonists: Mapping of the Receptor Binding Pocket by in Silico Docking Studies

Synthesis and pharmacological characterisation of 2,4-Dicarboxy-pyrroles as selective non-Competitive mGluR1 antagonists

Synthesis and SAR of New 5-Phenyl-3-ureido-1,5-benzodiazepines as Cholecystokinin-B Receptor Antagonists

Substituted Analogues of GV150526 as Potent Glycine Binding Site Antagonists in Animal Models of Cerebral Ischemia

(E)-3-(2-(N-Phenylcarbamoyl)vinyl)pyrrole-2-carboxylic Acid Derivatives. A Novel Class of Glycine Site Antagonists

Cholinergic Agents Structurally Related to Furtrethonium. 2. Synthesis and Antimuscarinic Activity of a Series of N-[5-[(1'-Substituted-acetoxy)methyl]-2-furfuryl]dialkylamines

Synthesis and biological evaluation of 4-heterotribactams

3-Methyl pyrrole-2,4-dicarboxylic acid 2-propyl ester 4-(1,2,2-trimethyl-propyl) ester: an exploration of the C-2 position. Part I

Benzoazepine derivative as potent antagonists of the glycine binding site associated to the NMDA receptor

Synthesis and SAR of New 5-Phenyl-3-ureido-1,5-benzodiazepines as Cholecystokinin-B Receptor Antagonists

(E)-3-(2-(N-Phenylcarbamoyl)vinyl)pyrrole-2-carboxylic Acid Derivatives. A Novel Class of Glycine Site Antagonists

Statistical analysis on a series of glycine antagonists

Cycloalkyl Indole-2-Carboxylates as Useful Tools for Mapping the "North-Eastern" Region of the Glycine Binding Site Associated with the NMDA Receptor

A Combinatorial Approach to [1,5]Benzothiazepine Derivatives as Potential Antibacterial Agents

Novel glycine antagonists as potent neuroprotective agents

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