UB Paderborn / Katalog / Suche / in CDI

Design and Synthesis of 8-Hydroxy-[1,6]Naphthyridines as Novel Inhibitors of HIV-1 Integrase in Vitro and in Infected Cells

Journal of medicinal chemistry, 2003-02, Vol.46 (4), p.453-456

2003

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4-Aryl-2,4-dioxobutanoic Acid Inhibitors of HIV-1 Integrase and Viral Replication in Cells

Journal of medicinal chemistry, 2000-12, Vol.43 (26), p.4923-4926

2000

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Isolation, structure, and HIV-1-integrase inhibitory activity of structurally diverse fungal metabolites

Journal of industrial microbiology & biotechnology, 2003-12, Vol.30 (12), p.721-731

2003

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The Complestatins as HIV-1 Integrase Inhibitors. Efficient Isolation, Structure Elucidation, and Inhibitory Activities of Isocomplestatin, Chloropeptin I, New Complestatins, A and B, and Acid-Hydrolysis Products of Chloropeptin I

Journal of natural products (Washington, D.C.), 2001-07, Vol.64 (7), p.874-882

2001

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Differential divalent cation requirements uncouple the assembly and catalytic reactions of human immunodeficiency virus type 1 integrase

Journal of Virology, 1997-09, Vol.71 (9), p.7005-7011

1997

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Diketo Acid Inhibitor Mechanism and HIV-1 Integrase: Implications for Metal Binding in the Active Site of Phosphotransferase Enzymes

Proceedings of the National Academy of Sciences - PNAS, 2002-05, Vol.99 (10), p.6661-6666

2002

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Inhibitors of Strand Transfer That Prevent Integration and Inhibit HIV-1 Replication in Cells

Science (American Association for the Advancement of Science), 2000-01, Vol.287 (5453), p.646-650

2000

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Isolation, Structure, Absolute Stereochemistry, and HIV-1 Integrase Inhibitory Activity of Integrasone, a Novel Fungal Polyketide

Journal of natural products (Washington, D.C.), 2004-05, Vol.67 (5), p.872-874

2004

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Conformational change in the floor of the human rhinovirus canyon blocks adsorption to HeLa cell receptors

Journal of Virology, 1989-05, Vol.63 (5), p.2002-2007

1989

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HIV-1 Integrase Inhibitors That Compete with the Target DNA Substrate Define a Unique Strand Transfer Conformation for Integrase

Proceedings of the National Academy of Sciences - PNAS, 2000-10, Vol.97 (21), p.11244-11249

2000

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Isolation, Structure, and HIV-1 Integrase Inhibitory Activity of Cytosporic Acid, a Fungal Metabolite Produced by a Cytospora sp

Journal of natural products (Washington, D.C.), 2003-04, Vol.66 (4), p.551-553

2003

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The role of manganese in promoting multimerization and assembly of human immunodeficiency virus type 1 integrase as a catalytically active complex on immobilized long terminal repeat substrates

Journal of Virology, 1996-03, Vol.70 (3), p.1424-1432

1996

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Crystal structure of human rhinovirus serotype 1A (HRV1A)

Journal of molecular biology, 1989-11, Vol.210 (1), p.91-111

1989

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A Naphthyridine Carboxamide Provides Evidence for Discordant Resistance between Mechanistically Identical Inhibitors of HIV-1 Integrase

Proceedings of the National Academy of Sciences - PNAS, 2004-08, Vol.101 (31), p.11233-11238

2004

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Isolation, Structure and HIV-1 Integrase Inhibitory Activity of Exophillic Acid, a Novel Fungal Metabolite from Exophiala pisciphila

The Journal of Antibiotics, 2003/12/25, Vol.56(12), pp.1018-1023

2003

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Equivalent inhibition of half-site and full-site retroviral strand transfer reactions by structurally diverse compounds

Journal of Virology, 1997-01, Vol.71 (1), p.807-811

1997

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Integrastatins: structure and HIV-1 integrase inhibitory activities of two novel racemic tetracyclic aromatic heterocycles produced by two fungal species

Tetrahedron letters, 2002-03, Vol.43 (13), p.2351-2354

2002

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Structure, Stereochemistry, and Biological Activity of Integramycin, a Novel Hexacyclic Natural Product Produced by Actinoplanes sp. that Inhibits HIV-1 Integrase

Organic letters, 2002-04, Vol.4 (7), p.1123-1126

2002

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Structure and absolute stereochemistry of HIV-1 integrase inhibitor integric acid. A novel eremophilane sesquiterpenoid produced by a Xylaria sp

Tetrahedron letters, 1999-12, Vol.40 (50), p.8775-8779

1999

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X-ray structure of simian immunodeficiency virus integrase containing the core and C-terminal domain (residues 50-293)--an initial glance of the viral DNA binding platform

Journal of molecular biology, 2000-02, Vol.296 (2), p.521-533

2000

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A series of 5-(5,6)-dihydrouracil substituted 8-hydroxy-[1,6]naphthyridine-7-carboxylic acid 4-fluorobenzylamide inhibitors of HIV-1 integrase and viral replication in cells

Bioorganic & medicinal chemistry letters, 2005-10, Vol.15 (20), p.4550-4554

2005

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Four novel bis-(naphtho-γ-pyrones) isolated from Fusarium species as inhibitors of HIV-1 integrase

Bioorganic & medicinal chemistry letters, 2003-02, Vol.13 (4), p.713-717

2003

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A series of 5-aminosubstituted 4-fluorobenzyl-8-hydroxy-[1,6]naphthyridine-7-carboxamide HIV-1 integrase inhibitors

Bioorganic & medicinal chemistry letters, 2006-06, Vol.16 (11), p.2900-2904

2006

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Chemical and enzymatic modifications of integric acid and HIV-1 integrase inhibitory activity

Bioorganic & medicinal chemistry letters, 2000-02, Vol.10 (3), p.235-238

2000

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Isolation and Characterization of Novel Human Immunodeficiency Virus Integrase Inhibitors from Fungal Metabolites

Antiviral chemistry & chemotherapy, 1999-04, Vol.10 (2), p.63-70

1999

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Design and Synthesis of 8-Hydroxy-[1,6]Naphthyridines as Novel Inhibitors of HIV-1 Integrase in Vitro and in Infected Cells

4-Aryl-2,4-dioxobutanoic Acid Inhibitors of HIV-1 Integrase and Viral Replication in Cells

Isolation, structure, and HIV-1-integrase inhibitory activity of structurally diverse fungal metabolites

The Complestatins as HIV-1 Integrase Inhibitors. Efficient Isolation, Structure Elucidation, and Inhibitory Activities of Isocomplestatin, Chloropeptin I, New Complestatins, A and B, and Acid-Hydrolysis Products of Chloropeptin I

Differential divalent cation requirements uncouple the assembly and catalytic reactions of human immunodeficiency virus type 1 integrase

Diketo Acid Inhibitor Mechanism and HIV-1 Integrase: Implications for Metal Binding in the Active Site of Phosphotransferase Enzymes

Inhibitors of Strand Transfer That Prevent Integration and Inhibit HIV-1 Replication in Cells

Isolation, Structure, Absolute Stereochemistry, and HIV-1 Integrase Inhibitory Activity of Integrasone, a Novel Fungal Polyketide

Conformational change in the floor of the human rhinovirus canyon blocks adsorption to HeLa cell receptors

HIV-1 Integrase Inhibitors That Compete with the Target DNA Substrate Define a Unique Strand Transfer Conformation for Integrase

Isolation, Structure, and HIV-1 Integrase Inhibitory Activity of Cytosporic Acid, a Fungal Metabolite Produced by a Cytospora sp

The role of manganese in promoting multimerization and assembly of human immunodeficiency virus type 1 integrase as a catalytically active complex on immobilized long terminal repeat substrates

Crystal structure of human rhinovirus serotype 1A (HRV1A)

A Naphthyridine Carboxamide Provides Evidence for Discordant Resistance between Mechanistically Identical Inhibitors of HIV-1 Integrase

Isolation, Structure and HIV-1 Integrase Inhibitory Activity of Exophillic Acid, a Novel Fungal Metabolite from Exophiala pisciphila

Equivalent inhibition of half-site and full-site retroviral strand transfer reactions by structurally diverse compounds

Integrastatins: structure and HIV-1 integrase inhibitory activities of two novel racemic tetracyclic aromatic heterocycles produced by two fungal species

Structure, Stereochemistry, and Biological Activity of Integramycin, a Novel Hexacyclic Natural Product Produced by Actinoplanes sp. that Inhibits HIV-1 Integrase

Structure and absolute stereochemistry of HIV-1 integrase inhibitor integric acid. A novel eremophilane sesquiterpenoid produced by a Xylaria sp

X-ray structure of simian immunodeficiency virus integrase containing the core and C-terminal domain (residues 50-293)--an initial glance of the viral DNA binding platform

A series of 5-(5,6)-dihydrouracil substituted 8-hydroxy-[1,6]naphthyridine-7-carboxylic acid 4-fluorobenzylamide inhibitors of HIV-1 integrase and viral replication in cells

Four novel bis-(naphtho-γ-pyrones) isolated from Fusarium species as inhibitors of HIV-1 integrase

A series of 5-aminosubstituted 4-fluorobenzyl-8-hydroxy-[1,6]naphthyridine-7-carboxamide HIV-1 integrase inhibitors

Chemical and enzymatic modifications of integric acid and HIV-1 integrase inhibitory activity

Isolation and Characterization of Novel Human Immunodeficiency Virus Integrase Inhibitors from Fungal Metabolites

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