UB Paderborn / Katalog / Suche / in CDI

Sortiert nach

Einfacher Volltextzugriff von (fast) überall

Installieren Sie die LibKey Nomad-Browsererweiterung und erhalten Sie von vielen Webseiten einfachen Zugriff auf lizenzierte Volltexte oder Open Access Publikationen. Mehr erfahren...

Structure of class C GPCR metabotropic glutamate receptor 5 transmembrane domain

Nature (London), 2014-07, Vol.511 (7511), p.557-562

2014

Volltextzugriff (PDF)

Crystal structure of the GLP-1 receptor bound to a peptide agonist

Nature (London), 2017-06, Vol.546 (7657), p.254-258

2017

Volltextzugriff (PDF)

Controlling the Dissociation of Ligands from the Adenosine A2A Receptor through Modulation of Salt Bridge Strength

Journal of medicinal chemistry, 2016-07, Vol.59 (13), p.6470-6479

2016

Volltextzugriff (PDF)

Extra-helical binding site of a glucagon receptor antagonist

Nature (London), 2016-05, Vol.533 (7602), p.274-277

2016

Volltextzugriff (PDF)

Towards high throughput GPCR crystallography: In Meso soaking of Adenosine A2A Receptor crystals

Scientific reports, 2018-01, Vol.8 (1), p.1-41, Article 41

2018

Volltextzugriff (PDF)

Comparison of Orexin 1 and Orexin 2 Ligand Binding Modes Using X‑ray Crystallography and Computational Analysis

Journal of medicinal chemistry, 2020-02, Vol.63 (4), p.1528-1543

2020

Volltextzugriff (PDF)

Biophysical Fragment Screening of the β1‑Adrenergic Receptor: Identification of High Affinity Arylpiperazine Leads Using Structure-Based Drug Design

Journal of medicinal chemistry, 2013-05, Vol.56 (9), p.3446-3455

2013

Volltextzugriff (PDF)

Fragment and Structure-Based Drug Discovery for a Class C GPCR: Discovery of the mGlu5 Negative Allosteric Modulator HTL14242 (3-Chloro-5-[6-(5-fluoropyridin-2-yl)pyrimidin-4-yl]benzonitrile)

Journal of medicinal chemistry, 2015-08, Vol.58 (16), p.6653-6664

2015

Volltextzugriff (PDF)

From Disulfide- to Thioether-Linked Glycoproteins

Angewandte Chemie (International ed.), 2008-03, Vol.47 (12), p.2244-2247

2008

Volltextzugriff (PDF)

Mechanistic Insight into Enzymatic Glycosyl Transfer with Retention of Configuration through Analysis of Glycomimetic Inhibitors

Angewandte Chemie (International ed.), 2010-02, Vol.49 (7), p.1234-1237

2010

Volltextzugriff (PDF)

Structures of Human A1 and A2A Adenosine Receptors with Xanthines Reveal Determinants of Selectivity

Structure (London), 2017-08, Vol.25 (8), p.1275-1285.e4

2017

Volltextzugriff (PDF)

Intracellular allosteric antagonism of the CCR9 receptor

Nature (London), 2016-12, Vol.540 (7633), p.462-465

2016

Volltextzugriff (PDF)

Production of membrane proteins in industry: The example of GPCRs

Protein expression and purification, 2020-05, Vol.169, p.105569-105569, Article 105569

2020

Volltextzugriff (PDF)

Structure of the adenosine A(2A) receptor in complex with ZM241385 and the xanthines XAC and caffeine

Structure (London), 2011-09, Vol.19 (9), p.1283

2011

Volltextzugriff (PDF)

Precise Probing of Residue Roles by Post-Translational β,γ-C,N Aza-Michael Mutagenesis in Enzyme Active Sites

ACS central science, 2017-11, Vol.3 (11), p.1168-1173

2017

Volltextzugriff (PDF)

Preparation of purified GPCRs for structural studies

Biochemical Society transactions, 2013-02, Vol.41 (1), p.185-190

2013

Volltextzugriff (PDF)

Mechanistic evidence for a front-side, SNi-type reaction in a retaining glycosyltransferase

Nature chemical biology, 2011-08, Vol.7 (9), p.631-638

2011

Volltextzugriff (PDF)

From structure to clinic: Design of a muscarinic M1 receptor agonist with potential to treatment of Alzheimer's disease

Cell, 2021-11, Vol.184 (24), p.5886

2021

Volltextzugriff (PDF)

Structure-Based Optimization Strategies for G Protein-Coupled Receptor (GPCR) Allosteric Modulators: A Case Study from Analyses of New Metabotropic Glutamate Receptor 5 (mGlu5) X‑ray Structures

Journal of medicinal chemistry, 2019-01, Vol.62 (1), p.207-222

2019

Volltextzugriff (PDF)

Facile Conversion of Cysteine and Alkyl Cysteines to Dehydroalanine on Protein Surfaces: Versatile and Switchable Access to Functionalized Proteins

Journal of the American Chemical Society, 2008-04, Vol.130 (15), p.5052-5053

2008

Volltextzugriff (PDF)

Probing the Breadth of Macrolide Glycosyltransferases: In Vitro Remodeling of a Polyketide Antibiotic Creates Active Bacterial Uptake and Enhances Potency

Journal of the American Chemical Society, 2005-07, Vol.127 (26), p.9336-9337

2005

Volltextzugriff (PDF)

Atomic-Scale Detection of Organic Molecules Coupled to Single-Walled Carbon Nanotubes

Journal of the American Chemical Society, 2007-09, Vol.129 (36), p.10966-10967

2007

Volltextzugriff (PDF)

Functional Characterization of a Novel ArgA from Mycobacterium tuberculosis

Journal of Bacteriology, 2005-05, Vol.187 (9), p.3039-3044

2005

Volltextzugriff (PDF)

Functional Annotation and Kinetic Characterization of PhnO from Salmonella enterica

Biochemistry (Easton), 2006-03, Vol.45 (9), p.3033-3039

2006

Volltextzugriff (PDF)

Flexible enzymatic and chemo-enzymatic approaches to a broad range of uridine-diphospho-sugars

Chemical communications (Cambridge, England), 2004-12 (23), p.2706-2707

2004

Volltextzugriff (PDF)

1 – 25 von 71

Suche als RSS-Feed

Suchergebnisse filtern

Filter anzeigen

Nur zeigen

Geprüft (Peer-Review)
(66)
Mit Volltextzugriff
(58)

Publikationsform

Artikel
(70)
Buchkapitel
(1)

Sprache

Englisch
(70)
Deutsch
(2)

Erscheinungsjahr

n.n

Thema

Science & Technology
(34)
Models, Molecular
(19)
Life Sciences & Biomedicine
(17)
Chemistry
(16)
Humans
(15)
Physical Sciences
(15)
Biochemistry & Molecular Biology
(12)
Ligands
(11)
Binding Sites
(10)
Chemistry, Multidisciplinary
(10)
Crystallography, X-Ray
(10)
Hek293 Cells
(8)
Kinetics
(8)
Drug Design
(7)
Molecular Structure
(7)
Receptor, Adenosine A2a - Chemistry
(7)
Receptor, Adenosine A2a - Metabolism
(7)
Substrate Specificity
(7)
631/535/1266
(6)
Animals
(6)

15 weitere anzeigen...

Weniger anzeigen...

Zeitschrift / Serie

5 weitere anzeigen...

Weniger anzeigen...

Neu hinzugefügt

... seit 30 Tagen
(1)

Menü

Weitere Dienste

Einstellungen

Structure of class C GPCR metabotropic glutamate receptor 5 transmembrane domain

Crystal structure of the GLP-1 receptor bound to a peptide agonist

Controlling the Dissociation of Ligands from the Adenosine A2A Receptor through Modulation of Salt Bridge Strength

Extra-helical binding site of a glucagon receptor antagonist

Towards high throughput GPCR crystallography: In Meso soaking of Adenosine A2A Receptor crystals

Comparison of Orexin 1 and Orexin 2 Ligand Binding Modes Using X‑ray Crystallography and Computational Analysis

Biophysical Fragment Screening of the β1‑Adrenergic Receptor: Identification of High Affinity Arylpiperazine Leads Using Structure-Based Drug Design

Fragment and Structure-Based Drug Discovery for a Class C GPCR: Discovery of the mGlu5 Negative Allosteric Modulator HTL14242 (3-Chloro-5-[6-(5-fluoropyridin-2-yl)pyrimidin-4-yl]benzonitrile)

From Disulfide- to Thioether-Linked Glycoproteins

Mechanistic Insight into Enzymatic Glycosyl Transfer with Retention of Configuration through Analysis of Glycomimetic Inhibitors

Structures of Human A1 and A2A Adenosine Receptors with Xanthines Reveal Determinants of Selectivity

Intracellular allosteric antagonism of the CCR9 receptor

Production of membrane proteins in industry: The example of GPCRs

Structure of the adenosine A(2A) receptor in complex with ZM241385 and the xanthines XAC and caffeine

Precise Probing of Residue Roles by Post-Translational β,γ-C,N Aza-Michael Mutagenesis in Enzyme Active Sites

Preparation of purified GPCRs for structural studies

Mechanistic evidence for a front-side, SNi-type reaction in a retaining glycosyltransferase

From structure to clinic: Design of a muscarinic M1 receptor agonist with potential to treatment of Alzheimer's disease

Structure-Based Optimization Strategies for G Protein-Coupled Receptor (GPCR) Allosteric Modulators: A Case Study from Analyses of New Metabotropic Glutamate Receptor 5 (mGlu5) X‑ray Structures

Facile Conversion of Cysteine and Alkyl Cysteines to Dehydroalanine on Protein Surfaces: Versatile and Switchable Access to Functionalized Proteins

Probing the Breadth of Macrolide Glycosyltransferases: In Vitro Remodeling of a Polyketide Antibiotic Creates Active Bacterial Uptake and Enhances Potency

Atomic-Scale Detection of Organic Molecules Coupled to Single-Walled Carbon Nanotubes

Functional Characterization of a Novel ArgA from Mycobacterium tuberculosis

Functional Annotation and Kinetic Characterization of PhnO from Salmonella enterica

Flexible enzymatic and chemo-enzymatic approaches to a broad range of uridine-diphospho-sugars

Suchergebnisse filtern