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Identification and Biological Evaluation of 4-(3-Trifluoromethylpyridin-2-yl)piperazine-1-carboxylic Acid (5-Trifluoromethylpyridin-2-yl)amide, a High Affinity TRPV1 (VR1) Vanilloid Receptor Antagonist

Journal of medicinal chemistry, 2005-03, Vol.48 (6), p.1857-1872

2005

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Population Pharmacokinetic-Pharmacodynamic Model of Oxfendazole in Healthy Adults in a Multiple Ascending Dose and Food Effect Study and Target Attainment Analysis

Antimicrobial agents and chemotherapy, 2022-01, Vol.66 (1), p.e0143221

2022

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JNJ-20788560 [9-(8-azabicyclo[3.2.1]oct-3-ylidene)-9H-xanthene-3-carboxylic acid diethylamide], a selective delta opioid receptor agonist, is a potent and efficacious antihyperalgesic agent that does not produce respiratory depression, pharmacologic tolerance, or physical dependence

The Journal of pharmacology and experimental therapeutics, 2009-04, Vol.329 (1), p.241

2009

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Oxfendazole: a promising agent for the treatment and control of helminth infections in humans

Expert review of anti-infective therapy, 2019-01, Vol.17 (1), p.51-56

2019

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Tramadol and several anticonvulsants synergize in attenuating nerve injury-induced allodynia

Pain (Amsterdam), 2008-02, Vol.134 (3), p.254-262

2008

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Pharmacokinetics, Safety, and Tolerability of Oxfendazole in Healthy Adults in an Open-Label Phase 1 Multiple Ascending Dose and Food Effect Study

Antimicrobial agents and chemotherapy, 2020-10, Vol.64 (11)

2020

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Preclinical safety assessment of JNJ-10450232 (NTM-006), a structural analog of acetaminophen, that does not cause hepatotoxicity at supratherapeutic doses

Regulatory toxicology and pharmacology, 2023-01, p.105334, Article 105334

2023

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Pharmacokinetics, Safety, and Tolerability of Oxfendazole in Healthy Volunteers: a Randomized, Placebo-Controlled First-in-Human Single-Dose Escalation Study

Antimicrobial agents and chemotherapy, 2019-04, Vol.63 (4)

2019

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Diabetogenic Effect of a Series of Tricyclic Delta Opioid Agonists Structurally Related to Cyproheptadine

Toxicological sciences, 2010-10, Vol.117 (2), p.493-504

2010

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α2 Adrenoceptor Agonists as Potential Analgesic Agents. 3. Imidazolylmethylthiophenes

Journal of medicinal chemistry, 2001-03, Vol.44 (6), p.863-872

2001

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Preclinical Studies on the Pharmacokinetics, Safety, and Toxicology of Oxfendazole: Toward First in Human Studies

International journal of toxicology, 2015-03, Vol.34 (2), p.129-137

2015

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Dynamic mass redistribution as a means to measure and differentiate signaling via opioid and cannabinoid receptors

Assay and drug development technologies, 2011-08, Vol.9 (4), p.362-372

2011

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Heteroaryl β-tetralin ureas as novel antagonists of human TRPV1

Bioorganic & medicinal chemistry, 2007-11, Vol.17 (22), p.6160-6163

2007

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Ex vivo delta opioid receptor autoradiography: CNS receptor occupancy of two novel compounds over their antihyperalgesic dose range

Pharmacology, biochemistry and behavior, 2010-08, Vol.96 (2), p.130-135

2010

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N-Pyridin-3-yl- and N-quinolin-3-yl-benzamides: Modulators of Human Vanilloid Receptor 1 (TRPV1)

Bioorganic & medicinal chemistry letters, 2008-04, Vol.18 (8), p.2730-2734

2008

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High-throughput screening for N-type calcium channel blockers using a scintillation proximity assay

Journal of biomolecular screening, 2006-09, Vol.11 (6), p.672-677

2006

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Parallel methods for the preparation and SAR exploration of N-ethyl-4-[(8-alkyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-aryl-methyl]-benzamides, powerful mu and delta opioid agonists

Bioorganic & medicinal chemistry letters, 2004-11, Vol.14 (22), p.5493-5498

2004

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N, N-Dialkyl-4-[(8-azabicyclo[3.2.1]-oct-3-ylidene)phenylmethyl]-benzamides, potent, selective δ opioid agonists

Bioorganic & medicinal chemistry letters, 2004-05, Vol.14 (9), p.2109-2112

2004

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Design and synthesis of novel pyrrolidine-containing bradykinin antagonists

Bioorganic & medicinal chemistry letters, 2003-06, Vol.13 (11), p.1879-1882

2003

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Lack of binding of acetaminophen to 5-HT receptor or uptake sites (or eleven other binding/uptake assays)

Life sciences (1973), 1996, Vol.59 (2), p.PL37-PL40

1996

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N-Alkyl-4-[(8-azabicyclo[3.2.1]-oct-3-ylidene)phenylmethyl]-benzamides, μ and δ opioid agonists: a μ address

Bioorganic & medicinal chemistry letters, 2004-05, Vol.14 (9), p.2113-2116

2004

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Functional studies of bradykinin receptors in Chinese hamster ovary cells stably expressing the human B2 bradykinin receptor

International immunopharmacology, 2001-05, Vol.1 (5), p.955-965

2001

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Molecular cloning and characterization of the human voltage-gated calcium channel alpha(2)delta-4 subunit

Molecular pharmacology, 2002-09, Vol.62 (3), p.485-496

2002

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Synthesis and structure–Activity relationships of aroylpyrrole alkylamide bradykinin (B 2) antagonists

Bioorganic & medicinal chemistry letters, 2003-04, Vol.13 (7), p.1341-1344

2003

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α2 Adrenoceptor Agonists as Potential Analgesic Agents. 1. (Imidazolylmethyl)oxazoles and -thiazoles

Journal of medicinal chemistry, 1999-12, Vol.42 (25), p.5064-5071

1999

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Identification and Biological Evaluation of 4-(3-Trifluoromethylpyridin-2-yl)piperazine-1-carboxylic Acid (5-Trifluoromethylpyridin-2-yl)amide, a High Affinity TRPV1 (VR1) Vanilloid Receptor Antagonist

Population Pharmacokinetic-Pharmacodynamic Model of Oxfendazole in Healthy Adults in a Multiple Ascending Dose and Food Effect Study and Target Attainment Analysis

JNJ-20788560 [9-(8-azabicyclo[3.2.1]oct-3-ylidene)-9H-xanthene-3-carboxylic acid diethylamide], a selective delta opioid receptor agonist, is a potent and efficacious antihyperalgesic agent that does not produce respiratory depression, pharmacologic tolerance, or physical dependence

Oxfendazole: a promising agent for the treatment and control of helminth infections in humans

Tramadol and several anticonvulsants synergize in attenuating nerve injury-induced allodynia

Pharmacokinetics, Safety, and Tolerability of Oxfendazole in Healthy Adults in an Open-Label Phase 1 Multiple Ascending Dose and Food Effect Study

Preclinical safety assessment of JNJ-10450232 (NTM-006), a structural analog of acetaminophen, that does not cause hepatotoxicity at supratherapeutic doses

Pharmacokinetics, Safety, and Tolerability of Oxfendazole in Healthy Volunteers: a Randomized, Placebo-Controlled First-in-Human Single-Dose Escalation Study

Diabetogenic Effect of a Series of Tricyclic Delta Opioid Agonists Structurally Related to Cyproheptadine

α2 Adrenoceptor Agonists as Potential Analgesic Agents. 3. Imidazolylmethylthiophenes

Preclinical Studies on the Pharmacokinetics, Safety, and Toxicology of Oxfendazole: Toward First in Human Studies

Dynamic mass redistribution as a means to measure and differentiate signaling via opioid and cannabinoid receptors

Heteroaryl β-tetralin ureas as novel antagonists of human TRPV1

Ex vivo delta opioid receptor autoradiography: CNS receptor occupancy of two novel compounds over their antihyperalgesic dose range

N-Pyridin-3-yl- and N-quinolin-3-yl-benzamides: Modulators of Human Vanilloid Receptor 1 (TRPV1)

High-throughput screening for N-type calcium channel blockers using a scintillation proximity assay

Parallel methods for the preparation and SAR exploration of N-ethyl-4-[(8-alkyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-aryl-methyl]-benzamides, powerful mu and delta opioid agonists

N, N-Dialkyl-4-[(8-azabicyclo[3.2.1]-oct-3-ylidene)phenylmethyl]-benzamides, potent, selective δ opioid agonists

Design and synthesis of novel pyrrolidine-containing bradykinin antagonists

Lack of binding of acetaminophen to 5-HT receptor or uptake sites (or eleven other binding/uptake assays)

N-Alkyl-4-[(8-azabicyclo[3.2.1]-oct-3-ylidene)phenylmethyl]-benzamides, μ and δ opioid agonists: a μ address

Functional studies of bradykinin receptors in Chinese hamster ovary cells stably expressing the human B2 bradykinin receptor

Molecular cloning and characterization of the human voltage-gated calcium channel alpha(2)delta-4 subunit

Synthesis and structure–Activity relationships of aroylpyrrole alkylamide bradykinin (B 2) antagonists

α2 Adrenoceptor Agonists as Potential Analgesic Agents. 1. (Imidazolylmethyl)oxazoles and -thiazoles

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