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A Virtual Screening Approach to Finding Novel and Potent Antagonists at the Melanin-Concentrating Hormone 1 Receptor

Journal of medicinal chemistry, 2004-07, Vol.47 (16), p.3962-3971

2004

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Identification of Imidazo-Pyrrolopyridines as Novel and Potent JAK1 Inhibitors

Journal of medicinal chemistry, 2012-06, Vol.55 (12), p.5901-5921

2012

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Quinazolinethiones and quinazolinediones, novel inhibitors of inosine monophosphate dehydrogenase: synthesis and initial structure–activity relationships

Bioorganic & medicinal chemistry letters, 2005-02, Vol.15 (3), p.751-754

2005

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Update on the therapeutic potential of PDE4 inhibitors

Expert opinion on investigational drugs, 2002-01, Vol.11 (1), p.1-13

2002

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Novel triazolo-pyrrolopyridines as inhibitors of Janus kinase 1

Bioorganic & medicinal chemistry letters, 2013-06, Vol.23 (12), p.3592-3598

2013

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1H-Pyrazolo[3,4-g]hexahydro-isoquinolines as selective glucocorticoid receptor antagonists with high functional activity

Bioorganic & medicinal chemistry, 2008-02, Vol.18 (4), p.1312-1317

2008

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Novel 5,6-dihydropyrazolo-[3,4-E][1,4]diazepin-4 (1H)-one derivatives for the treatment of asthma and chronic obstructive pulmonary disease: AstraZeneca: WO2007040435

Expert opinion on therapeutic patents, 2007-09, Vol.17 (9), p.1183-1189

Dyke, Hazel J

2007

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Identification and hit-to-lead exploration of a novel series of histamine H4 receptor inverse agonists

Bioorganic & medicinal chemistry letters, 2010-04, Vol.20 (8), p.2516-2519

2010

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Novel 5,6-dihydropyrazolo-[3,4-E][1,4]diazepin-4 (1H)-one derivatives for the treatment of asthma and chronic obstructive pulmonary disease

Expert opinion on therapeutic patents, 2007-09, Vol.17 (9), p.1183-1189

Dyke, Hazel J

2007

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Increasing Selectivity of CC Chemokine Receptor 8 Antagonists by Engineering Nondesolvation Related Interactions with the Intended and Off-Target Binding Sites

Journal of medicinal chemistry, 2009-12, Vol.52 (23), p.7706-7723

2009

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Synthesis and profile of SCH351591, a novel PDE4 inhibitor

Bioorganic & medicinal chemistry letters, 2002-06, Vol.12 (12), p.1621-1623

2002

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Histone deacetylase inhibitors: an analysis of recent patenting activity

Expert opinion on therapeutic patents, 2007-07, Vol.17 (7), p.745-765

2007

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Novel 7-methoxy-6-oxazol-5-yl-2,3-dihydro-1H-quinazolin-4-ones as IMPDH inhibitors

Bioorganic & medicinal chemistry letters, 2005-12, Vol.15 (23), p.5335-5339

2005

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Identification and optimisation of a series of substituted 5-(1 H-pyrazol-3-yl)-thiophene-2-hydroxamic acids as potent histone deacetylase (HDAC) inhibitors

Bioorganic & medicinal chemistry letters, 2007-01, Vol.17 (2), p.370-375

2007

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Quinazoline and benzimidazole MCH-1R antagonists

Bioorganic & medicinal chemistry letters, 2007-03, Vol.17 (5), p.1403-1407

2007

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Discovery and optimization of novel, non-steroidal glucocorticoid receptor modulators

Bioorganic & medicinal chemistry letters, 2007-09, Vol.17 (17), p.4901-4905

2007

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Structure–activity relationships of a novel series of melanin-concentrating hormone (MCH) receptor antagonists

Bioorganic & medicinal chemistry letters, 2004-08, Vol.14 (15), p.4099-4102

2004

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Identification and optimisation of a series of substituted 5-pyridin-2-yl-thiophene-2-hydroxamic acids as potent histone deacetylase (HDAC) inhibitors

Bioorganic & medicinal chemistry letters, 2007-01, Vol.17 (2), p.363-369

2007

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2-Benzenesulfonyl-8a-benzyl-hexahydro-2H-isoquinolin-6-ones as selective glucocorticoid receptor antagonists

Bioorganic & medicinal chemistry letters, 2007-10, Vol.17 (20), p.5704-5708

2007

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Synthesis and structure–activity relationships of guanine analogues as phosphodiesterase 7 (PDE7) inhibitors

Bioorganic & medicinal chemistry letters, 2001-04, Vol.11 (8), p.1081-1083

2001

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8-Methoxyquinolines as PDE4 inhibitors

Bioorganic & medicinal chemistry letters, 2002-06, Vol.12 (12), p.1617-1619

2002

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7-Methoxyfuro[2,3- c]pyridine-4-carboxamides as PDE4 Inhibitors: A Potential Treatment for Asthma

Bioorganic & medicinal chemistry letters, 2002-02, Vol.12 (3), p.509-512

2002

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8-Methoxyquinoline-5-carboxamides as PDE4 inhibitors: a potential treatment for asthma

Bioorganic & medicinal chemistry letters, 2002-06, Vol.12 (12), p.1613-1615

2002

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7-Methoxybenzofuran-4-carboxamides as PDE 4 inhibitors: a potential treatment for asthma

Bioorganic & medicinal chemistry letters, 2000-09, Vol.10 (18), p.2137-2140

2000

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Aryl sulfonamides as selective PDE4 inhibitors

Bioorganic & medicinal chemistry letters, 1998-10, Vol.8 (19), p.2635-2640

1998

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A Virtual Screening Approach to Finding Novel and Potent Antagonists at the Melanin-Concentrating Hormone 1 Receptor

Identification of Imidazo-Pyrrolopyridines as Novel and Potent JAK1 Inhibitors

Quinazolinethiones and quinazolinediones, novel inhibitors of inosine monophosphate dehydrogenase: synthesis and initial structure–activity relationships

Update on the therapeutic potential of PDE4 inhibitors

Novel triazolo-pyrrolopyridines as inhibitors of Janus kinase 1

1H-Pyrazolo[3,4-g]hexahydro-isoquinolines as selective glucocorticoid receptor antagonists with high functional activity

Novel 5,6-dihydropyrazolo-[3,4-E][1,4]diazepin-4 (1H)-one derivatives for the treatment of asthma and chronic obstructive pulmonary disease: AstraZeneca: WO2007040435

Identification and hit-to-lead exploration of a novel series of histamine H4 receptor inverse agonists

Novel 5,6-dihydropyrazolo-[3,4-E][1,4]diazepin-4 (1H)-one derivatives for the treatment of asthma and chronic obstructive pulmonary disease

Increasing Selectivity of CC Chemokine Receptor 8 Antagonists by Engineering Nondesolvation Related Interactions with the Intended and Off-Target Binding Sites

Synthesis and profile of SCH351591, a novel PDE4 inhibitor

Histone deacetylase inhibitors: an analysis of recent patenting activity

Novel 7-methoxy-6-oxazol-5-yl-2,3-dihydro-1H-quinazolin-4-ones as IMPDH inhibitors

Identification and optimisation of a series of substituted 5-(1 H-pyrazol-3-yl)-thiophene-2-hydroxamic acids as potent histone deacetylase (HDAC) inhibitors

Quinazoline and benzimidazole MCH-1R antagonists

Discovery and optimization of novel, non-steroidal glucocorticoid receptor modulators

Structure–activity relationships of a novel series of melanin-concentrating hormone (MCH) receptor antagonists

Identification and optimisation of a series of substituted 5-pyridin-2-yl-thiophene-2-hydroxamic acids as potent histone deacetylase (HDAC) inhibitors

2-Benzenesulfonyl-8a-benzyl-hexahydro-2H-isoquinolin-6-ones as selective glucocorticoid receptor antagonists

Synthesis and structure–activity relationships of guanine analogues as phosphodiesterase 7 (PDE7) inhibitors

8-Methoxyquinolines as PDE4 inhibitors

7-Methoxyfuro[2,3- c]pyridine-4-carboxamides as PDE4 Inhibitors: A Potential Treatment for Asthma

8-Methoxyquinoline-5-carboxamides as PDE4 inhibitors: a potential treatment for asthma

7-Methoxybenzofuran-4-carboxamides as PDE 4 inhibitors: a potential treatment for asthma

Aryl sulfonamides as selective PDE4 inhibitors

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