UB Paderborn / Katalog / Suche / in CDI

1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors

Journal of medicinal chemistry, 2020-03, Vol.63 (5), p.2470-2488

2020

Volltextzugriff (PDF)

Design, synthesis and evaluation of N-substituted saccharin derivatives as selective inhibitors of tumor-associated carbonic anhydrase XII

Bioorganic & medicinal chemistry, 2014-03, Vol.22 (6), p.1821-1831

2014

Volltextzugriff (PDF)

Selective inhibition of human carbonic anhydrases by novel amide derivatives of probenecid: Synthesis, biological evaluation and molecular modelling studies

Bioorganic & medicinal chemistry, 2014-08, Vol.22 (15), p.3982-3988

2014

Volltextzugriff (PDF)

Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents

European journal of medicinal chemistry, 2011-01, Vol.46 (1), p.378-382

2011

Volltextzugriff (PDF)

New amide derivatives of Probenecid as selective inhibitors of carbonic anhydrase IX and XII: Biological evaluation and molecular modelling studies

Bioorganic & medicinal chemistry, 2015-07, Vol.23 (13), p.2975-2981

2015

Volltextzugriff (PDF)

Salen and tetrahydrosalen derivatives act as effective inhibitors of the tumor-associated carbonic anhydrase XII—A new scaffold for designing isoform-selective inhibitors

Bioorganic & medicinal chemistry letters, 2013-12, Vol.23 (24), p.6759-6763

2013

Volltextzugriff (PDF)

Exploring 4-substituted-2-thiazolylhydrazones from 2-, 3-, and 4-acetylpyridine as selective and reversible hMAO-B inhibitors

European journal of medicinal chemistry, 2013-08, Vol.66, p.221-227

2013

Volltextzugriff (PDF)

(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies

Journal of enzyme inhibition and medicinal chemistry, 2015-11, Vol.30 (6), p.908-919

2015

Volltextzugriff (PDF)

Identification of the stereochemical requirements in the 4-aryl-2-cycloalkylidenhydrazinylthiazole scaffold for the design of selective human monoamine oxidase B inhibitors

Bioorganic & medicinal chemistry, 2014-05, Vol.22 (10), p.2887-2895

2014

Volltextzugriff (PDF)

Selective MAO-B inhibitors: a lesson from natural products

Molecular diversity, 2014-02, Vol.18 (1), p.219-243

2014

Volltextzugriff (PDF)

4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis

Journal of enzyme inhibition and medicinal chemistry, 2019-01, Vol.34 (1), p.597-612

2019

Volltextzugriff (PDF)

Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms

Journal of enzyme inhibition and medicinal chemistry, 2017-12, Vol.32 (1), p.51-59

2017

Volltextzugriff (PDF)

Discovery and optimization of pyrazoline derivatives as promising monoamine oxidase inhibitors

Current topics in medicinal chemistry, 2012-10, Vol.12 (20), p.2240

2012

Volltextzugriff (PDF)

A Combined Crystallographic and Theoretical Study Explains the Capability of Carboxylic Acids to Adopt Multiple Binding Modes in the Active Site of Carbonic Anhydrases

Chemistry : a European journal, 2016-01, Vol.22 (1), p.97-100

2016

Volltextzugriff (PDF)

Patent-related survey on new monoamine oxidase inhibitors and their therapeutic potential

Expert opinion on therapeutic patents, 2012-07, Vol.22 (7), p.759-801

2012

Volltextzugriff (PDF)

Synthesis, biological evaluation and quantitative structure-active relationships of 1,3-thiazolidin-4-one derivatives. A promising chemical scaffold endowed with high antifungal potency and low cytotoxicity

European journal of medicinal chemistry, 2017-11, Vol.140, p.274-292

2017

Volltextzugriff (PDF)

Cyclic tertiary sulfamates: Selective inhibition of the tumor-associated carbonic anhydrases IX and XII by N- and O-substituted acesulfame derivatives

European journal of medicinal chemistry, 2014-09, Vol.84, p.240-246

2014

Volltextzugriff (PDF)

Recent advances in the development of selective human MAO-B inhibitors: (Hetero)arylidene-(4-substituted-thiazol-2-yl)hydrazines

European journal of medicinal chemistry, 2012-12, Vol.58, p.405-417

2012

Volltextzugriff (PDF)

Design, synthesis and biological characterization of thiazolidin-4-one derivatives as promising inhibitors of Toxoplasma gondii

European journal of medicinal chemistry, 2014-10, Vol.86, p.17-30

2014

Volltextzugriff (PDF)

Evaluation of a large library of (thiazol-2-yl)hydrazones and analogues as histone acetyltransferase inhibitors: Enzyme and cellular studies

European journal of medicinal chemistry, 2014-06, Vol.80, p.569-578

2014

Volltextzugriff (PDF)

Synthesis, anti-Candida activity, and cytotoxicity of new (4-(4-iodophenyl)thiazol-2-yl)hydrazine derivatives

European journal of medicinal chemistry, 2012-07, Vol.53, p.246-253

2012

Volltextzugriff (PDF)

Synthesis and pharmacological screening of a large library of 1,3,4-thiadiazolines as innovative therapeutic tools for the treatment of prostate cancer and melanoma

European journal of medicinal chemistry, 2015-11, Vol.105, p.245-262

2015

Volltextzugriff (PDF)

An Activity‐Based Probe Targeting Non‐Catalytic, Highly Conserved Amino Acid Residues within Bromodomains

Angewandte Chemie (International ed.), 2019-01, Vol.58 (4), p.1007-1012

International ed. in English, 2019

Volltextzugriff (PDF)

Microwave and Ultrasound-Assisted Synthesis of Thiosemicarbazones and Their Corresponding (4,5-Substituted-thiazol-2-yl)hydrazines

Journal of heterocyclic chemistry, 2014-11, Vol.51 (6), p.1856-1861

2014

Volltextzugriff (PDF)

Conventional and Microwave-Assisted Synthesis of Benzimidazole Derivatives and Their In Vitro Inhibition of Human Cyclooxygenase

Journal of heterocyclic chemistry, 2012-09, Vol.49 (5), p.1187-1195

2012

Volltextzugriff (PDF)

Menü

Weitere Dienste

Einstellungen

1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors

Design, synthesis and evaluation of N-substituted saccharin derivatives as selective inhibitors of tumor-associated carbonic anhydrase XII

Selective inhibition of human carbonic anhydrases by novel amide derivatives of probenecid: Synthesis, biological evaluation and molecular modelling studies

Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents

New amide derivatives of Probenecid as selective inhibitors of carbonic anhydrase IX and XII: Biological evaluation and molecular modelling studies

Salen and tetrahydrosalen derivatives act as effective inhibitors of the tumor-associated carbonic anhydrase XII—A new scaffold for designing isoform-selective inhibitors

Exploring 4-substituted-2-thiazolylhydrazones from 2-, 3-, and 4-acetylpyridine as selective and reversible hMAO-B inhibitors

(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies

Identification of the stereochemical requirements in the 4-aryl-2-cycloalkylidenhydrazinylthiazole scaffold for the design of selective human monoamine oxidase B inhibitors

Selective MAO-B inhibitors: a lesson from natural products

4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis

Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms

Discovery and optimization of pyrazoline derivatives as promising monoamine oxidase inhibitors

A Combined Crystallographic and Theoretical Study Explains the Capability of Carboxylic Acids to Adopt Multiple Binding Modes in the Active Site of Carbonic Anhydrases

Patent-related survey on new monoamine oxidase inhibitors and their therapeutic potential

Synthesis, biological evaluation and quantitative structure-active relationships of 1,3-thiazolidin-4-one derivatives. A promising chemical scaffold endowed with high antifungal potency and low cytotoxicity

Cyclic tertiary sulfamates: Selective inhibition of the tumor-associated carbonic anhydrases IX and XII by N- and O-substituted acesulfame derivatives

Recent advances in the development of selective human MAO-B inhibitors: (Hetero)arylidene-(4-substituted-thiazol-2-yl)hydrazines

Design, synthesis and biological characterization of thiazolidin-4-one derivatives as promising inhibitors of Toxoplasma gondii

Evaluation of a large library of (thiazol-2-yl)hydrazones and analogues as histone acetyltransferase inhibitors: Enzyme and cellular studies

Synthesis, anti-Candida activity, and cytotoxicity of new (4-(4-iodophenyl)thiazol-2-yl)hydrazine derivatives

Synthesis and pharmacological screening of a large library of 1,3,4-thiadiazolines as innovative therapeutic tools for the treatment of prostate cancer and melanoma

An Activity‐Based Probe Targeting Non‐Catalytic, Highly Conserved Amino Acid Residues within Bromodomains

Microwave and Ultrasound-Assisted Synthesis of Thiosemicarbazones and Their Corresponding (4,5-Substituted-thiazol-2-yl)hydrazines

Conventional and Microwave-Assisted Synthesis of Benzimidazole Derivatives and Their In Vitro Inhibition of Human Cyclooxygenase

Suchergebnisse filtern