UB Paderborn / Katalog / Suche / in CDI

Identification of a Series of Tricyclic Natural Products as Potent Broad-Spectrum Inhibitors of Metallo-β-Lactamases

Antimicrobial Agents and Chemotherapy, 2002-06, Vol.46 (6), p.1880-1886

2002

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Crystal Structure of the IMP-1 Metallo β-Lactamase from Pseudomonas aeruginosa and Its Complex with a Mercaptocarboxylate Inhibitor: Binding Determinants of a Potent, Broad-Spectrum Inhibitor

Biochemistry (Easton), 2000-04, Vol.39 (15), p.4288-4298

2000

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Anti-tumor Activity of the Type I PRMT Inhibitor, GSK3368715, Synergizes with PRMT5 Inhibition through MTAP Loss

Cancer cell, 2019-07, Vol.36 (1), p.100-114.e25

2019

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Structural Basis for Chk1 Inhibition by UCN-01

The Journal of biological chemistry, 2002-11, Vol.277 (48), p.46609-46615

2002

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Exploration of the P1 residue in 3CL protease inhibitors leading to the discovery of a 2-tetrahydrofuran P1 replacement

Bioorganic & medicinal chemistry, 2024-02, Vol.100, p.117618-117618, Article 117618

2024

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Long-Range Inhibitor-Induced Conformational Regulation of Human IRE1α Endoribonuclease Activity

Molecular pharmacology, 2015-12, Vol.88 (6), p.1011-1023

2015

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3-(1,1-Dioxo-2H-(1,2,4)-benzothiadiazin-3-yl)-4-hydroxy-2(1H)-quinolinones, Potent Inhibitors of Hepatitis C Virus RNA-Dependent RNA Polymerase

Journal of medicinal chemistry, 2006-02, Vol.49 (3), p.971-983

2006

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Crystal structure of the wide-spectrum binuclear zinc β-lactamase from Bacteroides fragilis

Structure (London), 1996-07, Vol.4 (7), p.823-836

1996

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Substituted benzothiadizine inhibitors of Hepatitis C virus polymerase

Bioorganic & medicinal chemistry letters, 2009-08, Vol.19 (15), p.4350-4353

2009

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Aminofurazans as potent inhibitors of AKT kinase

Bioorganic & medicinal chemistry letters, 2009-03, Vol.19 (5), p.1508-1511

2009

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Discovery of 5-pyrrolopyridinyl-2-thiophenecarboxamides as potent AKT kinase inhibitors

Bioorganic & medicinal chemistry letters, 2009-04, Vol.19 (8), p.2244-2248

2009

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2,3,5-Trisubstituted pyridines as selective AKT inhibitors—Part I: Substitution at 2-position of the core pyridine for ROCK1 selectivity

Bioorganic & medicinal chemistry letters, 2010-01, Vol.20 (2), p.673-678

2010

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Annexin V forms calcium-dependent trimeric units on phospholipid vesicles

FEBS letters, 1992-12, Vol.314 (2), p.159-162

1992

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Structure-based combinatorial library design: discovery of non-peptidic inhibitors of caspases 3 and 8

Journal of computer-aided molecular design, 2001-12, Vol.15 (12), p.1105-1117

2001

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Potent and Selective Nonpeptide Inhibitors of Caspases 3 and 7 Inhibit Apoptosis and Maintain Cell Functionality

The Journal of biological chemistry, 2000-05, Vol.275 (21), p.16007-16014

2000

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Crystal structures of the cadmium‐ and mercury‐substituted metallo‐β‐lactamase from Bacteroides fragilis

Protein science, 1997-12, Vol.6 (12), p.2671-2676

1997

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El microscopio bajo mis manos: breve historia, funcionamiento y aplicaciones de la microscopia

Ciencia ergo sum, 2023-01, Vol.30 (3), p.1-17

2023

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Secuelas oftalmológicas secundarias a Síndrome de Stevens - Johnson

MedUNAB, 2019-03, Vol.21 (2), p.8-11

2019

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Perfil bioquímico sanguíneo hepático de vicuñas criadas en cautiverio en Lima

Revista de investigaciones veterinarias del Perú, 2013-01, Vol.24 (1), p.38-45

2013

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Sangrado oscuro y anemia crónica severa: discusión sobre dos causas gastrointestinales subvaloradas en Colombia

Universitas médica, 2013-12, Vol.55 (2), p.229-234

2013

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Caracterización nutricional y de producción de biomasa de Sambucus peruviana, Sambucus nigra y Morus alba en un banco forrajero

Ciencia en desarrollo, 2019-07, Vol.10 (2), p.23-32

2019

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Identification of a Series of Tricyclic Natural Products as Potent Broad-Spectrum Inhibitors of Metallo-β-Lactamases

Crystal Structure of the IMP-1 Metallo β-Lactamase from Pseudomonas aeruginosa and Its Complex with a Mercaptocarboxylate Inhibitor: Binding Determinants of a Potent, Broad-Spectrum Inhibitor

Anti-tumor Activity of the Type I PRMT Inhibitor, GSK3368715, Synergizes with PRMT5 Inhibition through MTAP Loss

Structural Basis for Chk1 Inhibition by UCN-01

A DNA Hypomethylation Signature Predicts Antitumor Activity of LSD1 Inhibitors in SCLC

Exploration of the P1 residue in 3CL protease inhibitors leading to the discovery of a 2-tetrahydrofuran P1 replacement

Long-Range Inhibitor-Induced Conformational Regulation of Human IRE1α Endoribonuclease Activity

Identification of 4-(2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-{[(3S)-3-piperidinylmethyl]oxy}-1H-imidazo[4,5-c]pyridin-4-yl)-2-methyl-3-butyn-2-ol (GSK690693), a Novel Inhibitor of AKT Kinase

3-(1,1-Dioxo-2H-(1,2,4)-benzothiadiazin-3-yl)-4-hydroxy-2(1H)-quinolinones, Potent Inhibitors of Hepatitis C Virus RNA-Dependent RNA Polymerase

Crystal structure of the wide-spectrum binuclear zinc β-lactamase from Bacteroides fragilis

Substituted benzothiadizine inhibitors of Hepatitis C virus polymerase

Aminofurazans as potent inhibitors of AKT kinase

Discovery of 5-pyrrolopyridinyl-2-thiophenecarboxamides as potent AKT kinase inhibitors

2,3,5-Trisubstituted pyridines as selective AKT inhibitors—Part I: Substitution at 2-position of the core pyridine for ROCK1 selectivity

Annexin V forms calcium-dependent trimeric units on phospholipid vesicles

Structure-based combinatorial library design: discovery of non-peptidic inhibitors of caspases 3 and 8

Potent and Selective Nonpeptide Inhibitors of Caspases 3 and 7 Inhibit Apoptosis and Maintain Cell Functionality

Crystal structures of the cadmium‐ and mercury‐substituted metallo‐β‐lactamase from Bacteroides fragilis

Identification of 4-(2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-{[(3 S )-3-piperidinylmethyl]oxy}-1 H -imidazo[4,5- c ]pyridin-4-yl)-2-methyl-3-butyn-2-ol (GSK690693), a Novel Inhibitor of AKT Kinase

Identification of 4-2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-([(3S)-3-piperidinylmethyl]oxy}-1H-imidazo[4,5-c]pyridin-4-yl)-2-methyl-3-butyn-2-ol (GSK690693), a Novel Inhibitor of AKT Kinase

El microscopio bajo mis manos: breve historia, funcionamiento y aplicaciones de la microscopia

Secuelas oftalmológicas secundarias a Síndrome de Stevens - Johnson

Perfil bioquímico sanguíneo hepático de vicuñas criadas en cautiverio en Lima

Sangrado oscuro y anemia crónica severa: discusión sobre dos causas gastrointestinales subvaloradas en Colombia

Caracterización nutricional y de producción de biomasa de Sambucus peruviana, Sambucus nigra y Morus alba en un banco forrajero

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