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Synthesis and Biological Evaluation of 2-Indolyloxazolines as a New Class of Tubulin Polymerization Inhibitors. Discovery of A-289099 as an Orally Active Antitumor Agent

Bioorganic & medicinal chemistry letters, 2002-02, Vol.12 (3), p.465-469

2002

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Biological Activity of A-289099: An Orally Active Tubulin-binding Indolyloxazoline Derivative

Molecular cancer therapeutics, 2003-03, Vol.2 (3), p.227-233

2003

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Synthesis and Structure−Activity Relationships of 2-Pyridones: A Novel Series of Potent DNA Gyrase Inhibitors as Antibacterial Agents

Journal of medicinal chemistry, 1996-08, Vol.39 (16), p.3070-3088

1996

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Synthesis and SAR of indazole-pyridine based protein kinase B/Akt inhibitors

Bioorganic & medicinal chemistry, 2006-10, Vol.14 (20), p.6832-6846

2006

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Discovery of 1,4-dihydroindeno[1,2- c]pyrazoles as a novel class of potent and selective checkpoint kinase 1 inhibitors

Bioorganic & medicinal chemistry, 2007-04, Vol.15 (7), p.2759-2767

2007

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Synthesis and structure-activity relationships of novel arylfluoroquinolone antibacterial agents

Journal of medicinal chemistry, 1985-11, Vol.28 (11), p.1558-1564

1985

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Isoquinoline–pyridine-based protein kinase B/Akt antagonists: SAR and in vivo antitumor activity

Bioorganic & medicinal chemistry letters, 2006-06, Vol.16 (12), p.3150-3155

2006

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Practical Synthesis of 2-Pyridone Core: Ethyl 8-Chloro-1-cyclopropyl-7-fluoro-9-methyl-4-oxo-4H-quinolizinone-3-carboxylate

Heterocycles, 1999-06, Vol.51 (6), p.1345

1999

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Synthesis and structure-activity relationships of new arylfluoronaphthyridine antibacterial agents

Journal of medicinal chemistry, 1986-11, Vol.29 (11), p.2363-2369

1986

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Design, synthesis, and activity of achiral analogs of 2-quinolones and indoles as non-thiol farnesyltransferase inhibitors

Bioorganic & medicinal chemistry letters, 2005-04, Vol.15 (8), p.2033-2039

2005

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Design, synthesis, and activity of 4-quinolone and pyridone compounds as nonthiol-containing farnesyltransferase inhibitors

Bioorganic & medicinal chemistry letters, 2004-11, Vol.14 (21), p.5367-5370

2004

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Syntheses and antibacterial activity of novel 6-fluoro-7-(gem-disubstituted piperazin-1-yl)-quinolines

Canadian journal of chemistry, 1992-05, Vol.70 (5), p.1328-1337

1992

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1,4-Dihydroindeno[1,2- c]pyrazoles as potent checkpoint kinase 1 inhibitors: Extended exploration on phenyl ring substitutions and preliminary ADME/PK studies

Bioorganic & medicinal chemistry letters, 2007-07, Vol.17 (13), p.3618-3623

2007

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Cyanopyridyl containing 1,4-dihydroindeno[1,2- c]pyrazoles as potent checkpoint kinase 1 inhibitors: Improving oral biovailability

Bioorganic & medicinal chemistry letters, 2007-10, Vol.17 (20), p.5665-5670

2007

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L,4 -dihydroindeno[1,2 -c ]pyrazoles as potent checkpoint kinase 1 inhibitors : Extended exploration on phenyl ring substitutions and preliminary ADME/PK studies

Bioorganic & medicinal chemistry letters, 2007, Vol.17 (13), p.3618-3623

2007

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Synthesis and activity of 1-aryl-1'-imidazolyl methyl ethers as non-thiol farnesyltransferase inhibitors

Bioorganic & medicinal chemistry letters, 2004-11, Vol.14 (21), p.5371-5376

2004

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An alternative synthesis of temafloxacin, a potent antibacterial agent

Canadian journal of chemistry, 1992-05, Vol.70 (5), p.1323-1327

1992

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Synthesis and structure-activity relationships of 2-pyridones: II. 8-(Fluoro-substituted pyrrolidinyl)-2-pyridones as antibacterial agents

Bioorganic & medicinal chemistry letters, 1998-08, Vol.8 (15), p.1953-1958

1998

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A practical stereoselective synthesis of ( 2S, 4S)-4- tert-butoxycarbonylamino-2-methylpyrrolidine

Tetrahedron letters, 1995-11, Vol.36 (46), p.8391-8394

1995

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Short syntheses of 1,2,3,5‐tetrahydro‐5‐oxopyrrolo‐[1,2‐ a ]quinoline‐4‐carboxylic acid and 1,2,3,4‐tetrahydro‐6 H ‐6‐oxopyrido[1,2‐ a ]quinoline‐5‐carboxylic acid derivatives

Journal of heterocyclic chemistry, 1987-11, Vol.24 (6), p.1537-1539

1987

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Short syntheses of 1,2,3,5-tetrahydro-5-oxopyrrolo-[1,2-a]quinoline-4-carboxylic acid and 1,2,3,4-tetrahydro-6H-6-oxopyrido[1,2-a]quinoline-5-carboxylic acid derivatives

Journal of heterocyclic chemistry, 1987-11, Vol.24 (6), p.1537-1539

1987

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Synthesis and Biological Evaluation of 2-Indolyloxazolines as a New Class of Tubulin Polymerization Inhibitors. Discovery of A-289099 as an Orally Active Antitumor Agent

Biological Activity of A-289099: An Orally Active Tubulin-binding Indolyloxazoline Derivative

Synthesis and Structure−Activity Relationships of 2-Pyridones: A Novel Series of Potent DNA Gyrase Inhibitors as Antibacterial Agents

Synthesis and SAR of indazole-pyridine based protein kinase B/Akt inhibitors

Discovery of 1,4-dihydroindeno[1,2- c]pyrazoles as a novel class of potent and selective checkpoint kinase 1 inhibitors

Synthesis and structure-activity relationships of novel arylfluoroquinolone antibacterial agents

Isoquinoline–pyridine-based protein kinase B/Akt antagonists: SAR and in vivo antitumor activity

Practical Synthesis of 2-Pyridone Core: Ethyl 8-Chloro-1-cyclopropyl-7-fluoro-9-methyl-4-oxo-4H-quinolizinone-3-carboxylate

Synthesis and structure-activity relationships of new arylfluoronaphthyridine antibacterial agents

Design, synthesis, and activity of achiral analogs of 2-quinolones and indoles as non-thiol farnesyltransferase inhibitors

Design, synthesis, and activity of 4-quinolone and pyridone compounds as nonthiol-containing farnesyltransferase inhibitors

Syntheses and antibacterial activity of novel 6-fluoro-7-(gem-disubstituted piperazin-1-yl)-quinolines

1,4-Dihydroindeno[1,2- c]pyrazoles as potent checkpoint kinase 1 inhibitors: Extended exploration on phenyl ring substitutions and preliminary ADME/PK studies

Cyanopyridyl containing 1,4-dihydroindeno[1,2- c]pyrazoles as potent checkpoint kinase 1 inhibitors: Improving oral biovailability

L,4 -dihydroindeno[1,2 -c ]pyrazoles as potent checkpoint kinase 1 inhibitors : Extended exploration on phenyl ring substitutions and preliminary ADME/PK studies

Synthesis and activity of 1-aryl-1'-imidazolyl methyl ethers as non-thiol farnesyltransferase inhibitors

An alternative synthesis of temafloxacin, a potent antibacterial agent

Synthesis and structure-activity relationships of 2-pyridones: II. 8-(Fluoro-substituted pyrrolidinyl)-2-pyridones as antibacterial agents

A practical stereoselective synthesis of ( 2S, 4S)-4- tert-butoxycarbonylamino-2-methylpyrrolidine

Short syntheses of 1,2,3,5‐tetrahydro‐5‐oxopyrrolo‐[1,2‐ a ]quinoline‐4‐carboxylic acid and 1,2,3,4‐tetrahydro‐6 H ‐6‐oxopyrido[1,2‐ a ]quinoline‐5‐carboxylic acid derivatives

Short syntheses of 1,2,3,5-tetrahydro-5-oxopyrrolo-[1,2-a]quinoline-4-carboxylic acid and 1,2,3,4-tetrahydro-6H-6-oxopyrido[1,2-a]quinoline-5-carboxylic acid derivatives

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