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From Functional Fatty Acids to Potent and Selective Natural-Product-Inspired Mimetics via Conformational Profiling

ACS central science, 2024-02, Vol.10 (2), p.477-486

2024

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Catalyst-Controlled Regioselective Suzuki Couplings at Both Positions of Dihaloimidazoles, Dihalooxazoles, and Dihalothiazoles

Journal of organic chemistry, 2010-03, Vol.75 (5), p.1733-1739

2010

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Structure–Activity Relationship of Novel and Selective Biaryl-Chroman GPR40 AgoPAMs

ACS medicinal chemistry letters, 2018-07, Vol.9 (7), p.685-690

2018

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Structural basis for the cooperative allosteric activation of the free fatty acid receptor GPR40

Nature structural & molecular biology, 2017-07, Vol.24 (7), p.570

2017

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Highly Regioselective Palladium-Catalyzed Direct Arylation of Oxazole at C-2 or C-5 with Aryl Bromides, Chlorides, and Triflates

Organic letters, 2010-08, Vol.12 (16), p.3578-3581

2010

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Bioactivation of GPR40 Agonist MK-8666: Formation of Protein Adducts in Vitro from Reactive Acyl Glucuronide and Acyl CoA Thioester

Chemical research in toxicology, 2020-01, Vol.33 (1), p.191-201

2020

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Synthesis of a Lactone Diastereomer of the Cembranolide Uprolide D

Organic letters, 2010-10, Vol.12 (19), p.4328-4331

2010

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Driving to a Better Understanding of Acyl Glucuronide Transformations Using NMR and Molecular Modeling

Chemical research in toxicology, 2022-03, Vol.35 (3), p.459-474

2022

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Differentiation of Deprotonated Acyl‑, N‑, and O‑Glucuronide Drug Metabolites by Using Tandem Mass Spectrometry Based on Gas-Phase Ion–Molecule Reactions Followed by Collision-Activated Dissociation

Analytical chemistry (Washington), 2019-09, Vol.91 (17), p.11388-11396

2019

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Discovery of MK-8153, a Potent and Selective ROMK Inhibitor and Novel Diuretic/Natriuretic

Journal of medicinal chemistry, 2021-06, Vol.64 (11), p.7691-7701

2021

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Discovery of MK-7725, A Potent, Selective Bombesin Receptor Subtype-3 Agonist for the Treatment of Obesity

ACS medicinal chemistry letters, 2012-03, Vol.3 (3), p.252-256

2012

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GPR40 partial agonists and AgoPAMs: Differentiating effects on glucose and hormonal secretions in the rodent

PloS one, 2017-10, Vol.12 (10), p.e0186033-e0186033

2017

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Design, synthesis and biological evaluation of indane derived GPR40 agoPAMs

Bioorganic & medicinal chemistry letters, 2019-07, Vol.29 (14), p.1842-1848

2019

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Synthesis of novel 2-azabicyclo[3.1.1]heptane-5-carboxylic acid

Tetrahedron letters, 2016-03, Vol.57 (11), p.1268-1269

2016

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Lipase-Mediated Resolution of 4-TMS-3-butyn-2-ol and Use of the Mesylate Derivatives as a Precursor to a Highly Stereoselective Chiral Allenylindium Reagent

Organic letters, 2001-10, Vol.3 (21), p.3369-3372

2001

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The design and synthesis of novel spirocyclic heterocyclic sulfone ROMK inhibitors as diuretics

Bioorganic & medicinal chemistry letters, 2017-02, Vol.27 (4), p.1109-1114

2017

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Additions of Enantioenriched Allenylzinc and Indium Reagents to Lactic Aldehyde Ethers

Journal of organic chemistry, 2000-12, Vol.65 (24), p.8357-8360

2000

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The design and synthesis of potent, selective benzodiazepine sulfonamide bombesin receptor subtype 3 (BRS-3) agonists with an increased barrier of atropisomerization

Bioorganic & medicinal chemistry, 2012-05, Vol.20 (9), p.2845-2849

2012

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Improved Stability of Proline-Derived Direct Thrombin Inhibitors through Hydroxyl to Heterocycle Replacement

ACS medicinal chemistry letters, 2015-05, Vol.6 (5), p.553-557

2015

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Coupling of AlkynylTMS Derivatives with Vinylic Iodides. An Efficient Route to 1,3-Enynes and Dienes

Organic letters, 2001-12, Vol.3 (25), p.4107-4110

2001

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Discovery of Benzodiazepine Sulfonamide-Based Bombesin Receptor Subtype 3 Agonists and Their Unusual Chirality

ACS medicinal chemistry letters, 2011-12, Vol.2 (12), p.933-937

2011

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Pyridinesulfonylureas and pyridinesulfonamides as selective bombesin receptor subtype-3 (BRS-3) agonists

Bioorganic & medicinal chemistry letters, 2011-04, Vol.21 (7), p.2040-2043

2011

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Synthesis of 2,5-Disubstituted Tetrahydrofurans by Stereospecific Elimination−Cyclization of 1-Iodomethyl-1,5-bis-epoxides

Organic letters, 2003-05, Vol.5 (11), p.1931-1933

2003

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Efficient syntheses of four stable-isotope labeled (1R)-menthyl (1S,2S)-(+)-2-phenylcyclopropanecarboxylates

Organic & biomolecular chemistry, 2006-01, Vol.4 (14), p.2777-2784

2006

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From Functional Fatty Acids to Potent and Selective Natural-Product-Inspired Mimetics via Conformational Profiling

Catalyst-Controlled Regioselective Suzuki Couplings at Both Positions of Dihaloimidazoles, Dihalooxazoles, and Dihalothiazoles

Structure–Activity Relationship of Novel and Selective Biaryl-Chroman GPR40 AgoPAMs

Structural basis for the cooperative allosteric activation of the free fatty acid receptor GPR40

Highly Regioselective Palladium-Catalyzed Direct Arylation of Oxazole at C-2 or C-5 with Aryl Bromides, Chlorides, and Triflates

Bioactivation of GPR40 Agonist MK-8666: Formation of Protein Adducts in Vitro from Reactive Acyl Glucuronide and Acyl CoA Thioester

Synthesis of a Lactone Diastereomer of the Cembranolide Uprolide D

Driving to a Better Understanding of Acyl Glucuronide Transformations Using NMR and Molecular Modeling

Differentiation of Deprotonated Acyl‑, N‑, and O‑Glucuronide Drug Metabolites by Using Tandem Mass Spectrometry Based on Gas-Phase Ion–Molecule Reactions Followed by Collision-Activated Dissociation

Discovery of MK-8153, a Potent and Selective ROMK Inhibitor and Novel Diuretic/Natriuretic

Discovery of MK-7725, A Potent, Selective Bombesin Receptor Subtype-3 Agonist for the Treatment of Obesity

GPR40 partial agonists and AgoPAMs: Differentiating effects on glucose and hormonal secretions in the rodent

Design, synthesis and biological evaluation of indane derived GPR40 agoPAMs

Synthesis of novel 2-azabicyclo[3.1.1]heptane-5-carboxylic acid

Lipase-Mediated Resolution of 4-TMS-3-butyn-2-ol and Use of the Mesylate Derivatives as a Precursor to a Highly Stereoselective Chiral Allenylindium Reagent

The design and synthesis of novel spirocyclic heterocyclic sulfone ROMK inhibitors as diuretics

Additions of Enantioenriched Allenylzinc and Indium Reagents to Lactic Aldehyde Ethers

Discovery of MK-4409, a Novel Oxazole FAAH Inhibitor for the Treatment of Inflammatory and Neuropathic Pain

The design and synthesis of potent, selective benzodiazepine sulfonamide bombesin receptor subtype 3 (BRS-3) agonists with an increased barrier of atropisomerization

Improved Stability of Proline-Derived Direct Thrombin Inhibitors through Hydroxyl to Heterocycle Replacement

Coupling of AlkynylTMS Derivatives with Vinylic Iodides. An Efficient Route to 1,3-Enynes and Dienes

Discovery of Benzodiazepine Sulfonamide-Based Bombesin Receptor Subtype 3 Agonists and Their Unusual Chirality

Pyridinesulfonylureas and pyridinesulfonamides as selective bombesin receptor subtype-3 (BRS-3) agonists

Synthesis of 2,5-Disubstituted Tetrahydrofurans by Stereospecific Elimination−Cyclization of 1-Iodomethyl-1,5-bis-epoxides

Efficient syntheses of four stable-isotope labeled (1R)-menthyl (1S,2S)-(+)-2-phenylcyclopropanecarboxylates

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