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Aripiprazole, a novel antipsychotic, is a high-affinity partial agonist at human dopamine D2 receptors

The Journal of pharmacology and experimental therapeutics, 2002-07, Vol.302 (1), p.381

2002

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Forebrain-selective AMPA-receptor antagonism guided by TARP γ-8 as an antiepileptic mechanism

Nature medicine, 2016-12, Vol.22 (12), p.1496-1501

2016

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The novel antipsychotic aripiprazole is a partial agonist at short and long isoforms of D2 receptors linked to the regulation of adenylyl cyclase activity and prolactin release

Brain research, 2004-04, Vol.1003 (1-2), p.9-17

2004

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Bias analyses of preclinical and clinical D2 dopamine ligands: studies with immediate and complex signaling pathways

The Journal of pharmacology and experimental therapeutics, 2015-03, Vol.352 (3), p.480

2015

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JBS Special Issue: Innovative Screening Methodologies to Identify New Compounds for the Treatment of Central Nervous System Disorders

SLAS discovery, 2016-06, Vol.21 (5), p.425-426

2016

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Modulation of TARP γ 8-Containing AMPA Receptors as a Novel Therapeutic Approach for Chronic Pain

The Journal of pharmacology and experimental therapeutics, 2019-06, Vol.369 (3), p.345

2019

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Interaction of the novel antipsychotic aripiprazole with 5-HT1A and 5-HT2A receptors : functional receptor-binding and in vivo electrophysiological studies

Psychopharmacologia, 2007-02, Vol.190 (3), p.373-382

2007

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An Integrated Approach for Screening and Identification of Positive Allosteric Modulators of N-Methyl-D-Aspartate Receptors

Journal of biomolecular screening, 2016-06, Vol.21 (5), p.468-479

2016

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Optimization of a High-Throughput Assay for Calcium Channel Modulators on IonWorks Barracuda

Assay and drug development technologies, 2016-03, Vol.14 (2), p.75

2016

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IonWorks Barracuda Assay for Assessment of State-Dependent Sodium Channel Modulators

Assay and drug development technologies, 2016-03, Vol.14 (2), p.84

2016

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Aripiprazole's low intrinsic activities at human dopamine D2L and D2S receptors render it a unique antipsychotic

European journal of pharmacology, 2005-05, Vol.515 (1-3), p.10-19

2005

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Mechanism of Action of Aripiprazole Predicts Clinical Efficacy and a Favourable Side-Effect Profile

Journal of psychopharmacology (Oxford), 2004-09, Vol.18 (3), p.375-383

2004

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Drug-induced sensitization of adenylyl cyclase: assay streamlining and miniaturization for small molecule and siRNA screening applications

Journal of visualized experiments, 2014-01 (83), p.e51218-e51218

2014

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Oxime Carbamate—Discovery of a series of novel FAAH inhibitors

Bioorganic & medicinal chemistry letters, 2010-02, Vol.20 (3), p.1272-1277

2010

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Design, synthesis and evaluation of constrained tetrahydroimidazopyrimidine derivatives as antagonists of corticotropin-releasing factor type 1 receptor (CRF 1R)

Bioorganic & medicinal chemistry letters, 2010-03, Vol.20 (6), p.1905-1909

2010

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Focused Library Screening for Isoform Selective Adenylyl Cyclase 1 Inhibitors as Non‐Opioid Alternatives for Chronic and Inflammatory Pain

The FASEB journal, 2020-04, Vol.34 (S1), p.1-1

2020

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Diminished catalepsy and dopamine metabolism distinguish aripiprazole from haloperidol or risperidone

European journal of pharmacology, 2003-07, Vol.472 (1), p.89-97

2003

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Synthesis, structure–activity relationships, and anxiolytic activity of 7-aryl-6,7-dihydroimidazoimidazole corticotropin-releasing factor 1 receptor antagonists

Bioorganic & medicinal chemistry letters, 2005-09, Vol.15 (17), p.3870-3873

2005

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Synthesis and SAR exploration of dinapsoline analogues

Bioorganic & medicinal chemistry, 2004-02, Vol.12 (4), p.715-734

2004

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2-Arylaminothiazoles as high-affinity corticotropin-Releasing factor 1 receptor (CRF 1R) antagonists: synthesis, binding studies and behavioral efficacy

Bioorganic & medicinal chemistry letters, 2003-11, Vol.13 (22), p.3997-4000

2003

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(+)-Dinapsoline: An Efficient Synthesis and Pharmacological Profile of a Novel Dopamine Agonist

Journal of medicinal chemistry, 2002-08, Vol.45 (17), p.3660-3668

2002

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Supervised Machine Learning Applications to Winter Road Impacts

Burris, Kevin D

2018

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Drug-induced Sensitization of Adenylyl Cyclase: Assay Streamlining and Miniaturization for Small Molecule and siRNA Screening Applications

Journal of visualized experiments, 2014-01 (83)

2014

Volltextzugriff (PDF)

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Aripiprazole, a novel antipsychotic, is a high-affinity partial agonist at human dopamine D2 receptors

Forebrain-selective AMPA-receptor antagonism guided by TARP γ-8 as an antiepileptic mechanism

The novel antipsychotic aripiprazole is a partial agonist at short and long isoforms of D2 receptors linked to the regulation of adenylyl cyclase activity and prolactin release

Bias analyses of preclinical and clinical D2 dopamine ligands: studies with immediate and complex signaling pathways

Discovery of the First α‑Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptor Antagonist Dependent upon Transmembrane AMPA Receptor Regulatory Protein (TARP) γ‑8

JBS Special Issue: Innovative Screening Methodologies to Identify New Compounds for the Treatment of Central Nervous System Disorders

Modulation of TARP γ 8-Containing AMPA Receptors as a Novel Therapeutic Approach for Chronic Pain

Interaction of the novel antipsychotic aripiprazole with 5-HT1A and 5-HT2A receptors : functional receptor-binding and in vivo electrophysiological studies

An Integrated Approach for Screening and Identification of Positive Allosteric Modulators of N-Methyl-D-Aspartate Receptors

Optimization of a High-Throughput Assay for Calcium Channel Modulators on IonWorks Barracuda

IonWorks Barracuda Assay for Assessment of State-Dependent Sodium Channel Modulators

Aripiprazole's low intrinsic activities at human dopamine D2L and D2S receptors render it a unique antipsychotic

Mechanism of Action of Aripiprazole Predicts Clinical Efficacy and a Favourable Side-Effect Profile

Drug-induced sensitization of adenylyl cyclase: assay streamlining and miniaturization for small molecule and siRNA screening applications

Oxime Carbamate—Discovery of a series of novel FAAH inhibitors

Design, synthesis and evaluation of constrained tetrahydroimidazopyrimidine derivatives as antagonists of corticotropin-releasing factor type 1 receptor (CRF 1R)

Focused Library Screening for Isoform Selective Adenylyl Cyclase 1 Inhibitors as Non‐Opioid Alternatives for Chronic and Inflammatory Pain

Diminished catalepsy and dopamine metabolism distinguish aripiprazole from haloperidol or risperidone

Synthesis, structure–activity relationships, and anxiolytic activity of 7-aryl-6,7-dihydroimidazoimidazole corticotropin-releasing factor 1 receptor antagonists

Synthesis and SAR exploration of dinapsoline analogues

2-Arylaminothiazoles as high-affinity corticotropin-Releasing factor 1 receptor (CRF 1R) antagonists: synthesis, binding studies and behavioral efficacy

(+)-Dinapsoline: An Efficient Synthesis and Pharmacological Profile of a Novel Dopamine Agonist

Forebrain-selective AMPA-receptor antagonism guided by TARP [gamma]-8 as an antiepileptic mechanism.(alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid)

Supervised Machine Learning Applications to Winter Road Impacts

Drug-induced Sensitization of Adenylyl Cyclase: Assay Streamlining and Miniaturization for Small Molecule and siRNA Screening Applications

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