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Design and Synthesis of trans-3-(2-(4-((3-(3-(5-Methyl-1,2,4-oxadiazolyl))- phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro- 1H-3-benzazepine (SB-414796): A Potent and Selective Dopamine D3 Receptor Antagonist

Journal of medicinal chemistry, 2003-11, Vol.46 (23), p.4952-4964

2003

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Probing the Molecular Mechanism of Interaction between 4-n-Butyl-1-[4-(2-methylphenyl)-4-oxo-1-butyl]-piperidine (AC-42) and the Muscarinic M1 Receptor: Direct Pharmacological Evidence That AC-42 Is an Allosteric Agonist

Molecular pharmacology, 2006-01, Vol.69 (1), p.236

2006

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Design and Synthesis of trans-N-[4-[2-(6-Cyano-1,2,3,4-tetrahydroisoquinolin-2- yl)ethyl]cyclohexyl]-4-quinolinecarboxamide (SB-277011): A Potent and Selective Dopamine D3 Receptor Antagonist with High Oral Bioavailability and CNS Penetration in the Rat

Journal of medicinal chemistry, 2000-05, Vol.43 (9), p.1878-1885

2000

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Novel C-2 Substituted Carbapenem Derivatives: Part IV. Synthesis and Biological Activity of Five Membered Heteroaromatic Derivatives

The Journal of Antibiotics, 1998/02/25, Vol.51(2), pp.210-220

1998

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Design and synthesis of novel 2,3-dihydro-1H-isoindoles with high affinity and selectivity for the dopamine D3 receptor

Bioorganic & medicinal chemistry letters, 2001-03, Vol.11 (5), p.685-688

2001

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Probing the Molecular Mechanism of Interaction between 4- n -Butyl-1-[4-(2-methylphenyl)-4-oxo-1-butyl]-piperidine (AC-42) and the Muscarinic M 1 Receptor: Direct Pharmacological Evidence That AC-42 Is an Allosteric Agonist

Molecular pharmacology, 2006-01, Vol.69 (1), p.236-246

2006

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Novel 2,3,4,5-tetrahydro-1H-3-benzazepines with high affinity and selectivity for the dopamine D3 receptor

Bioorganic & medicinal chemistry letters, 2000-11, Vol.10 (22), p.2553-2555

2000

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Structure-activity relationships within a series of C(7)-substitutedoxyiminocephalosporins containing the C(3)-methylaminopyridiniumthiomethyl substituent : synthesis and biological properties of BRL 57342 and some close analogues

Journal of antibiotics, 1995, Vol.48 (5), p.417-424

1995

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Probing the molecular mechanism of interaction between 4-n-butyl-1-[4-(2-methylphenyl)-4-oxo-1-butyl]-piperidine (AC-42) and the muscarinic M(1) receptor: direct pharmacological evidence that AC-42 is an allosteric agonist

Molecular pharmacology, 2006-01, Vol.69 (1), p.236-246

2006

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Probing the Molecular Mechanism of Interaction between 4-n-Butyl-1-[4-(2-methylphenyl)-4-oxo-1-butyl]-piperidine (AC-42) and the Muscarinic M sub(1) Receptor: Direct Pharmacological Evidence That AC-42 Is an Allosteric Agonist

Molecular pharmacology, 2006-01, Vol.69 (1), p.236-246

2006

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Synthesis and biological properties of some 3-((N-subtstituted-amino)pyridinium-4-thiomethyl)-7-((2-amino-thiazol-4-yl)-2-(Z)-(methoxyimino)acetamido)ceph-3-em-4-carboxylates

Journal of antibiotics, 1993, Vol.46 (8), p.1289-1299

1993

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Synthesis and biological activity of 3-(N-substituted pyridinium-4-thiomethyl)-7.ALPHA.-formamido cephalosporins

Journal of antibiotics, 1993, Vol.46 (8), p.1279-1288

1993

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Synthesis of novel fused β-lactams by intramolecular 1,3-dipolar cycloadditions. Part 9. Preparation of the 7-oxo-1,3-diazabicyclo[3.2.0]- heptane-2-carboxylate and 8-oxo-1,3-diazabicyclo[4.2.0]octane-2-carboxylate ring systems

J. Chem. Soc., Perkin Trans. 1, 1986, p.1077-1095

1986

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Studies on semi-synthetic 7.ALPHA.-formamidocephalosporins. II Synthesis and antibacterial activity of some 7.ALPHA.-formamidoceph-3-em-1-oxide and 7.ALPHA.-formamido-1-oxadethiaceph-3-em derivatives

Journal of antibiotics, 1986, Vol.39 (12), p.1792-1795

1986

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An Expedient Synthesis of Allylic Polyprenyl Phosphates

Synthetic communications, 1999-08, Vol.29 (15), p.2639-2644

1999

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Synthesis of novel fused β-lactams by intramolecular 1,3-dipolar cycloadditions. Part 10. The 9-oxo-6-thia-1,3-diazabicyclo[5.2.0]nonene, 8-oxo-5-thia-1,3-diazabicyclo[4.2.0]octene, and 8-oxo-5-oxa-1,3-diazabicyclo[4.2.0]octene ring systems

J. Chem. Soc., Perkin Trans. 1, 1986, p.1097-1100

1986

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Direct incorporation of a 6α(7α)-formamido group into penicillin and cephalosporin sulphides and sulphoxides

J. Chem. Soc., Perkin Trans. 1, 1988 (10), p.2865-2873

1988

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Design and synthesis of trans-3-2-4-3-(3-(5-methyl-1,2,4-oxadiazolyl))-phenylcarboxamidocyclohexyl ethyl-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzazepine (SB-414796): A potent and selective dopamine D3 receptor antagonist

Journal of medicinal chemistry, 2003, Vol.46 (23), p.4952-4964

2003

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Synthesis of (2RS, 5RS, 6SR)-3-methoxycarbonyl-7-oxo-6-phenoxyacetamido-1-azabicyclo[3.2.0]hept-3-ene-2-carboxylic acid

Journal of the Chemical Society, Perkin Transactions 1, 1982, p.2123

1982

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Synthesis of some 1-oxa-1-dethiacephalosporins

Journal of the Chemical Society, Perkin Transactions 1, 1979, p.2268

1979

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Synthesis of novel fused β-lactams by intramolecular 1,3-dipolar cyclo-additions. Part 7. (9RS,9aRS)-9,9a-dihydro-5-methyl-8-oxo-9-phenoxyacetamido-8H-azeto[1,2-a]-v-triazolo[5,1-c]pyrazine-6-carboxylic acids and (3bRS,4RS,7SR)-4,5-dihydro-5-oxo-4-phenoxyacetamido-3bH-azeto[1′,2′:3,4]-imidazo[1,5-c]-v-triazole-7-carboxylic acid

J. Chem. Soc., Perkin Trans. 1, 1985, p.1491-1498

1985

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Studies on semi-synthetic 7.ALPHA.-formamidocephalosporins. III. Synthesis and antibacterial activity of some 7.BETA.-(D-2-(aryl)-2-((4-ethyl-2,3-dioxopiperazin-1-yl)-carbonylamino)acetamido)-7.ALPHA.-formamido-ceph-3-em-4-carboxylate derivatives

Journal of antibiotics, 1987, Vol.40 (5), p.646-651

1987

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Novel 1,2,3,4-tetrahydroisoquinolines with high affinity and selectivity for the dopamine D 3 receptor

Bioorganic & medicinal chemistry letters, 1999-01, Vol.9 (2), p.179-184

1999

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Design and Synthesis of trans-3-(2-(4-((3-(3-(5-Methyl-1,2,4-oxadiazolyl))- phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro- 1H-3-benzazepine (SB-414796): A Potent and Selective Dopamine D3 Receptor Antagonist

Probing the Molecular Mechanism of Interaction between 4-n-Butyl-1-[4-(2-methylphenyl)-4-oxo-1-butyl]-piperidine (AC-42) and the Muscarinic M1 Receptor: Direct Pharmacological Evidence That AC-42 Is an Allosteric Agonist

Design and Synthesis of trans-N-[4-[2-(6-Cyano-1,2,3,4-tetrahydroisoquinolin-2- yl)ethyl]cyclohexyl]-4-quinolinecarboxamide (SB-277011): A Potent and Selective Dopamine D3 Receptor Antagonist with High Oral Bioavailability and CNS Penetration in the Rat

Novel C-2 Substituted Carbapenem Derivatives: Part IV. Synthesis and Biological Activity of Five Membered Heteroaromatic Derivatives

Design and synthesis of novel 2,3-dihydro-1H-isoindoles with high affinity and selectivity for the dopamine D3 receptor

Probing the Molecular Mechanism of Interaction between 4- n -Butyl-1-[4-(2-methylphenyl)-4-oxo-1-butyl]-piperidine (AC-42) and the Muscarinic M 1 Receptor: Direct Pharmacological Evidence That AC-42 Is an Allosteric Agonist

Novel 2,3,4,5-tetrahydro-1H-3-benzazepines with high affinity and selectivity for the dopamine D3 receptor

Structure-activity relationships within a series of C(7)-substitutedoxyiminocephalosporins containing the C(3)-methylaminopyridiniumthiomethyl substituent : synthesis and biological properties of BRL 57342 and some close analogues

Design and Synthesis of trans - N -[4-[2-(6-Cyano-1,2,3,4-tetrahydroisoquinolin-2- yl)ethyl]cyclohexyl]-4-quinolinecarboxamide (SB-277011): A Potent and Selective Dopamine D 3 Receptor Antagonist with High Oral Bioavailability and CNS Penetration in the Rat

Probing the molecular mechanism of interaction between 4-n-butyl-1-[4-(2-methylphenyl)-4-oxo-1-butyl]-piperidine (AC-42) and the muscarinic M(1) receptor: direct pharmacological evidence that AC-42 is an allosteric agonist

Probing the Molecular Mechanism of Interaction between 4-n-Butyl-1-[4-(2-methylphenyl)-4-oxo-1-butyl]-piperidine (AC-42) and the Muscarinic M sub(1) Receptor: Direct Pharmacological Evidence That AC-42 Is an Allosteric Agonist

Synthesis and biological properties of some 3-((N-subtstituted-amino)pyridinium-4-thiomethyl)-7-((2-amino-thiazol-4-yl)-2-(Z)-(methoxyimino)acetamido)ceph-3-em-4-carboxylates

Synthesis and biological activity of 3-(N-substituted pyridinium-4-thiomethyl)-7.ALPHA.-formamido cephalosporins

Synthesis of novel fused β-lactams by intramolecular 1,3-dipolar cycloadditions. Part 9. Preparation of the 7-oxo-1,3-diazabicyclo[3.2.0]- heptane-2-carboxylate and 8-oxo-1,3-diazabicyclo[4.2.0]octane-2-carboxylate ring systems

Studies on semi-synthetic 7.ALPHA.-formamidocephalosporins. II Synthesis and antibacterial activity of some 7.ALPHA.-formamidoceph-3-em-1-oxide and 7.ALPHA.-formamido-1-oxadethiaceph-3-em derivatives

An Expedient Synthesis of Allylic Polyprenyl Phosphates

Synthesis of novel fused β-lactams by intramolecular 1,3-dipolar cycloadditions. Part 10. The 9-oxo-6-thia-1,3-diazabicyclo[5.2.0]nonene, 8-oxo-5-thia-1,3-diazabicyclo[4.2.0]octene, and 8-oxo-5-oxa-1,3-diazabicyclo[4.2.0]octene ring systems

Design and Synthesis of trans -3-(2-(4-((3-(3-(5-Methyl-1,2,4-oxadiazolyl))- phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro- 1 H -3-benzazepine (SB-414796): A Potent and Selective Dopamine D 3 Receptor Antagonist

Direct incorporation of a 6α(7α)-formamido group into penicillin and cephalosporin sulphides and sulphoxides

Design and synthesis of trans-3-2-4-3-(3-(5-methyl-1,2,4-oxadiazolyl))-phenylcarboxamidocyclohexyl ethyl-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzazepine (SB-414796): A potent and selective dopamine D3 receptor antagonist

Synthesis of (2RS, 5RS, 6SR)-3-methoxycarbonyl-7-oxo-6-phenoxyacetamido-1-azabicyclo[3.2.0]hept-3-ene-2-carboxylic acid

Synthesis of some 1-oxa-1-dethiacephalosporins

Studies on semi-synthetic 7.ALPHA.-formamidocephalosporins. III. Synthesis and antibacterial activity of some 7.BETA.-(D-2-(aryl)-2-((4-ethyl-2,3-dioxopiperazin-1-yl)-carbonylamino)acetamido)-7.ALPHA.-formamido-ceph-3-em-4-carboxylate derivatives

Novel 1,2,3,4-tetrahydroisoquinolines with high affinity and selectivity for the dopamine D 3 receptor

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