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Discovery of Cyclic Boronic Acid QPX7728, an Ultrabroad-Spectrum Inhibitor of Serine and Metallo-β-lactamases

Journal of medicinal chemistry, 2020-07, Vol.63 (14), p.7491-7507

2020

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Discovery of a Cyclic Boronic Acid β‑Lactamase Inhibitor (RPX7009) with Utility vs Class A Serine Carbapenemases

Journal of medicinal chemistry, 2015-05, Vol.58 (9), p.3682-3692

2015

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Selection of QPX7831, an Orally Bioavailable Prodrug of Boronic Acid β‑Lactamase Inhibitor QPX7728

Journal of medicinal chemistry, 2021-12, Vol.64 (23), p.17523-17529

2021

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Targeting thyroid hormone receptor-β agonists to the liver reduces cholesterol and triglycerides and improves the therapeutic index

Proceedings of the National Academy of Sciences - PNAS, 2007-09, Vol.104 (39), p.15490-15495

2007

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Scalable Synthesis of β‑Lactamase Inhibitor QPX7728 by Sequential Nickel-Catalyzed Boron Insertion into a Benzofuran Substrate and Enantioselective Cyclopropanation of the Resulting Vinylboronate

Organic process research & development, 2022-03, Vol.26 (3), p.925-935

2022

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Development of a Continuous Flow Process for a Matteson Reaction: From Lab Scale to Full-Scale Production of a Pharmaceutical Intermediate

Organic process research & development, 2019-05, Vol.23 (5), p.1069-1077

2019

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Scalable On-Demand Production of Purified Diazomethane Suitable for Sensitive Catalytic Reactions

Organic process research & development, 2021-03, Vol.25 (3), p.522-528

2021

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Antiviral Efficacy upon Administration of a HepDirect Prodrug of 2′-C-Methylcytidine to Hepatitis C Virus-Infected Chimpanzees

Antimicrobial Agents and Chemotherapy, 2011-08, Vol.55 (8), p.3854-3860

2011

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Pradefovir: A Prodrug That Targets Adefovir to the Liver for the Treatment of Hepatitis B

Journal of medicinal chemistry, 2008-02, Vol.51 (3), p.666-676

2008

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A Potent and Selective AMPK Activator That Inhibits de Novo Lipogenesis

ACS medicinal chemistry letters, 2010-12, Vol.1 (9), p.478-482

2010

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Synthesis and Biological Evaluation of a Series of Liver-Selective Phosphonic Acid Thyroid Hormone Receptor Agonists and Their Prodrugs

Journal of medicinal chemistry, 2008-11, Vol.51 (22), p.7075-7093

2008

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Synthesis and Characterization of a Novel Liver-Targeted Prodrug of Cytosine-1-β-d-arabinofuranoside Monophosphate for the Treatment of Hepatocellular Carcinoma

Journal of medicinal chemistry, 2006-12, Vol.49 (26), p.7711-7720

2006

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Liver-Targeted Prodrugs of 2‘-C-Methyladenosine for Therapy of Hepatitis C Virus Infection

Journal of medicinal chemistry, 2007-08, Vol.50 (16), p.3891-3896

2007

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Delivery of high levels of anti-proliferative nucleoside triphosphates to CYP3A-expressing cells as a potential treatment for hepatocellular carcinoma

Cancer chemotherapy and pharmacology, 2009-10, Vol.64 (5), p.981-991

2009

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Adenosine Kinase Inhibitors. 5. Synthesis, Enzyme Inhibition, and Analgesic Activity of Diaryl-erythro-furanosyltubercidin Analogues

Journal of medicinal chemistry, 2005-10, Vol.48 (20), p.6430-6441

2005

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Le fonds Léonce Beaumadier : le folklore réinventé

Patrimoines du Sud, 2022-03

Boyer, Serge

2022

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Le fonds Léonce Beaumadier : le folklore réinventé

Patrimoines du Sud, 2022-03 (15)

Boyer, Serge

2022

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Design, Synthesis, and Characterization of a Series of Cytochrome P450 3A-Activated Prodrugs (HepDirect Prodrugs) Useful for Targeting Phosph(on)ate-Based Drugs to the Liver

Journal of the American Chemical Society, 2004-04, Vol.126 (16), p.5154-5163

2004

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Stereoselective synthesis of 4- C-methyl-2,3,5-tri- O-benzyl- d-ribofuranose and 4- C-methyl-2,3,5-tri- O-benzyl- l-lyxofuranose

Tetrahedron letters, 2003-05, Vol.44 (21), p.4109-4112

2003

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Specific Inhibition of Formation of Transcription Complexes by a Calicheamicin Oligosaccharide: A Paradigm for the Development of Transcriptional Antagonists

Proceedings of the National Academy of Sciences - PNAS, 1994-09, Vol.91 (20), p.9203-9207

1994

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Design, Synthesis, and Characterization of a Series of Cytochrome P 450 3A-Activated Prodrugs (HepDirect Prodrugs) Useful for Targeting Phosph(on)ate-Based Drugs to the Liver

Journal of the American Chemical Society, 2004-04, Vol.126 (16), p.5154-5163

2004

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Studies Related to the Carbohydrate Sectors of Esperamicin and Calicheamicin: Definition of the Stability Limits of the Esperamicin Domain and Fashioning of a Glycosyl Donor from the Calicheamicin Domain

Journal of the American Chemical Society, 1995-05, Vol.117 (21), p.5720-5749

1995

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Interaction of calicheamicin γ1I and its related carbohydrates with DNA–protein complexes

Proceedings of the National Academy of Sciences - PNAS, 1999-09, Vol.96 (19), p.10643-10648

1999

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Stereoselective synthesis of nucleoside monophosphate HepDirect™ prodrugs

Tetrahedron letters, 2005-06, Vol.46 (25), p.4321-4324

2005

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A Remarkable Glycosidation Reaction: The Total Synthesis of Calicheamicin .gamma.1I

Journal of the American Chemical Society, 1995-05, Vol.117 (21), p.5750-5756

1995

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Discovery of Cyclic Boronic Acid QPX7728, an Ultrabroad-Spectrum Inhibitor of Serine and Metallo-β-lactamases

Discovery of a Cyclic Boronic Acid β‑Lactamase Inhibitor (RPX7009) with Utility vs Class A Serine Carbapenemases

Selection of QPX7831, an Orally Bioavailable Prodrug of Boronic Acid β‑Lactamase Inhibitor QPX7728

Targeting thyroid hormone receptor-β agonists to the liver reduces cholesterol and triglycerides and improves the therapeutic index

Scalable Synthesis of β‑Lactamase Inhibitor QPX7728 by Sequential Nickel-Catalyzed Boron Insertion into a Benzofuran Substrate and Enantioselective Cyclopropanation of the Resulting Vinylboronate

Development of a Continuous Flow Process for a Matteson Reaction: From Lab Scale to Full-Scale Production of a Pharmaceutical Intermediate

Scalable On-Demand Production of Purified Diazomethane Suitable for Sensitive Catalytic Reactions

Antiviral Efficacy upon Administration of a HepDirect Prodrug of 2′-C-Methylcytidine to Hepatitis C Virus-Infected Chimpanzees

Pradefovir: A Prodrug That Targets Adefovir to the Liver for the Treatment of Hepatitis B

A Potent and Selective AMPK Activator That Inhibits de Novo Lipogenesis

Synthesis and Biological Evaluation of a Series of Liver-Selective Phosphonic Acid Thyroid Hormone Receptor Agonists and Their Prodrugs

Synthesis and Characterization of a Novel Liver-Targeted Prodrug of Cytosine-1-β-d-arabinofuranoside Monophosphate for the Treatment of Hepatocellular Carcinoma

Liver-Targeted Prodrugs of 2‘-C-Methyladenosine for Therapy of Hepatitis C Virus Infection

Delivery of high levels of anti-proliferative nucleoside triphosphates to CYP3A-expressing cells as a potential treatment for hepatocellular carcinoma

Adenosine Kinase Inhibitors. 5. Synthesis, Enzyme Inhibition, and Analgesic Activity of Diaryl-erythro-furanosyltubercidin Analogues

Le fonds Léonce Beaumadier : le folklore réinventé

Le fonds Léonce Beaumadier : le folklore réinventé

Design, Synthesis, and Characterization of a Series of Cytochrome P450 3A-Activated Prodrugs (HepDirect Prodrugs) Useful for Targeting Phosph(on)ate-Based Drugs to the Liver

Stereoselective synthesis of 4- C-methyl-2,3,5-tri- O-benzyl- d-ribofuranose and 4- C-methyl-2,3,5-tri- O-benzyl- l-lyxofuranose

Specific Inhibition of Formation of Transcription Complexes by a Calicheamicin Oligosaccharide: A Paradigm for the Development of Transcriptional Antagonists

Design, Synthesis, and Characterization of a Series of Cytochrome P 450 3A-Activated Prodrugs (HepDirect Prodrugs) Useful for Targeting Phosph(on)ate-Based Drugs to the Liver

Studies Related to the Carbohydrate Sectors of Esperamicin and Calicheamicin: Definition of the Stability Limits of the Esperamicin Domain and Fashioning of a Glycosyl Donor from the Calicheamicin Domain

Interaction of calicheamicin γ1I and its related carbohydrates with DNA–protein complexes

Stereoselective synthesis of nucleoside monophosphate HepDirect™ prodrugs

A Remarkable Glycosidation Reaction: The Total Synthesis of Calicheamicin .gamma.1I

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