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Glutaminase is essential for the growth of triple-negative breast cancer cells with a deregulated glutamine metabolism pathway and its suppression synergizes with mTOR inhibition

PloS one, 2017-09, Vol.12 (9), p.e0185092-e0185092

2017

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Heterodimerization of V1a and V2 Vasopressin Receptors Determines the Interaction with β-Arrestin and Their Trafficking Patterns

Proceedings of the National Academy of Sciences - PNAS, 2004-02, Vol.101 (6), p.1548-1553

2004

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Oxytocin and Vasopressin V1a and V2 Receptors Form Constitutive Homo- and Heterodimers during Biosynthesis

Molecular endocrinology (Baltimore, Md.), 2003-04, Vol.17 (4), p.677-691

2003

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Probing the Existence of G Protein-Coupled Receptor Dimers by Positive and Negative Ligand-Dependent Cooperative Binding

Molecular pharmacology, 2006-11, Vol.70 (5), p.1783-1791

2006

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Combination of PIM and JAK2 inhibitors synergistically suppresses cell proliferation and overcomes drug resistance of myeloproliferative neoplasms

Oncotarget, 2014-05, Vol.5 (10), p.3362-3374

2014

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Characterization of (2S,4R)-1-[5-chloro-1-[(2,4-dimethoxyphenyl)sulfonyl]-3-(2-methoxy-phenyl)-2-oxo-2,3-dihydro-1H-indol-3-yl]-4-hydroxy-N,N-dimethyl-2-pyrrolidine carboxamide (SSR149415), a selective and orally active vasopressin V1b receptor antagonist

The Journal of pharmacology and experimental therapeutics, 2002-03, Vol.300 (3), p.1122

2002

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Cu(I)-catalyzed intramolecular cyclization of ene-carbamates: synthesis of indoles and pyrrolo[2,3- c]pyridines

Tetrahedron letters, 2005-12, Vol.46 (51), p.8877-8880

2005

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Identification of the Binding Sites of the SR49059 Nonpeptide Antagonist into the V1a Vasopressin Receptor Using Sulfydryl-reactive Ligands and Cysteine Mutants as Chemical Sensors

The Journal of biological chemistry, 2003-10, Vol.278 (41), p.40010-40019

2003

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Molecular cloning of the receptor for human antidiuretic hormone

Nature (London), 1992-05, Vol.357 (6376), p.333-335

1992

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Vasopressin and oxytocin receptors in the central nervous system

Critical reviews in neurobiology, 1996, Vol.10 (1), p.119

1996

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Pharmacology of (2S,4Z)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-(methoxyimino) -1-[(2'-methyl[1,1'-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamide, a new potent and selective nonpeptide antagonist of the oxytocin receptor

The Journal of pharmacology and experimental therapeutics, 2003-07, Vol.306 (1), p.253

2003

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Discovery of N-substituted 7-azaindoles as PIM1 kinase inhibitors – Part I

Bioorganic & medicinal chemistry letters, 2017-10, Vol.27 (20), p.4730-4734

2017

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Design of Benzophenone-Containing Photoactivatable Linear Vasopressin Antagonists: Pharmacological and Photoreactive Properties

Journal of medicinal chemistry, 2005-05, Vol.48 (9), p.3379-3388

2005

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Identification of Residues Responsible for the Selective Binding of Peptide Antagonists and Agonists in the V2 Vasopressin Receptor

The Journal of biological chemistry, 1998-11, Vol.273 (45), p.29462-29468

1998

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Two aromatic residues regulate the response of the human oxytocin receptor to the partial agonist arginine vasopressin

FEBS letters, 1996-11, Vol.397 (2), p.201-206

1996

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Rapid access to N -Boc phenylglycine derivatives via benzylic lithiation reactions

Tetrahedron, 2001-04, Vol.57 (15), p.2965-2972

2001

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Discovery of SARxxxx92, a pan-PIM kinase inhibitor, efficacious in a KG1 tumor model

Bioorganic & medicinal chemistry letters, 2020-12, Vol.30 (23), p.127625-127625, Article 127625

2020

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Abstract 5472: Basal-like breast cancer subtype is characterized by deregulated glutamine metabolism and is sensitive to GLS inhibition

Cancer research (Chicago, Ill.), 2018-07, Vol.78 (13_Supplement), p.5472-5472

2018

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Vasopressin receptors in the mouse (Mus musculus) brain: sex-related expression in the medial preoptic area and hypothalamus

Brain research, 1996-12, Vol.743 (1), p.32-39

1996

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Discovery of N-substituted 7-azaindoles as Pan-PIM kinases inhibitors – Lead optimization – Part III

Bioorganic & medicinal chemistry letters, 2019-02, Vol.29 (3), p.491-495

2019

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Discovery of N-substituted 7-azaindoles as Pan-PIM kinase inhibitors – Lead series identification – Part II

Bioorganic & medicinal chemistry letters, 2017-10, Vol.27 (20), p.4735-4740

2017

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Mapping Peptide-binding Domains of the Human V1a Vasopressin Receptor with a Photoactivatable Linear Peptide Antagonist

The Journal of biological chemistry, 1997-10, Vol.272 (42), p.26536-26544

1997

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A 13C NMR approach to categorizing potential limitations of α,β-unsaturated carbonyl systems in drug-like molecules

Bioorganic & medicinal chemistry letters, 2004-11, Vol.14 (22), p.5503-5507

2004

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Localization and characterization of vasopressin binding sites in the rat brain using an iodinated linear AVP antagonist

Brain research, 1993-09, Vol.622 (1), p.9-16

1993

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Glutaminase is essential for the growth of triple-negative breast cancer cells with a deregulated glutamine metabolism pathway and its suppression synergizes with mTOR inhibition

Heterodimerization of V1a and V2 Vasopressin Receptors Determines the Interaction with β-Arrestin and Their Trafficking Patterns

Oxytocin and Vasopressin V1a and V2 Receptors Form Constitutive Homo- and Heterodimers during Biosynthesis

Probing the Existence of G Protein-Coupled Receptor Dimers by Positive and Negative Ligand-Dependent Cooperative Binding

Combination of PIM and JAK2 inhibitors synergistically suppresses cell proliferation and overcomes drug resistance of myeloproliferative neoplasms

Characterization of (2S,4R)-1-[5-chloro-1-[(2,4-dimethoxyphenyl)sulfonyl]-3-(2-methoxy-phenyl)-2-oxo-2,3-dihydro-1H-indol-3-yl]-4-hydroxy-N,N-dimethyl-2-pyrrolidine carboxamide (SSR149415), a selective and orally active vasopressin V1b receptor antagonist

Cu(I)-catalyzed intramolecular cyclization of ene-carbamates: synthesis of indoles and pyrrolo[2,3- c]pyridines

Identification of the Binding Sites of the SR49059 Nonpeptide Antagonist into the V1a Vasopressin Receptor Using Sulfydryl-reactive Ligands and Cysteine Mutants as Chemical Sensors

Molecular cloning of the receptor for human antidiuretic hormone

Vasopressin and oxytocin receptors in the central nervous system

Pharmacology of (2S,4Z)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-(methoxyimino) -1-[(2'-methyl[1,1'-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamide, a new potent and selective nonpeptide antagonist of the oxytocin receptor

Discovery of N-substituted 7-azaindoles as PIM1 kinase inhibitors – Part I

Design of Benzophenone-Containing Photoactivatable Linear Vasopressin Antagonists: Pharmacological and Photoreactive Properties

Identification of Residues Responsible for the Selective Binding of Peptide Antagonists and Agonists in the V2 Vasopressin Receptor

Two aromatic residues regulate the response of the human oxytocin receptor to the partial agonist arginine vasopressin

Rapid access to N -Boc phenylglycine derivatives via benzylic lithiation reactions

Discovery of SARxxxx92, a pan-PIM kinase inhibitor, efficacious in a KG1 tumor model

PIM inhibitors target CD25-positive AML cells through concomitant suppression of STAT5 activation and degradation of MYC oncogene

Abstract 5472: Basal-like breast cancer subtype is characterized by deregulated glutamine metabolism and is sensitive to GLS inhibition

Vasopressin receptors in the mouse (Mus musculus) brain: sex-related expression in the medial preoptic area and hypothalamus

Discovery of N-substituted 7-azaindoles as Pan-PIM kinases inhibitors – Lead optimization – Part III

Discovery of N-substituted 7-azaindoles as Pan-PIM kinase inhibitors – Lead series identification – Part II

Mapping Peptide-binding Domains of the Human V1a Vasopressin Receptor with a Photoactivatable Linear Peptide Antagonist

A 13C NMR approach to categorizing potential limitations of α,β-unsaturated carbonyl systems in drug-like molecules

Localization and characterization of vasopressin binding sites in the rat brain using an iodinated linear AVP antagonist

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