UB Paderborn / Katalog / Suche / in CDI

1 – 25 von 161

Sortiert nach

Bias Factor and Therapeutic Window Correlate to Predict Safer Opioid Analgesics

Cell, 2017-11, Vol.171 (5), p.1165-1175.e13

2017

Volltextzugriff (PDF)

KLF5 Is Induced by FOXO1 and Causes Oxidative Stress and Diabetic Cardiomyopathy

Circulation research, 2021-02, Vol.128 (3), p.335-357

2021

Volltextzugriff (PDF)

Blocking Lactate Export by Inhibiting the Myc Target MCT1 Disables Glycolysis and Glutathione Synthesis

Cancer research (Chicago, Ill.), 2014-02, Vol.74 (3), p.908-920

2014

Volltextzugriff (PDF)

An ADAM10 Exosite Inhibitor Is Efficacious in an In Vivo Collagen-Induced Arthritis Model

Pharmaceuticals (Basel, Switzerland), 2024-01, Vol.17 (1), p.87

2024

Volltextzugriff (PDF)

Synthesis and Structure–Activity Relationships of Pteridine Dione and Trione Monocarboxylate Transporter 1 Inhibitors

Journal of medicinal chemistry, 2014-09, Vol.57 (17), p.7317-7324

2014

Volltextzugriff (PDF)

1,3-Diphenylureido hydroxamate as a promising scaffold for generation of potent antimalarial histone deacetylase inhibitors

Scientific reports, 2023-11, Vol.13 (1), p.21006-21006, Article 21006

2023

Volltextzugriff (PDF)

Pharmacoperone rescue of vasopressin 2 receptor mutants reveals unexpected constitutive activity and coupling bias

PloS one, 2017-08, Vol.12 (8), p.e0181830-e0181830

2017

Volltextzugriff (PDF)

Rescue of mutant gonadotropin-releasing hormone receptor function independent of cognate receptor activity

Scientific reports, 2020-06, Vol.10 (1), p.10579-10579, Article 10579

2020

Volltextzugriff (PDF)

Discovery and Optimization of Selective Inhibitors of Meprin α (Part I)

Pharmaceuticals (Basel, Switzerland), 2021-02, Vol.14 (3), p.197

2021

Volltextzugriff (PDF)

Hyperactivity in Mice Induced by Opioid Agonists with Partial Intrinsic Efficacy and Biased Agonism Administered Alone and in Combination with Morphine

Biomolecules (Basel, Switzerland), 2023-06, Vol.13 (6), p.935

2023

Volltextzugriff (PDF)

Site‐Selective γ‐C(sp3)−H and γ‐C(sp2)−H Arylation of Free Amino Esters Promoted by a Catalytic Transient Directing Group

Chemistry : a European journal, 2018-07, Vol.24 (38), p.9535-9541

2018

Volltextzugriff (PDF)

High throughput screening for drugs that inhibit 3C-like protease in SARS-CoV-2

SLAS discovery, 2023-04, Vol.28 (3), p.95-101

2023

Volltextzugriff (PDF)

Sequential Sonagashira and Larock Indole Synthesis Reactions in a General Strategy To Prepare Biologically Active β‑Carboline-Containing Alkaloids

Organic letters, 2014-12, Vol.16 (23), p.6124-6127

2014

Volltextzugriff (PDF)

Identification of potent small molecule inhibitors of SARS-CoV-2 entry

SLAS discovery, 2022-01, Vol.27 (1), p.8-19

2022

Volltextzugriff (PDF)

Selective Targeting of Extracellular Insulin-Degrading Enzyme by Quasi-Irreversible Thiol-Modifying Inhibitors

ACS chemical biology, 2015-12, Vol.10 (12), p.2716-2724

2015

Volltextzugriff (PDF)

Identification of small molecules that disrupt signaling between ABL and its positive regulator RIN1

PloS one, 2015-03, Vol.10 (3), p.e0121833-e0121833

2015

Volltextzugriff (PDF)

Native Directed Site-Selective δ‑C(sp3)–H and δ‑C(sp2)–H Arylation of Primary Amines

ACS catalysis, 2019-06, Vol.9 (6), p.4887-4891

2019

Volltextzugriff (PDF)

A G protein signaling-biased agonist at the μ-opioid receptor reverses morphine tolerance while preventing morphine withdrawal

Neuropsychopharmacology (New York, N.Y.), 2020-01, Vol.45 (2), p.416-425

2020

Volltextzugriff (PDF)

G protein signaling-biased mu opioid receptor agonists that produce sustained G protein activation are noncompetitive agonists

Proceedings of the National Academy of Sciences - PNAS, 2021-11, Vol.118 (48)

2021

Volltextzugriff (PDF)

Cardiomyocyte Krüppel-Like Factor 5 Promotes De Novo Ceramide Biosynthesis and Contributes to Eccentric Remodeling in Ischemic Cardiomyopathy

Circulation (New York, N.Y.), 2021-03, Vol.143 (11), p.1139-1156

2021

Volltextzugriff (PDF)

Preparation of tetrasubstituted pyrimido[4,5-d]pyrimidine diones

Tetrahedron letters, 2015-04, Vol.56 (15), p.1949-1952

2015

Volltextzugriff (PDF)

Comparison of morphine, oxycodone and the biased MOR agonist SR-17018 for tolerance and efficacy in mouse models of pain

Neuropharmacology, 2021-03, Vol.185, p.108439-108439, Article 108439

2021

Volltextzugriff (PDF)

Optimization of a Series of Mu Opioid Receptor (MOR) Agonists with High G Protein Signaling Bias

Journal of medicinal chemistry, 2018-10, Vol.61 (19), p.8895-8907

2018

Volltextzugriff (PDF)

Synthesis and Cytoxicity of Sempervirine and Analogues

Journal of organic chemistry, 2016-03, Vol.81 (5), p.2194-2200

2016

Volltextzugriff (PDF)

Irreversible and noncompetitive mu opioid receptor agonists

The FASEB journal, 2022-05, Vol.36 (S1), p.n/a

2022

Volltextzugriff (PDF)

1 – 25 von 161

Suche als RSS-Feed

Suchergebnisse filtern

Filter anzeigen

Nur zeigen

Geprüft (Peer-Review)
(126)
Mit Volltextzugriff
(155)

Publikationsform

Sprache

Englisch
(159)
Japanisch
(12)
Deutsch
(1)

Erscheinungsjahr

n.n

Thema

Science & Technology
(93)
Life Sciences & Biomedicine
(55)
Physical Sciences
(45)
Humans
(42)
Chemistry
(33)
Animals
(20)
Physics
(19)
Pharmacology & Pharmacy
(18)
Biological And Medical Sciences
(16)
Chemistry, Medicinal
(16)
Chemistry, Organic
(16)
Male
(16)
Female
(15)
Medical Sciences
(15)
Biochemistry & Molecular Biology
(14)
Mice
(14)
Physics, Atomic, Molecular & Chemical
(14)
Atomic And Molecular Physics
(12)
Molecular Structure
(12)
Cross Sections
(11)

15 weitere anzeigen...

Weniger anzeigen...

Zeitschrift / Serie

5 weitere anzeigen...

Weniger anzeigen...

Neu hinzugefügt

... seit 7 Tagen
(1)
... seit 90 Tagen
(2)

Menü

Weitere Dienste

Einstellungen

Bias Factor and Therapeutic Window Correlate to Predict Safer Opioid Analgesics

KLF5 Is Induced by FOXO1 and Causes Oxidative Stress and Diabetic Cardiomyopathy

Blocking Lactate Export by Inhibiting the Myc Target MCT1 Disables Glycolysis and Glutathione Synthesis

An ADAM10 Exosite Inhibitor Is Efficacious in an In Vivo Collagen-Induced Arthritis Model

Synthesis and Structure–Activity Relationships of Pteridine Dione and Trione Monocarboxylate Transporter 1 Inhibitors

1,3-Diphenylureido hydroxamate as a promising scaffold for generation of potent antimalarial histone deacetylase inhibitors

Pharmacoperone rescue of vasopressin 2 receptor mutants reveals unexpected constitutive activity and coupling bias

Rescue of mutant gonadotropin-releasing hormone receptor function independent of cognate receptor activity

Discovery and Optimization of Selective Inhibitors of Meprin α (Part I)

Hyperactivity in Mice Induced by Opioid Agonists with Partial Intrinsic Efficacy and Biased Agonism Administered Alone and in Combination with Morphine

Site‐Selective γ‐C(sp3)−H and γ‐C(sp2)−H Arylation of Free Amino Esters Promoted by a Catalytic Transient Directing Group

High throughput screening for drugs that inhibit 3C-like protease in SARS-CoV-2

Sequential Sonagashira and Larock Indole Synthesis Reactions in a General Strategy To Prepare Biologically Active β‑Carboline-Containing Alkaloids

Identification of potent small molecule inhibitors of SARS-CoV-2 entry

Selective Targeting of Extracellular Insulin-Degrading Enzyme by Quasi-Irreversible Thiol-Modifying Inhibitors

Identification of small molecules that disrupt signaling between ABL and its positive regulator RIN1

Native Directed Site-Selective δ‑C(sp3)–H and δ‑C(sp2)–H Arylation of Primary Amines

A G protein signaling-biased agonist at the μ-opioid receptor reverses morphine tolerance while preventing morphine withdrawal

G protein signaling-biased mu opioid receptor agonists that produce sustained G protein activation are noncompetitive agonists

Cardiomyocyte Krüppel-Like Factor 5 Promotes De Novo Ceramide Biosynthesis and Contributes to Eccentric Remodeling in Ischemic Cardiomyopathy

Preparation of tetrasubstituted pyrimido[4,5-d]pyrimidine diones

Comparison of morphine, oxycodone and the biased MOR agonist SR-17018 for tolerance and efficacy in mouse models of pain

Optimization of a Series of Mu Opioid Receptor (MOR) Agonists with High G Protein Signaling Bias

Synthesis and Cytoxicity of Sempervirine and Analogues

Irreversible and noncompetitive mu opioid receptor agonists

Suchergebnisse filtern