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Structural basis of small-molecule inhibition of human multidrug transporter ABCG2

Nature structural & molecular biology, 2018-04, Vol.25 (4), p.333

2018

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The extracellular loop 2 (ECL2) of the human histamine H4 receptor substantially contributes to ligand binding and constitutive activity

PloS one, 2015, Vol.10 (1), p.e0117185

2015

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Paradoxical stimulatory effects of the "standard" histamine H4-receptor antagonist JNJ7777120: the H4 receptor joins the club of 7 transmembrane domain receptors exhibiting functional selectivity

Molecular pharmacology, 2011-04, Vol.79 (4), p.631-638

2011

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Dimeric carbamoylguanidine-type histamine H2 receptor ligands: A new class of potent and selective agonists

Bioorganic & medicinal chemistry, 2015-07, Vol.23 (14), p.3957-3969

2015

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Potent and Selective Inhibitors of Breast Cancer Resistance Protein (ABCG2) Derived from the p-Glycoprotein (ABCB1) Modulator Tariquidar

Journal of medicinal chemistry, 2009-02, Vol.52 (4), p.1190-1197

2009

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High Affinity Agonists of the Neuropeptide Y (NPY) Y4 Receptor Derived from the C‑Terminal Pentapeptide of Human Pancreatic Polypeptide (hPP): Synthesis, Stereochemical Discrimination, and Radiolabeling

Journal of medicinal chemistry, 2016-07, Vol.59 (13), p.6045-6058

2016

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Highly Potent, Stable, and Selective Dimeric Hetarylpropylguanidine-Type Histamine H2 Receptor Agonists

ACS omega, 2018-03, Vol.3 (3), p.2865-2882

2018

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Synthesis and Structure−Activity Relationships of Cyanoguanidine-Type and Structurally Related Histamine H4 Receptor Agonists

Journal of medicinal chemistry, 2009-10, Vol.52 (20), p.6297-6313

2009

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Synthesis and dual histamine H₁ and H₂ receptor antagonist activity of cyanoguanidine derivatives

Molecules (Basel, Switzerland), 2013-11, Vol.18 (11), p.14186-14202

2013

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Luciferase reporter gene assay on human, murine and rat histamine H4 receptor orthologs: correlations and discrepancies between distal and proximal readouts

PloS one, 2013, Vol.8 (9), p.e73961

2013

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Fluorescence- and Radiolabeling of [Lys4,Nle17,30]hPP Yields Molecular Tools for the NPY Y4 Receptor

Bioconjugate chemistry, 2017-04, Vol.28 (4), p.1291-1304

2017

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Esters of Bendamustine Are by Far More Potent Cytotoxic Agents than the Parent Compound against Human Sarcoma and Carcinoma Cells

PloS one, 2015-07, Vol.10 (7), p.e0133743

2015

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[3H]UR-DE257: Development of a Tritium-Labeled Squaramide-Type Selective Histamine H2 Receptor Antagonist

ChemMedChem, 2015-01, Vol.10 (1), p.83-93

2015

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Dissociations in the effects of β2-adrenergic receptor agonists on cAMP formation and superoxide production in human neutrophils: support for the concept of functional selectivity

PloS one, 2013-05, Vol.8 (5), p.e64556

2013

Volltextzugriff (PDF)

Autodisplay of Human Hyaluronidase Hyal-1 on Escherichia coli and Identification of Plant-Derived Enzyme Inhibitors

Molecules (Basel, Switzerland), 2015-08, Vol.20 (9), p.15449-15468

2015

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Synthesis and Functional Characterization of Imbutamine Analogs as Histamine H3 and H4 Receptor Ligands

Archiv der Pharmazie (Weinheim), 2014-02, Vol.347 (2), p.77-88

2014

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The Neuropeptide Y Y1 Receptor: A Diagnostic Marker? Expression in MCF-7 Breast Cancer Cells Is Down-Regulated by Antiestrogens In Vitro and in Xenografts

PloS one, 2012-12, Vol.7 (12), p.e51032

2012

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G protein-coupled receptors function as logic gates for nanoparticle binding and cell uptake

Proceedings of the National Academy of Sciences - PNAS, 2010-06, Vol.107 (23), p.10667-10672

2010

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Structure‐Activity Relationship of Hetarylpropylguanidines Aiming at the Development of Selective Histamine Receptor Ligands

ChemistryOpen (Weinheim), 2019-03, Vol.8 (3), p.285-297

2019

Volltextzugriff (PDF)

Expression and functional properties of canine, rat, and murine histamine H4 receptors in Sf9 insect cells

Naunyn-Schmiedeberg's archives of pharmacology, 2011-05, Vol.383 (5), p.457-470

2011

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Toward Labeled Argininamide-Type NPY Y1 Receptor Antagonists: Identification of a Favorable Propionylation Site in BIBO3304

Archiv der Pharmazie (Weinheim), 2015-06, Vol.348 (6), p.390-398

2015

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Effect of the ABCB1 modulators elacridar and tariquidar on the distribution of paclitaxel in nude mice

Journal of cancer research and clinical oncology, 2008-05, Vol.134 (5), p.597-607

2008

Volltextzugriff (PDF)

Synthesis and Application of the First Radioligand Targeting the Allosteric Binding Pocket of Chemokine Receptor CXCR3

ChemMedChem, 2012-08, Vol.7 (8), p.1481-1489

2012

Volltextzugriff (PDF)

In Search of NPY Y4R Antagonists: Incorporation of Carbamoylated Arginine, Aza-Amino Acids, or d‑Amino Acids into Oligopeptides Derived from the C‑Termini of the Endogenous Agonists

ACS omega, 2017-07, Vol.2 (7), p.3616-3631

2017

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Constitutive activity and ligand selectivity of human, guinea pig, rat, and canine histamine H2 receptors

The Journal of pharmacology and experimental therapeutics, 2007-06, Vol.321 (3), p.983

2007

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Structural basis of small-molecule inhibition of human multidrug transporter ABCG2

The extracellular loop 2 (ECL2) of the human histamine H4 receptor substantially contributes to ligand binding and constitutive activity

Paradoxical stimulatory effects of the "standard" histamine H4-receptor antagonist JNJ7777120: the H4 receptor joins the club of 7 transmembrane domain receptors exhibiting functional selectivity

Dimeric carbamoylguanidine-type histamine H2 receptor ligands: A new class of potent and selective agonists

Potent and Selective Inhibitors of Breast Cancer Resistance Protein (ABCG2) Derived from the p-Glycoprotein (ABCB1) Modulator Tariquidar

High Affinity Agonists of the Neuropeptide Y (NPY) Y4 Receptor Derived from the C‑Terminal Pentapeptide of Human Pancreatic Polypeptide (hPP): Synthesis, Stereochemical Discrimination, and Radiolabeling

Highly Potent, Stable, and Selective Dimeric Hetarylpropylguanidine-Type Histamine H2 Receptor Agonists

Synthesis and Structure−Activity Relationships of Cyanoguanidine-Type and Structurally Related Histamine H4 Receptor Agonists

Synthesis and dual histamine H₁ and H₂ receptor antagonist activity of cyanoguanidine derivatives

Luciferase reporter gene assay on human, murine and rat histamine H4 receptor orthologs: correlations and discrepancies between distal and proximal readouts

Fluorescence- and Radiolabeling of [Lys4,Nle17,30]hPP Yields Molecular Tools for the NPY Y4 Receptor

Esters of Bendamustine Are by Far More Potent Cytotoxic Agents than the Parent Compound against Human Sarcoma and Carcinoma Cells

[3H]UR-DE257: Development of a Tritium-Labeled Squaramide-Type Selective Histamine H2 Receptor Antagonist

Dissociations in the effects of β2-adrenergic receptor agonists on cAMP formation and superoxide production in human neutrophils: support for the concept of functional selectivity

Autodisplay of Human Hyaluronidase Hyal-1 on Escherichia coli and Identification of Plant-Derived Enzyme Inhibitors

Synthesis and Functional Characterization of Imbutamine Analogs as Histamine H3 and H4 Receptor Ligands

The Neuropeptide Y Y1 Receptor: A Diagnostic Marker? Expression in MCF-7 Breast Cancer Cells Is Down-Regulated by Antiestrogens In Vitro and in Xenografts

G protein-coupled receptors function as logic gates for nanoparticle binding and cell uptake

Structure‐Activity Relationship of Hetarylpropylguanidines Aiming at the Development of Selective Histamine Receptor Ligands

Expression and functional properties of canine, rat, and murine histamine H4 receptors in Sf9 insect cells

Toward Labeled Argininamide-Type NPY Y1 Receptor Antagonists: Identification of a Favorable Propionylation Site in BIBO3304

Effect of the ABCB1 modulators elacridar and tariquidar on the distribution of paclitaxel in nude mice

Synthesis and Application of the First Radioligand Targeting the Allosteric Binding Pocket of Chemokine Receptor CXCR3

In Search of NPY Y4R Antagonists: Incorporation of Carbamoylated Arginine, Aza-Amino Acids, or d‑Amino Acids into Oligopeptides Derived from the C‑Termini of the Endogenous Agonists

Constitutive activity and ligand selectivity of human, guinea pig, rat, and canine histamine H2 receptors

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