UB Paderborn / Katalog / Suche / in CDI

1 – 25 von 127

Sortiert nach

SCYX-7158, an orally-active benzoxaborole for the treatment of stage 2 human African trypanosomiasis

PLoS neglected tropical diseases, 2011-06, Vol.5 (6), p.e1151

2011

Volltextzugriff (PDF)

Assessment of a pretomanid analogue library for African trypanosomiasis: Hit-to-lead studies on 6-substituted 2-nitro-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazine 8-oxides

Bioorganic & medicinal chemistry letters, 2018-01, Vol.28 (2), p.207-213

2018

Volltextzugriff (PDF)

In Memoriam: Michael Levandowsky (1935–2016)

The Journal of eukaryotic microbiology, 2017-07, Vol.64 (4), p.558-559

2017

Volltextzugriff (PDF)

Identification and characterization of a novel flavin-containing spermine oxidase of mammalian cell origin

Biochemical journal, 2002-11, Vol.367 (Pt 3), p.665-675

2002

Volltextzugriff (PDF)

Dibenzosuberyl substituted polyamines and analogs of clomipramine as effective inhibitors of trypanothione reductase; molecular docking, and assessment of trypanocidal activities

Bioorganic & medicinal chemistry, 2015-03, Vol.23 (5), p.996-1010

2015

Volltextzugriff (PDF)

Discovery of Novel Orally Bioavailable Oxaborole 6-Carboxamides That Demonstrate Cure in a Murine Model of Late-Stage Central Nervous System African Trypanosomiasis

Antimicrobial Agents and Chemotherapy, 2010-10, Vol.54 (10), p.4379-4388

2010

Volltextzugriff (PDF)

Alkanediamide-Linked Bisbenzamidines Are Promising Antiparasitic Agents

Pharmaceuticals (Basel, Switzerland), 2016-04, Vol.9 (2), p.20

2016

Volltextzugriff (PDF)

Pharmacokinetics and pharmacodynamics utilizing unbound target tissue exposure as part of a disposition-based rationale for lead optimization of benzoxaboroles in the treatment of Stage 2 Human African Trypanosomiasis

Parasitology, 2014-01, Vol.141 (1), p.104-118

2014

Volltextzugriff (PDF)

Trypanocidal Activity of 8-Methyl-5′-{[(Z)-4-Aminobut-2-enyl]-(Methylamino)}Adenosine (Genz-644131), an Adenosylmethionine Decarboxylase Inhibitor

Antimicrobial Agents and Chemotherapy, 2009-08, Vol.53 (8), p.3269-3272

2009

Volltextzugriff (PDF)

Novel S-Adenosylmethionine Decarboxylase Inhibitors for the Treatment of Human African Trypanosomiasis

Antimicrobial Agents and Chemotherapy, 2009-05, Vol.53 (5), p.2052-2058

2009

Volltextzugriff (PDF)

Benzoxaboroles: a new class of potential drugs for human African trypanosomiasis

Future medicinal chemistry, 2011-08, Vol.3 (10), p.1259-1278

2011

Volltextzugriff (PDF)

Discovery of Novel Benzoxaborole-Based Potent Antitrypanosomal Agents

ACS medicinal chemistry letters, 2010-07, Vol.1 (4), p.165-169

2010

Volltextzugriff (PDF)

2,4-Diaminopyrimidines as potent inhibitors of Trypanosoma brucei and identification of molecular targets by a chemical proteomics approach

PLoS neglected tropical diseases, 2011-02, Vol.5 (2), p.e956

2011

Volltextzugriff (PDF)

Novel alkylpolyaminoguanidines and alkylpolyaminobiguanides with potent antitrypanosomal activity

Bioorganic & medicinal chemistry letters, 2006-06, Vol.16 (12), p.3229-3232

2006

Volltextzugriff (PDF)

Synthesis and SAR of alkanediamide-linked bisbenzamidines with anti-trypanosomal and anti-pneumocystis activity

Bioorganic & medicinal chemistry letters, 2009-10, Vol.19 (20), p.5884-5886

2009

Volltextzugriff (PDF)

Metabolism of an Alkyl Polyamine Analog by a Polyamine Oxidase from the Microsporidian Encephalitozoon cuniculi

Antimicrobial Agents and Chemotherapy, 2009-06, Vol.53 (6), p.2599-2604

2009

Volltextzugriff (PDF)

Multiple Triclosan Targets in Trypanosoma brucei

Eukaryotic Cell, 2004-08, Vol.3 (4), p.855-861

2004

Volltextzugriff (PDF)

Selective Antimicrotubule Activity of N1-Phenyl-3,5-dinitro-N4,N4-di-n-propylsulfanilamide (GB-II-5) against Kinetoplastid Parasites

Molecular pharmacology, 2003-12, Vol.64 (6), p.1325

2003

Volltextzugriff (PDF)

Chemotherapy of Human African Trypanosomiasis

Interdisciplinary Perspectives on Infectious Diseases, 2009-01, Vol.2009, p.195040-5

2009

Volltextzugriff (PDF)

Novel Trypanocidal Analogs of 5′-(Methylthio)-Adenosine

Antimicrobial Agents and Chemotherapy, 2008-01, Vol.52 (1), p.211-219

2008

Volltextzugriff (PDF)

SAR of 2-amino and 2,4-diamino pyrimidines with in vivo efficacy against Trypanosoma brucei

Bioorganic & medicinal chemistry letters, 2011-05, Vol.21 (10), p.2816-2819

2011

Volltextzugriff (PDF)

Novel Synthetic Polyamines Are Effective in the Treatment of Experimental Microsporidiosis, an Opportunistic AIDS-Associated Infection

Antimicrobial Agents and Chemotherapy, 2002-01, Vol.46 (1), p.55-61

2002

Volltextzugriff (PDF)

Trypanocidal activity of piperazine-linked bisbenzamidines and bisbenzamidoxime, an orally active prodrug

International journal of antimicrobial agents, 2007-12, Vol.30 (6), p.555-561

2007

Volltextzugriff (PDF)

Polyamines with N-(3-phenylpropyl) substituents are effective competitive inhibitors of trypanothione reductase and trypanocidal agents

Bioorganic & medicinal chemistry letters, 2001-01, Vol.11 (2), p.251-254

2001

Volltextzugriff (PDF)

Inducible Resistance to Oxidant Stress in the Protozoan Leishmania chagasi

The Journal of biological chemistry, 2000-10, Vol.275 (43), p.33883-33889

2000

Volltextzugriff (PDF)

1 – 25 von 127

Suche als RSS-Feed

Suchergebnisse filtern

Filter anzeigen

Nur zeigen

Geprüft (Peer-Review)
(115)
Mit Volltextzugriff
(116)

Publikationsform

Sprache

Englisch
(127)
Japanisch
(6)

Erscheinungsjahr

n.n

Thema

Life Sciences & Biomedicine
(90)
Science & Technology
(90)
Animals
(87)
Pharmacology & Pharmacy
(48)
Biological And Medical Sciences
(47)
Medical Sciences
(39)
Mice
(37)
Pharmacology. Drug Treatments
(35)
Antibiotics. Antiinfectious Agents. Antiparasitic Agents
(34)
Trypanosoma Brucei Brucei - Drug Effects
(33)
Trypanocidal Agents - Pharmacology
(32)
Trypanosomiasis, African - Drug Therapy
(29)
Antiparasitic Agents
(25)
Trypanosoma Brucei Brucei
(25)
Microbiology
(24)
Chemistry, Medicinal
(22)
Humans
(21)
Trypanosoma Brucei
(21)
Female
(19)
Biochemistry & Molecular Biology
(18)

15 weitere anzeigen...

Weniger anzeigen...

Menü

Weitere Dienste

Einstellungen

SCYX-7158, an orally-active benzoxaborole for the treatment of stage 2 human African trypanosomiasis

Assessment of a pretomanid analogue library for African trypanosomiasis: Hit-to-lead studies on 6-substituted 2-nitro-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazine 8-oxides

In Memoriam: Michael Levandowsky (1935–2016)

Identification and characterization of a novel flavin-containing spermine oxidase of mammalian cell origin

Dibenzosuberyl substituted polyamines and analogs of clomipramine as effective inhibitors of trypanothione reductase; molecular docking, and assessment of trypanocidal activities

Discovery of Novel Orally Bioavailable Oxaborole 6-Carboxamides That Demonstrate Cure in a Murine Model of Late-Stage Central Nervous System African Trypanosomiasis

Alkanediamide-Linked Bisbenzamidines Are Promising Antiparasitic Agents

Pharmacokinetics and pharmacodynamics utilizing unbound target tissue exposure as part of a disposition-based rationale for lead optimization of benzoxaboroles in the treatment of Stage 2 Human African Trypanosomiasis

Trypanocidal Activity of 8-Methyl-5′-{[(Z)-4-Aminobut-2-enyl]-(Methylamino)}Adenosine (Genz-644131), an Adenosylmethionine Decarboxylase Inhibitor

Novel S-Adenosylmethionine Decarboxylase Inhibitors for the Treatment of Human African Trypanosomiasis

Benzoxaboroles: a new class of potential drugs for human African trypanosomiasis

Discovery of Novel Benzoxaborole-Based Potent Antitrypanosomal Agents

2,4-Diaminopyrimidines as potent inhibitors of Trypanosoma brucei and identification of molecular targets by a chemical proteomics approach

Novel alkylpolyaminoguanidines and alkylpolyaminobiguanides with potent antitrypanosomal activity

Synthesis and SAR of alkanediamide-linked bisbenzamidines with anti-trypanosomal and anti-pneumocystis activity

Metabolism of an Alkyl Polyamine Analog by a Polyamine Oxidase from the Microsporidian Encephalitozoon cuniculi

Multiple Triclosan Targets in Trypanosoma brucei

Selective Antimicrotubule Activity of N1-Phenyl-3,5-dinitro-N4,N4-di-n-propylsulfanilamide (GB-II-5) against Kinetoplastid Parasites

Chemotherapy of Human African Trypanosomiasis

Novel Trypanocidal Analogs of 5′-(Methylthio)-Adenosine

SAR of 2-amino and 2,4-diamino pyrimidines with in vivo efficacy against Trypanosoma brucei

Novel Synthetic Polyamines Are Effective in the Treatment of Experimental Microsporidiosis, an Opportunistic AIDS-Associated Infection

Trypanocidal activity of piperazine-linked bisbenzamidines and bisbenzamidoxime, an orally active prodrug

Polyamines with N-(3-phenylpropyl) substituents are effective competitive inhibitors of trypanothione reductase and trypanocidal agents

Inducible Resistance to Oxidant Stress in the Protozoan Leishmania chagasi

Suchergebnisse filtern