UB Paderborn / Katalog / Suche / in CDI

1 – 25 von 29

Sortiert nach

Structure–Activity and Structure–Toxicity Relationships of Peptoid‐Based Histone Deacetylase Inhibitors with Dual‐Stage Antiplasmodial Activity

ChemMedChem, 2019-05, Vol.14 (9), p.912-926

2019

Link zum Volltext

Verfügbarkeit prüfen

Open-source discovery of chemical leads for next-generation chemoprotective antimalarials

Science (American Association for the Advancement of Science), 2018-12, Vol.362 (6419)

2018

Link zum Volltext

Verfügbarkeit prüfen

Synthesis of (+)-7,20-Diisocyanoadociane and Liver-Stage Antiplasmodial Activity of the Isocyanoterpene Class

Journal of the American Chemical Society, 2016-06, Vol.138 (23), p.7268-7271

2016

Link zum Volltext

Verfügbarkeit prüfen

Sustained activation of Akt elicits mitochondrial dysfunction to block Plasmodium falciparum infection in the mosquito host

PLoS pathogens, 2013-02, Vol.9 (2), p.e1003180

2013

Link zum Volltext

Verfügbarkeit prüfen

Synthesis and Bioactivity of Phthalimide Analogs as Potential Drugs to Treat Schistosomiasis, a Neglected Disease of Poverty

Pharmaceuticals (Basel, Switzerland), 2020-02, Vol.13 (2), p.25

2020

Link zum Volltext

Verfügbarkeit prüfen

Design and Synthesis of Terephthalic Acid‐Based Histone Deacetylase Inhibitors with Dual‐Stage Anti‐Plasmodium Activity

ChemMedChem, 2017-10, Vol.12 (19), p.1627-1636

2017

Link zum Volltext

Verfügbarkeit prüfen

Two inhibitors of yeast plasma membrane ATPase 1 (ScPma1p): toward the development of novel antifungal therapies

Journal of cheminformatics, 2018-02, Vol.10 (1), p.6-9, Article 6

2018

Link zum Volltext

Verfügbarkeit prüfen

Cyclization-blocked proguanil as a strategy to improve the antimalarial activity of atovaquone

Communications biology, 2019-05, Vol.2 (1), p.166, Article 166

2019

Link zum Volltext

Verfügbarkeit prüfen

Development of a Potent Inhibitor of the Plasmodium Proteasome with Reduced Mammalian Toxicity

Journal of medicinal chemistry, 2017-08, Vol.60 (15), p.6721-6732

2017

Link zum Volltext

Verfügbarkeit prüfen

Validation of the protein kinase PfCLK3 as a multistage cross-species malarial drug target

Science (American Association for the Advancement of Science), 2019-08, Vol.365 (6456)

2019

Link zum Volltext

Verfügbarkeit prüfen

One-pot, multi-component synthesis and structure-activity relationships of peptoid-based histone deacetylase (HDAC) inhibitors targeting malaria parasites

European journal of medicinal chemistry, 2018-10, Vol.158, p.801-813

2018

Link zum Volltext

Verfügbarkeit prüfen

Investigation of the in vitro and in vivo efficacy of peptoid-based HDAC inhibitors with dual-stage antiplasmodial activity

European journal of medicinal chemistry, 2021-02, Vol.211, p.113065-113065, Article 113065

2021

Link zum Volltext

Verfügbarkeit prüfen

Synthesis of (+)-7,20-Diisocyanoadociane and Liver Stage Antiplasmodial Activity of the ICT Class

Journal of the American Chemical Society, 2016-05, Vol.138 (23), p.7268-7271

2016

Link zum Volltext

Verfügbarkeit prüfen

Overexpression of phosphatase and tensin homolog improves fitness and decreases Plasmodium falciparum development in Anopheles stephensi

Microbes and infection, 2013-11, Vol.15 (12), p.775-787

2013

Link zum Volltext

Verfügbarkeit prüfen

Probing the Open Global Health Chemical Diversity Library for Multistage-Active Starting Points for Next-Generation Antimalarials

ACS infectious diseases, 2020-04, Vol.6 (4), p.613-628

2020

Link zum Volltext

Verfügbarkeit prüfen

High-Throughput Luciferase-Based Assay for the Discovery of Therapeutics That Prevent Malaria

ACS infectious diseases, 2016-04, Vol.2 (4), p.281-293

2016

Link zum Volltext

Verfügbarkeit prüfen

Front Cover: Structure–Activity and Structure–Toxicity Relationships of Peptoid‐Based Histone Deacetylase Inhibitors with Dual‐Stage Antiplasmodial Activity (ChemMedChem 9/2019)

ChemMedChem, 2019-05, Vol.14 (9), p.887-887

2019

Link zum Volltext

Verfügbarkeit prüfen

Structure-Activity and Structure-Toxicity Relationships of Novel Peptoid-Based Histone Deacetylase Inhibitors with Dual-Stage Antiplasmodial Activity

ChemMedChem, 2019-02, Vol.14 (9), p.912-926

2019

Link zum Volltext

Verfügbarkeit prüfen

Validation of the protein kinase Pf CLK3 as a multistage cross-species malarial drug target

Science (American Association for the Advancement of Science), 2019-08, Vol.365 (6456)

2019

Link zum Volltext

Verfügbarkeit prüfen

Open Source Drug Discovery: Highly Potent Antimalarial Compounds Derived from the Tres Cantos Arylpyrroles

ACS central science, 2016-10, Vol.2 (10), p.687-701

2016

Link zum Volltext

Verfügbarkeit prüfen

1 – 25 von 29

Suche als RSS-Feed

Suchergebnisse filtern

Filter anzeigen

Nur zeigen

Geprüft (Peer-Review)
(23)
Mit Volltextzugriff
(26)

Publikationsform

Sprache

Englisch
(29)
Japanisch
(4)

Erscheinungsjahr

n.n

Thema

Science & Technology
(20)
Life Sciences & Biomedicine
(14)
Malaria
(12)
Chemistry, Medicinal
(11)
Humans
(11)
Pharmacology & Pharmacy
(11)
Antimalarials - Pharmacology
(10)
Plasmodium Falciparum - Drug Effects
(10)
Plasmodium Falciparum
(9)
Animals
(8)
Antimalarials - Chemistry
(7)
Drug Discovery
(6)
Parasites
(6)
Antimalarial Agents
(5)
Hep G2 Cells
(5)
Structure-Activity Relationship
(5)
Antimalarials - Chemical Synthesis
(4)
Histone Deacetylase
(4)
Histone Deacetylase Inhibitors - Pharmacology
(4)
Inhibitors
(4)

15 weitere anzeigen...

Weniger anzeigen...

Zeitschrift / Serie

5 weitere anzeigen...

Weniger anzeigen...

Menü

Weitere Dienste

Einstellungen

Structure–Activity and Structure–Toxicity Relationships of Peptoid‐Based Histone Deacetylase Inhibitors with Dual‐Stage Antiplasmodial Activity

Exploring a Tetrahydroquinoline Antimalarial Hit from the Medicines for Malaria Pathogen Box and Identification of its Mode of Resistance as PfeEF2

Chemoprotective antimalarials identified through quantitative high-throughput screening of Plasmodium blood and liver stage parasites

Substituted Aminoacetamides as Novel Leads for Malaria Treatment

Open-source discovery of chemical leads for next-generation chemoprotective antimalarials

Synthesis of (+)-7,20-Diisocyanoadociane and Liver-Stage Antiplasmodial Activity of the Isocyanoterpene Class

Sustained activation of Akt elicits mitochondrial dysfunction to block Plasmodium falciparum infection in the mosquito host

Synthesis and Bioactivity of Phthalimide Analogs as Potential Drugs to Treat Schistosomiasis, a Neglected Disease of Poverty

Design and Synthesis of Terephthalic Acid‐Based Histone Deacetylase Inhibitors with Dual‐Stage Anti‐Plasmodium Activity

Two inhibitors of yeast plasma membrane ATPase 1 (ScPma1p): toward the development of novel antifungal therapies

Cyclization-blocked proguanil as a strategy to improve the antimalarial activity of atovaquone

Development of a Potent Inhibitor of the Plasmodium Proteasome with Reduced Mammalian Toxicity

Validation of the protein kinase PfCLK3 as a multistage cross-species malarial drug target

One-pot, multi-component synthesis and structure-activity relationships of peptoid-based histone deacetylase (HDAC) inhibitors targeting malaria parasites

Investigation of the in vitro and in vivo efficacy of peptoid-based HDAC inhibitors with dual-stage antiplasmodial activity

Identification of a Potential Antimalarial Drug Candidate from a Series of 2‑Aminopyrazines by Optimization of Aqueous Solubility and Potency across the Parasite Life Cycle

Exploring a Tetrahydroquinoline Antimalarial Hit from the Medicines for Malaria Pathogen Box and Identification of its Mode of Resistance as Pf eEF2

Synthesis of (+)-7,20-Diisocyanoadociane and Liver Stage Antiplasmodial Activity of the ICT Class

Overexpression of phosphatase and tensin homolog improves fitness and decreases Plasmodium falciparum development in Anopheles stephensi

Probing the Open Global Health Chemical Diversity Library for Multistage-Active Starting Points for Next-Generation Antimalarials

High-Throughput Luciferase-Based Assay for the Discovery of Therapeutics That Prevent Malaria

Front Cover: Structure–Activity and Structure–Toxicity Relationships of Peptoid‐Based Histone Deacetylase Inhibitors with Dual‐Stage Antiplasmodial Activity (ChemMedChem 9/2019)

Structure-Activity and Structure-Toxicity Relationships of Novel Peptoid-Based Histone Deacetylase Inhibitors with Dual-Stage Antiplasmodial Activity

Validation of the protein kinase Pf CLK3 as a multistage cross-species malarial drug target

Open Source Drug Discovery: Highly Potent Antimalarial Compounds Derived from the Tres Cantos Arylpyrroles

Suchergebnisse filtern