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Pharmacological characterization of a novel, potent adenosine A1 and A2A receptor dual antagonist, 5-[5-amino-3-(4-fluorophenyl)pyrazin-2-yl]-1-isopropylpyridine-2(1H)-one (ASP5854), in models of Parkinson's disease and cognition

The Journal of pharmacology and experimental therapeutics, 2007-11, Vol.323 (2), p.708

2007

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Pharmacological Characterization of FR194921, a New Potent, Selective, and Orally Active Antagonist for Central Adenosine A1 Receptors

Journal of Pharmacological Sciences, 2004, Vol.96(1), pp.42-52

2004

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Design, Synthesis and Biological Evaluation of a Novel Series of Potent, Orally Active Adenosine A1 Receptor Antagonists with High Blood-Brain Barrier Permeability

Chemical and Pharmaceutical Bulletin, 2001, Vol.49(8), pp.988-998

2001

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Species differences in brain adenosine A1 receptor pharmacology revealed by use of xanthine and pyrazolopyridine based antagonists

British journal of pharmacology, 1997-11, Vol.122 (6), p.1202-1208

1997

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Discovery of FR166124, a novel water-soluble pyrazolo-[1,5-a]pyridine adenosine A1 receptor antagonist

Bioorganic & medicinal chemistry letters, 1999-07, Vol.9 (14), p.1979-1984

1999

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Synthesis of the water-soluble adenosine A1 receptor antagonist FR166124 through a novel sequential Horner-Emmons / isomerization reaction

Tetrahedron, , Vol.55 (34), p.10351-10364

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Novel adenosine A 1 receptor antagonists. Synthesis and structure–activity relationships of a novel series of 3-(2-cyclohexenyl-3-oxo-2,3-dihydropyridazin-6-yl)-2-phenylpyrazolo[1,5- a ]pyridines

Bioorganic & medicinal chemistry, 2000-01, Vol.8 (1), p.55-64

2000

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Species differences in brain adenosine A 1 receptor pharmacology revealed by use of xanthine and pyrazolopyridine based antagonists

British journal of pharmacology, 2009-02, Vol.122 (6), p.1202-1208

2009

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Discovery of 6-Oxo-3-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1(6H)-pyridazinebutanoic Acid (FK 838): A Novel Non-Xanthine Adenosine A1 Receptor Antagonist with Potent Diuretic Activity

Journal of medicinal chemistry, 1999-03, Vol.42 (5), p.779-783

1999

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Chiral formamidines. Asymmetric synthesis of 1,1-disubstituted tetrahydroisoquinolines

Tetrahedron letters, 1991-09, Vol.32 (40), p.5501-5504

1991

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Synthesis and Anticholinergic Activity of the Four Stereoisomers of 4-(Dimethylamino)-2-phenyl-2-(2-pyridyl)pentanamide

Journal of medicinal chemistry, 1994-04, Vol.37 (9), p.1378-1381

1994

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Chiral formamidines. The mechanism of mono- and di-alkylation leading to chiral, non-racemic tetrahydroisoquinolines

Tetrahedron letters, 1991-09, Vol.32 (40), p.5509-5512

1991

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P2I-34 ASP5854, a novel potent adenosine A1 & A2A receptor dual antagonist, improves motor disabilities and neuronal degeneration in models of Parkinson's disease

Journal of Pharmacological Sciences, 2008, Vol.106 (suppl.2), p.181-181

2008

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Pharmacological characterization of a simple behavioral response mediated selectively by central adenosine A1 receptors, using in vivo and in vitro techniques

The Journal of pharmacology and experimental therapeutics, 1998-06, Vol.285 (3), p.1023

1998

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Novel adenosine A1 receptor antagonists. Synthesis and structure-activity relationships of a novel series of 3-(2-cyclohexenyl-3-oxo-2,3-dihydropyridazin-6-yl)-2-phenylpyrazolo[1,5 -a]pyridines

Bioorganic & medicinal chemistry, 2000-01, Vol.8 (1), p.55-64

2000

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Syntheses of arborescin, 1,10-epiarborescin, and (11S)-guaia-3,10(14)-dieno-13,6.alpha.-lactone, the key intermediate in Greene and Crabbe's estafiatin synthesis, and the stereochemical assignment of arborescin

Journal of organic chemistry, 1982-09, Vol.47 (20), p.3909-3916

1982

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Discovery of FK453, a novel non-xanthine adenosine A1 receptor antagonist

Bioorganic & medicinal chemistry letters, 1996-09, Vol.6 (17), p.2059-2062

1996

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STUDIES ON THE SYNTHESES OF SESQUITERPENE LACTONES V. TOTAL SYNTHESIS OF ARBORESCIN

Chemistry letters, 1978-07, Vol.7 (7), p.727-730

1978

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Pyrazolopyridine derivatives act as competitive antagonists of brain adenosine A1 receptors : [35S]GTPγS binding studies

European journal of pharmacology, 1999-01, Vol.365 (2-3), p.309-315

1999

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Synthesis of the water-soluble adenosine A 1 receptor antagonist FR166124 through a novel sequential Horner-Emmons / isomerization reaction

Tetrahedron, 1999, Vol.55 (34), p.10351-10364

1999

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Pyrazolopyridine derivatives act as competitive antagonists of brain adenosine A 1 receptors: [ [formula omitted]]GTPγS binding studies

European journal of pharmacology, 1999, Vol.365 (2), p.309-315

1999

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Discovery of FR166124, a novel water-soluble pyrazolo-[1,5-α]pyridine adenosine A 1 receptor antagonist

Bioorganic & medicinal chemistry letters, 1999, Vol.9 (14), p.1979-1984

1999

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Discovery of 6-Oxo-3-(2-phenylpyrazolo[1,5- a ]pyridin-3-yl)-1(6 H )-pyridazinebutanoic Acid (FK 838): A Novel Non-Xanthine Adenosine A 1 Receptor Antagonist with Potent Diuretic Activity

Journal of medicinal chemistry, 1999-03, Vol.42 (5), p.779-783

1999

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A novel non-xanthine adenosine A1 receptor antagonist

European journal of pharmacology, 1995-06, Vol.279 (2-3), p.217-225

1995

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A reinvestigation of the reported synthesis of the spirobenzyl isoquinoline alkaloid, iso-ochotensine

Tetrahedron letters, 1997-06, Vol.38 (24), p.4195-4198

1997

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Pharmacological characterization of a novel, potent adenosine A1 and A2A receptor dual antagonist, 5-[5-amino-3-(4-fluorophenyl)pyrazin-2-yl]-1-isopropylpyridine-2(1H)-one (ASP5854), in models of Parkinson's disease and cognition

Pharmacological Characterization of FR194921, a New Potent, Selective, and Orally Active Antagonist for Central Adenosine A1 Receptors

Design, Synthesis and Biological Evaluation of a Novel Series of Potent, Orally Active Adenosine A1 Receptor Antagonists with High Blood-Brain Barrier Permeability

Species differences in brain adenosine A1 receptor pharmacology revealed by use of xanthine and pyrazolopyridine based antagonists

Discovery of FR166124, a novel water-soluble pyrazolo-[1,5-a]pyridine adenosine A1 receptor antagonist

Synthesis of the water-soluble adenosine A1 receptor antagonist FR166124 through a novel sequential Horner-Emmons / isomerization reaction

Novel adenosine A 1 receptor antagonists. Synthesis and structure–activity relationships of a novel series of 3-(2-cyclohexenyl-3-oxo-2,3-dihydropyridazin-6-yl)-2-phenylpyrazolo[1,5- a ]pyridines

Species differences in brain adenosine A 1 receptor pharmacology revealed by use of xanthine and pyrazolopyridine based antagonists

Discovery of 6-Oxo-3-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1(6H)-pyridazinebutanoic Acid (FK 838): A Novel Non-Xanthine Adenosine A1 Receptor Antagonist with Potent Diuretic Activity

Chiral formamidines. Asymmetric synthesis of 1,1-disubstituted tetrahydroisoquinolines

Synthesis and Anticholinergic Activity of the Four Stereoisomers of 4-(Dimethylamino)-2-phenyl-2-(2-pyridyl)pentanamide

Chiral formamidines. The mechanism of mono- and di-alkylation leading to chiral, non-racemic tetrahydroisoquinolines

P2I-34 ASP5854, a novel potent adenosine A1 & A2A receptor dual antagonist, improves motor disabilities and neuronal degeneration in models of Parkinson's disease

Pharmacological characterization of a simple behavioral response mediated selectively by central adenosine A1 receptors, using in vivo and in vitro techniques

Novel adenosine A1 receptor antagonists. Synthesis and structure-activity relationships of a novel series of 3-(2-cyclohexenyl-3-oxo-2,3-dihydropyridazin-6-yl)-2-phenylpyrazolo[1,5 -a]pyridines

Syntheses of arborescin, 1,10-epiarborescin, and (11S)-guaia-3,10(14)-dieno-13,6.alpha.-lactone, the key intermediate in Greene and Crabbe's estafiatin synthesis, and the stereochemical assignment of arborescin

Discovery of FK453, a novel non-xanthine adenosine A1 receptor antagonist

STUDIES ON THE SYNTHESES OF SESQUITERPENE LACTONES V. TOTAL SYNTHESIS OF ARBORESCIN

Pyrazolopyridine derivatives act as competitive antagonists of brain adenosine A1 receptors : [35S]GTPγS binding studies

Synthesis of the water-soluble adenosine A 1 receptor antagonist FR166124 through a novel sequential Horner-Emmons / isomerization reaction

Pyrazolopyridine derivatives act as competitive antagonists of brain adenosine A 1 receptors: [ [formula omitted]]GTPγS binding studies

Discovery of FR166124, a novel water-soluble pyrazolo-[1,5-α]pyridine adenosine A 1 receptor antagonist

Discovery of 6-Oxo-3-(2-phenylpyrazolo[1,5- a ]pyridin-3-yl)-1(6 H )-pyridazinebutanoic Acid (FK 838): A Novel Non-Xanthine Adenosine A 1 Receptor Antagonist with Potent Diuretic Activity

A novel non-xanthine adenosine A1 receptor antagonist

A reinvestigation of the reported synthesis of the spirobenzyl isoquinoline alkaloid, iso-ochotensine

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