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Identification of a μ-δ opioid receptor heteromer-biased agonist with antinociceptive activity

Proceedings of the National Academy of Sciences - PNAS, 2013-07, Vol.110 (29), p.12072-12077

2013

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Discovery, Synthesis, And Structure-Based Optimization of a Series of N‑(tert-Butyl)-2‑(N‑arylamido)-2-(pyridin-3-yl) Acetamides (ML188) as Potent Noncovalent Small Molecule Inhibitors of the Severe Acute Respiratory Syndrome Coronavirus (SARS-CoV) 3CL Protease

Journal of medicinal chemistry, 2013-01, Vol.56 (2), p.534-546

2013

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Global Consequences of Activation Loop Phosphorylation on Protein Kinase A

The Journal of biological chemistry, 2010-02, Vol.285 (6), p.3825-3832

2010

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Label-free LC-MS based assay to characterize small molecule compound binding to cells

SLAS discovery, 2022-10, Vol.27 (7), p.405-412

2022

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Selective and Brain Penetrant Neuropeptide Y Y2 Receptor Antagonists Discovered by Whole-Cell High-Throughput Screening

Molecular pharmacology, 2010-01, Vol.77 (1), p.46-57

2010

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Inhibitors of VIM-2 by screening pharmacologically active and click-chemistry compound libraries

Bioorganic & medicinal chemistry, 2009-07, Vol.17 (14), p.5027-5037

2009

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Design, synthesis and SAR analysis of novel potent and selective small molecule antagonists of NPBWR1 (GPR7)

Bioorganic & medicinal chemistry letters, 2012-12, Vol.22 (23), p.7135-7141

2012

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PKA-I Holoenzyme Structure Reveals a Mechanism for cAMP-Dependent Activation

Cell, 2007-09, Vol.130 (6), p.1032-1043

2007

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Small-molecule proteostasis regulators for protein conformational diseases

Nature chemical biology, 2011-12, Vol.8 (2), p.185-196

2011

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The design and synthesis of inhibitors of pantothenate synthetase

Organic & biomolecular chemistry, 2006-01, Vol.4 (19), p.3598-3610

2006

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High-Throughput Mass Spectrometry for Hit Identification: Current Landscape and Future Perspectives

SLAS DISCOVERY: Advancing the Science of Drug Discovery, 2021-02, Vol.26 (2), p.168-191

2021

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Virtual Ligand Screening of the p300/CBP Histone Acetyltransferase: Identification of a Selective Small Molecule Inhibitor

Chemistry & biology, 2010-05, Vol.17 (5), p.471-482

2010

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High throughput screening of potentially selective MMP-13 exosite inhibitors utilizing a triple-helical FRET substrate

Bioorganic & medicinal chemistry, 2009-02, Vol.17 (3), p.990-1005

2009

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An Ultra-High-Throughput Screen for Catalytic Inhibitors of Serine/Threonine Protein Phosphatases Types 1 and 5 (PP1C and PP5C)

SLAS discovery, 2017-01, Vol.22 (1), p.21-31

2017

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Inhibition of Mycobacterium tuberculosis Pantothenate Synthetase by Analogues of the Reaction Intermediate

Chembiochem : a European journal of chemical biology, 2008-11, Vol.9 (16), p.2606-2611

2008

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Assay Principle for Modulators of Protein−Protein Interactions and Its Application to Non-ATP-Competitive Ligands Targeting Protein Kinase A

Analytical chemistry (Washington), 2006-12, Vol.78 (24), p.8265-8272

2006

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Implementing Fluorescence Anisotropy Screening and Crystallographic Analysis to Define PKA Isoform-Selective Activation by cAMP Analogs

ACS chemical biology, 2013-10, Vol.8 (10), p.2164-2172

2013

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De Novo Discovery of Serotonin N-Acetyltransferase Inhibitors

Journal of medicinal chemistry, 2007-11, Vol.50 (22), p.5330-5338

2007

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Organisation of the pantothenate (vitamin B5) biosynthesis pathway in higher plants

The Plant journal : for cell and molecular biology, 2004-01, Vol.37 (1), p.61-72

2004

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Small-molecule inhibitors of acetyltransferase p300 identified by high-throughput screening are potent anticancer agents

Molecular cancer therapeutics, 2013-05, Vol.12 (5), p.610-620

2013

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NH-1,2,3-Triazole-based Inhibitors of the VIM-2 Metallo-β-Lactamase: Synthesis and Structure-Activity Studies

ACS medicinal chemistry letters, 2010-07, Vol.1 (4), p.150-154

2010

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Small Molecule Activators of TRPML3

Chemistry & biology, 2010-02, Vol.17 (2), p.135-148

2010

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Abstract C133: Effective targeting of KRAS-driven tumors by the first-in-class, orally bioavailable SOS1::KRAS inhibitor BI-3406

Molecular cancer therapeutics, 2019-12, Vol.18 (12_Supplement), p.C133-C133

2019

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Small Molecules Block the Polymerization of Z α1-Antitrypsin and Increase the Clearance of Intracellular Aggregates

Journal of medicinal chemistry, 2007-11, Vol.50 (22), p.5357-5363

2007

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NH-1,2,3-Triazole Inhibitors of the VIM-2 Metallo-β-Lactamase

ACS medicinal chemistry letters, 2010-07, Vol.1 (4), p.150-154

2010

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Identification of a μ-δ opioid receptor heteromer-biased agonist with antinociceptive activity

Discovery, Synthesis, And Structure-Based Optimization of a Series of N‑(tert-Butyl)-2‑(N‑arylamido)-2-(pyridin-3-yl) Acetamides (ML188) as Potent Noncovalent Small Molecule Inhibitors of the Severe Acute Respiratory Syndrome Coronavirus (SARS-CoV) 3CL Protease

Global Consequences of Activation Loop Phosphorylation on Protein Kinase A

Label-free LC-MS based assay to characterize small molecule compound binding to cells

Selective and Brain Penetrant Neuropeptide Y Y2 Receptor Antagonists Discovered by Whole-Cell High-Throughput Screening

Inhibitors of VIM-2 by screening pharmacologically active and click-chemistry compound libraries

Design, synthesis and SAR analysis of novel potent and selective small molecule antagonists of NPBWR1 (GPR7)

PKA-I Holoenzyme Structure Reveals a Mechanism for cAMP-Dependent Activation

Small-molecule proteostasis regulators for protein conformational diseases

The design and synthesis of inhibitors of pantothenate synthetase

High-Throughput Mass Spectrometry for Hit Identification: Current Landscape and Future Perspectives

Virtual Ligand Screening of the p300/CBP Histone Acetyltransferase: Identification of a Selective Small Molecule Inhibitor

High throughput screening of potentially selective MMP-13 exosite inhibitors utilizing a triple-helical FRET substrate

An Ultra-High-Throughput Screen for Catalytic Inhibitors of Serine/Threonine Protein Phosphatases Types 1 and 5 (PP1C and PP5C)

Inhibition of Mycobacterium tuberculosis Pantothenate Synthetase by Analogues of the Reaction Intermediate

Assay Principle for Modulators of Protein−Protein Interactions and Its Application to Non-ATP-Competitive Ligands Targeting Protein Kinase A

Implementing Fluorescence Anisotropy Screening and Crystallographic Analysis to Define PKA Isoform-Selective Activation by cAMP Analogs

De Novo Discovery of Serotonin N-Acetyltransferase Inhibitors

Organisation of the pantothenate (vitamin B5) biosynthesis pathway in higher plants

Small-molecule inhibitors of acetyltransferase p300 identified by high-throughput screening are potent anticancer agents

NH-1,2,3-Triazole-based Inhibitors of the VIM-2 Metallo-β-Lactamase: Synthesis and Structure-Activity Studies

Small Molecule Activators of TRPML3

Abstract C133: Effective targeting of KRAS-driven tumors by the first-in-class, orally bioavailable SOS1::KRAS inhibitor BI-3406

Small Molecules Block the Polymerization of Z α1-Antitrypsin and Increase the Clearance of Intracellular Aggregates

NH-1,2,3-Triazole Inhibitors of the VIM-2 Metallo-β-Lactamase

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