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Discovery and structure activity relationships of 7-benzyl triazolopyridines as stable, selective, and reversible inhibitors of myeloperoxidase

Bioorganic & medicinal chemistry, 2020-11, Vol.28 (22), p.115723-115723, Article 115723

2020

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Mechanism of Inhibition for BMS-791325, a Novel Non-nucleoside Inhibitor of Hepatitis C Virus NS5B Polymerase

The Journal of biological chemistry, 2014-11, Vol.289 (48), p.33456-33468

2014

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Development of a RapidFire mass spectrometry assay and a fluorescence assay for the discovery of kynurenine aminotransferase II inhibitors to treat central nervous system disorders

Analytical biochemistry, 2016-05, Vol.501, p.56-65

2016

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Dissecting the activation of thienopyridines by cytochromes P450 using a pharmacodynamic assay in vitro

The Journal of pharmacology and experimental therapeutics, 2011-11, Vol.339 (2), p.589

2011

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Identification of Reversible Small Molecule Inhibitors of Endothelial Lipase (EL) That Demonstrate HDL‑C Increase In Vivo

Journal of medicinal chemistry, 2020-02, Vol.63 (4), p.1660-1670

2020

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Potent Triazolopyridine Myeloperoxidase Inhibitors

ACS medicinal chemistry letters, 2018-12, Vol.9 (12), p.1175-1180

2018

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Identification of substituted benzothiazole sulfones as potent and selective inhibitors of endothelial lipase

Bioorganic & medicinal chemistry letters, 2019-08, Vol.29 (15), p.1918-1921

2019

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Corrigendum to “Identification of substituted benzothiazole sulfones as potent and selective inhibitors of endothelial lipase” [Bioorg. Med. Chem. Lett. 29 (2019) 1918–1921]

Bioorganic & medicinal chemistry letters, 2019-09, Vol.29 (17), p.2525-2525

2019

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Understanding Intra-Abdominal Hypertension: From the Bench to the Bedside

Journal of Intensive Care Medicine, 2012-05, Vol.27 (3), p.145-160

2012

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Triazolopyrimidines identified as reversible myeloperoxidase inhibitors

MedChemComm, 2017-11, Vol.8 (11), p.2093-2099

2017

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Sulfonylated Benzothiazoles as Inhibitors of Endothelial Lipase

ACS medicinal chemistry letters, 2018-12, Vol.9 (12), p.1263-1268

2018

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PK/PD Disconnect Observed with a Reversible Endothelial Lipase Inhibitor

ACS medicinal chemistry letters, 2018-07, Vol.9 (7), p.673-678

2018

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Identifying critically ill patients at high risk for developing acute renal failure: A pilot study

Kidney international, 2005-11, Vol.68 (5), p.2274-2280

2005

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Nonclinical Toxicology Assessments Support the Chronic Safety of Dapagliflozin, a First-in-Class Sodium-Glucose Cotransporter 2 Inhibitor

International journal of toxicology, 2013-09, Vol.32 (5), p.336-350

2013

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Immune-modulating enzyme indoleamine 2,3-dioxygenase is effectively inhibited by targeting its apo-form

Proceedings of the National Academy of Sciences - PNAS, 2018-03, Vol.115 (13), p.3249-3254

2018

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Anion Gap, Anion Gap Corrected for Albumin, and Base Deficit Fail to Accurately Diagnose Clinically Significant Hyperlactatemia in Critically Ill Patients

Journal of intensive care medicine, 2008-03, Vol.23 (2), p.122-127

2008

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Development and validation of a platelet calcium flux assay using a fluorescent imaging plate reader

Analytical biochemistry, 2006-10, Vol.357 (2), p.216-224

2006

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Identification of RIPK3 Type II Inhibitors Using High-Throughput Mechanistic Studies in Hit Triage

ACS medicinal chemistry letters, 2020-03, Vol.11 (3), p.266-271

2020

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Cloning and functional expression of the small subunit of acetolactate synthase from Nicotiana plumbaginifolia

Plant molecular biology, 1999-07, Vol.40 (5), p.795-806

1999

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Oxygenase side reactions of acetolactate synthase and other carbanion-forming enzymes

Biochemistry (Easton), 1991-08, Vol.30 (32), p.7883-7887

1991

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Discovery of 2-(Phenoxypyridine)-3-phenylureas as Small Molecule P2Y 1 Antagonists

Journal of medicinal chemistry, 2013-02, Vol.56 (4), p.1704-1714

2013

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Discovery and synthesis of tetrahydropyrimidinedione-4-carboxamides as endothelial lipase inhibitors

Bioorganic & medicinal chemistry letters, 2018-12, Vol.28 (23-24), p.3721-3725

2018

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Discovery and structure activity relationships of 7-benzyl triazolopyridines as stable, selective, and reversible inhibitors of myeloperoxidase

Conformationally Constrained ortho-Anilino Diaryl Ureas: Discovery of 1‑(2-(1′-Neopentylspiro[indoline-3,4′-piperidine]-1-yl)phenyl)-3-(4-(trifluoromethoxy)phenyl)urea, a Potent, Selective, and Bioavailable P2Y1 Antagonist

Mechanism of Inhibition for BMS-791325, a Novel Non-nucleoside Inhibitor of Hepatitis C Virus NS5B Polymerase

Development of a RapidFire mass spectrometry assay and a fluorescence assay for the discovery of kynurenine aminotransferase II inhibitors to treat central nervous system disorders

Dissecting the activation of thienopyridines by cytochromes P450 using a pharmacodynamic assay in vitro

Identification of Reversible Small Molecule Inhibitors of Endothelial Lipase (EL) That Demonstrate HDL‑C Increase In Vivo

Potent Triazolopyridine Myeloperoxidase Inhibitors

Identification of substituted benzothiazole sulfones as potent and selective inhibitors of endothelial lipase

Corrigendum to “Identification of substituted benzothiazole sulfones as potent and selective inhibitors of endothelial lipase” [Bioorg. Med. Chem. Lett. 29 (2019) 1918–1921]

Understanding Intra-Abdominal Hypertension: From the Bench to the Bedside

Triazolopyrimidines identified as reversible myeloperoxidase inhibitors

Sulfonylated Benzothiazoles as Inhibitors of Endothelial Lipase

PK/PD Disconnect Observed with a Reversible Endothelial Lipase Inhibitor

Identifying critically ill patients at high risk for developing acute renal failure: A pilot study

Nonclinical Toxicology Assessments Support the Chronic Safety of Dapagliflozin, a First-in-Class Sodium-Glucose Cotransporter 2 Inhibitor

Immune-modulating enzyme indoleamine 2,3-dioxygenase is effectively inhibited by targeting its apo-form

Anion Gap, Anion Gap Corrected for Albumin, and Base Deficit Fail to Accurately Diagnose Clinically Significant Hyperlactatemia in Critically Ill Patients

Development and validation of a platelet calcium flux assay using a fluorescent imaging plate reader

Discovery of 12 (BMS-986172) as a Highly Potent MGAT2 Inhibitor that Achieved Targeted Efficacious Exposures at a Low Human Dose for the Treatment of Metabolic Disorders

Screening Hit to Clinical Candidate: Discovery of BMS-963272, a Potent, Selective MGAT2 Inhibitor for the Treatment of Metabolic Disorders

Identification of RIPK3 Type II Inhibitors Using High-Throughput Mechanistic Studies in Hit Triage

Cloning and functional expression of the small subunit of acetolactate synthase from Nicotiana plumbaginifolia

Oxygenase side reactions of acetolactate synthase and other carbanion-forming enzymes

Discovery of 2-(Phenoxypyridine)-3-phenylureas as Small Molecule P2Y 1 Antagonists

Discovery and synthesis of tetrahydropyrimidinedione-4-carboxamides as endothelial lipase inhibitors

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