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Insight on [1,3]thiazolo[4,5-e]isoindoles as tubulin polymerization inhibitors

European journal of medicinal chemistry, 2021-02, Vol.212, p.113122, Article 113122

2021

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New Arylthioindoles and Related Bioisosteres at the Sulfur Bridging Group. 4. Synthesis, Tubulin Polymerization, Cell Growth Inhibition, and Molecular Modeling Studies

Journal of medicinal chemistry, 2009-12, Vol.52 (23), p.7512-7527

2009

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Interactions of Halichondrin B and Eribulin with Tubulin

Journal of chemical information and modeling, 2011-06, Vol.51 (6), p.1393-1404

2011

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Synthesis, antiproliferative activity, and mechanism of action of a series of 2-{[(2 E)-3-phenylprop-2-enoyl]amino}benzamides

European journal of medicinal chemistry, 2011-07, Vol.46 (7), p.2786-2796

2011

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Comparison of the Activities of the Truncated Halichondrin B Analog NSC 707389 (E7389) with Those of the Parent Compound and a Proposed Binding Site on Tubulin

Molecular pharmacology, 2006-12, Vol.70 (6), p.1866-1875

2006

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Synthesis and Biological Evaluation of Dihydrobenzofuran Lignans and Related Compounds as Potential Antitumor Agents that Inhibit Tubulin Polymerization

Journal of medicinal chemistry, 1999-12, Vol.42 (26), p.5475-5481

1999

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Laulimalide and Paclitaxel: A Comparison of Their Effects on Tubulin Assembly and Their Synergistic Action When Present Simultaneously

Molecular pharmacology, 2004-07, Vol.66 (1), p.113-121

2004

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Diazonamide A and a Synthetic Structural Analog: Disruptive Effects on Mitosis and Cellular Microtubules and Analysis of Their Interactions with Tubulin

Molecular pharmacology, 2003-06, Vol.63 (6), p.1273-1280

2003

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Synthesis, cytotoxicity, and inhibitory effects on tubulin polymerization of a new 3-heterocyclo substituted 2-styrylquinazolinones

European journal of medicinal chemistry, 2004-04, Vol.39 (4), p.299-304

2004

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Interaction of a Cyclostreptin Analogue with the Microtubule Taxoid Site: The Covalent Reaction Rapidly Follows Binding

Journal of natural products (Washington, D.C.), 2008-03, Vol.71 (3), p.370-374

2008

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Identification of pyrrolo[3′,4’:3,4]cyclohepta[1,2-d][1,2]oxazoles as promising new candidates for the treatment of lymphomas

European journal of medicinal chemistry, 2023-06, Vol.254, p.115372-115372, Article 115372

2023

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Interaction of diazonamide A with tubulin

Archives of biochemistry and biophysics, 2020-02, Vol.680, p.108217-108217, Article 108217

2020

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RS6077 induces mitotic arrest and selectively activates cell death in human cancer cell lines and in a lymphoma tumor in vivo

European journal of medicinal chemistry, 2023-01, Vol.246, p.114997-114997, Article 114997

2023

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Total synthesis and biological evaluation of ustiloxin natural products and two analogs

Bioorganic & medicinal chemistry letters, 2006-09, Vol.16 (18), p.4804-4807

2006

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Structure Guided Design, Synthesis, and Biological Evaluation of Oxetane-Containing Indole Analogues

Bioorganic & medicinal chemistry, 2023-09, Vol.92, p.117400-117400, Article 117400

2023

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Synthesis and biological evaluation of structurally diverse 6-aryl-3-Aroyl-Indole analogues as inhibitors of tubulin polymerization

European journal of medicinal chemistry, 2024-01, Vol.263, p.115794-115794, Article 115794

2024

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Characterizing the Epothilone Binding Site on β‑Tubulin by Photoaffinity Labeling: Identification of β‑Tubulin Peptides TARGSQQY and TSRGSQQY as Targets of an Epothilone Photoprobe for Polymerized Tubulin

Journal of medicinal chemistry, 2016-04, Vol.59 (7), p.3499-3514

2016

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The Spongistatins, Potently Cytotoxic Inhibitors of Tubulin Polymerization, Bind in a Distinct Region of the Vinca Domain

Biochemistry (Easton), 1995-08, Vol.34 (30), p.9714-9721

1995

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Synthesis and Biological Evaluation of Novel Epothilone B Side Chain Analogues

ChemMedChem, 2015-12, Vol.10 (12), p.1974-1979

2015

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Dolastatin 15, a potent antimitotic depsipeptide derived from Dolabella auricularia: Interaction with tubulin and effects on cellular microtubules

Biochemical pharmacology, 1992-06, Vol.43 (12), p.2637-2645

1992

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Antiproliferative 4-(1,2,4-oxadiazol-5-yl)piperidine-1-carboxamides, a new tubulin inhibitor chemotype

Bioorganic & medicinal chemistry letters, 2014-09, Vol.24 (18), p.4477-4481

2014

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Novel Microtubule-Targeting 7‑Deazahypoxanthines Derived from Marine Alkaloid Rigidins with Potent in Vitro and in Vivo Anticancer Activities

Journal of medicinal chemistry, 2016-01, Vol.59 (1), p.480-485

2016

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Interaction of pseudolaric acid B with the colchicine site of tubulin

Biochemical pharmacology, 2012-08, Vol.84 (4), p.444-450

2012

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S‐(4‐Methoxyphenyl)‐4‐methoxybenzenesulfonothioate as a Promising Lead Compound for the Development of a Renal Carcinoma Agent

ChemMedChem, 2020-03, Vol.15 (5), p.449-458

2020

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Synthesis, Antitubulin, and Antiproliferative SAR of C3/C1-Substituted Tetrahydroisoquinolines

ChemMedChem, 2014-02, Vol.9 (2), p.350-370

2014

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Insight on [1,3]thiazolo[4,5-e]isoindoles as tubulin polymerization inhibitors

New Arylthioindoles and Related Bioisosteres at the Sulfur Bridging Group. 4. Synthesis, Tubulin Polymerization, Cell Growth Inhibition, and Molecular Modeling Studies

Interactions of Halichondrin B and Eribulin with Tubulin

Synthesis, antiproliferative activity, and mechanism of action of a series of 2-{[(2 E)-3-phenylprop-2-enoyl]amino}benzamides

Comparison of the Activities of the Truncated Halichondrin B Analog NSC 707389 (E7389) with Those of the Parent Compound and a Proposed Binding Site on Tubulin

Synthesis and Biological Evaluation of Dihydrobenzofuran Lignans and Related Compounds as Potential Antitumor Agents that Inhibit Tubulin Polymerization

Laulimalide and Paclitaxel: A Comparison of Their Effects on Tubulin Assembly and Their Synergistic Action When Present Simultaneously

Diazonamide A and a Synthetic Structural Analog: Disruptive Effects on Mitosis and Cellular Microtubules and Analysis of Their Interactions with Tubulin

Synthesis, cytotoxicity, and inhibitory effects on tubulin polymerization of a new 3-heterocyclo substituted 2-styrylquinazolinones

Interaction of a Cyclostreptin Analogue with the Microtubule Taxoid Site: The Covalent Reaction Rapidly Follows Binding

Identification of pyrrolo[3′,4’:3,4]cyclohepta[1,2-d][1,2]oxazoles as promising new candidates for the treatment of lymphomas

Interaction of diazonamide A with tubulin

RS6077 induces mitotic arrest and selectively activates cell death in human cancer cell lines and in a lymphoma tumor in vivo

Total synthesis and biological evaluation of ustiloxin natural products and two analogs

Structure Guided Design, Synthesis, and Biological Evaluation of Oxetane-Containing Indole Analogues

Synthesis and biological evaluation of structurally diverse 6-aryl-3-Aroyl-Indole analogues as inhibitors of tubulin polymerization

Characterizing the Epothilone Binding Site on β‑Tubulin by Photoaffinity Labeling: Identification of β‑Tubulin Peptides TARGSQQY and TSRGSQQY as Targets of an Epothilone Photoprobe for Polymerized Tubulin

The Spongistatins, Potently Cytotoxic Inhibitors of Tubulin Polymerization, Bind in a Distinct Region of the Vinca Domain

Synthesis and Biological Evaluation of Novel Epothilone B Side Chain Analogues

Dolastatin 15, a potent antimitotic depsipeptide derived from Dolabella auricularia: Interaction with tubulin and effects on cellular microtubules

Antiproliferative 4-(1,2,4-oxadiazol-5-yl)piperidine-1-carboxamides, a new tubulin inhibitor chemotype

Novel Microtubule-Targeting 7‑Deazahypoxanthines Derived from Marine Alkaloid Rigidins with Potent in Vitro and in Vivo Anticancer Activities

Interaction of pseudolaric acid B with the colchicine site of tubulin

S‐(4‐Methoxyphenyl)‐4‐methoxybenzenesulfonothioate as a Promising Lead Compound for the Development of a Renal Carcinoma Agent

Synthesis, Antitubulin, and Antiproliferative SAR of C3/C1-Substituted Tetrahydroisoquinolines

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