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L-type amino acid transporter 1 utilizing prodrugs: How to achieve effective brain delivery and low systemic exposure of drugs
Journal of controlled release, 2017-09, Vol.261, p.93-104
2017
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Pharmacoproteomics of Brain Barrier Transporters and Substrate Design for the Brain Targeted Drug Delivery
Pharmaceutical research, 2022-07, Vol.39 (7), p.1363-1392
2022
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Prodrugs - an efficient way to breach delivery and targeting barriers
Current topics in medicinal chemistry, 2011-09, Vol.11 (18), p.2265
2011
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Mechanistic Study on the Use of the l‑Type Amino Acid Transporter 1 for Brain Intracellular Delivery of Ketoprofen via Prodrug: A Novel Approach Supporting the Development of Prodrugs for Intracellular Targets
Molecular pharmaceutics, 2019-07, Vol.16 (7), p.3261-3274
2019
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Improving drug delivery to the brain: the prodrug approach
Expert opinion on drug delivery, 2024-05, Vol.21 (5), p.1-693
2024
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Systemic and Brain Pharmacokinetics of Perforin Inhibitor Prodrugs
Molecular pharmaceutics, 2016-07, Vol.13 (7), p.2484-2491
2016
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Amino Acid Promoieties Alter Valproic Acid Pharmacokinetics and Enable Extended Brain Exposure
Neurochemical research, 2016-10, Vol.41 (10), p.2797-2809
2016
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Aminopeptidase B can bioconvert L-type amino acid transporter 1 (LAT1)-utilizing amide prodrugs in the brain
Frontiers in pharmacology, 2022-10, Vol.13, p.1034964-1034964
2022
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Targeted efflux transporter inhibitors – A solution to improve poor cellular accumulation of anti-cancer agents
International journal of pharmaceutics, 2018-10, Vol.550 (1-2), p.278-289
2018
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L-type amino acid transporter 1 utilizing prodrugs of ferulic acid revealed structural features supporting the design of prodrugs for brain delivery
European journal of pharmaceutical sciences, 2019-03, Vol.129, p.99-109
2019
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Metformin derivatives – Researchers’ friends or foes?
Biochemical pharmacology, 2023-09, Vol.215, p.115743-115743, Article 115743
2023
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Targeting of Perforin Inhibitor into the Brain Parenchyma Via a Prodrug Approach Can Decrease Oxidative Stress and Neuroinflammation and Improve Cell Survival
Molecular neurobiology, 2020-11, Vol.57 (11), p.4563-4577
2020
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Hemocompatible L-Type amino acid transporter 1 (LAT1)-Utilizing prodrugs of perforin inhibitors can accumulate into the pancreas and alleviate inflammation-induced apoptosis
Chemico-biological interactions, 2021-08, Vol.345, p.109560-109560, Article 109560
2021
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Specific transport of temozolomide does not override DNA repair-mediated chemoresistance
European journal of pharmaceutical sciences, 2024-04, Vol.195, p.106661-106661, Article 106661
2024
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l-Type amino acid transporter 1 (lat1)-mediated targeted delivery of perforin inhibitors
International journal of pharmaceutics, 2016-02, Vol.498 (1-2), p.205-216
2016
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Secondary carbamate linker can facilitate the sustained release of dopamine from brain-targeted prodrug
Bioorganic & medicinal chemistry letters, 2018-09, Vol.28 (17), p.2856-2860
2018
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Glutathione-S-transferase selective release of metformin from its sulfonamide prodrug
Bioorganic & medicinal chemistry letters, 2014-11, Vol.24 (21), p.5034-5036
2014
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Amino acid ester prodrugs conjugated to the α-carboxylic acid group do not display affinity for the L-type amino acid transporter 1 (LAT1)
European journal of pharmaceutical sciences, 2015-01, Vol.66, p.36-40
2015
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Cytochrome P450-activated prodrugs: targeted drug delivery
Current medicinal chemistry, 2008-10, Vol.15 (23), p.2346
2008
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Convenient microwave-assisted synthesis of lipophilic sulfenamide prodrugs of metformin
European journal of pharmaceutical sciences, 2013-07, Vol.49 (4), p.624-628
2013
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Determination of metformin and its prodrugs in human and rat blood by hydrophilic interaction liquid chromatography
Journal of pharmaceutical and biomedical analysis, 2009-10, Vol.50 (3), p.469-474
2009
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Design, Synthesis, and Evaluation of Novel Cyclic Phosphates of 5‑Aminosalicylic Acid as Cytochrome P450-Activated Prodrugs
Molecular pharmaceutics, 2013-02, Vol.10 (2), p.532-537
2013
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Novel cyclic phosphate prodrug approach for cytochrome p450-activated drugs containing an alcohol functionality
Pharmaceutical research, 2007-04, Vol.24 (4), p.679-687
2007
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