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Nucleophilic (Radio)Fluorination of Redox-Active Esters via Radical-Polar Crossover Enabled by Photoredox Catalysis

Journal of the American Chemical Society, 2020-05, Vol.142 (20), p.9493-9500

2020

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Synthesis of a dual carbon‐14‐labeled calcitonin gene‐related peptide receptor antagonist for use in a human absorption–distribution–metabolism–elimination study

Journal of labelled compounds & radiopharmaceuticals, 2022-05, Vol.65 (5), p.126-139

2022

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Synthesis of carbon‐14 and stable isotope labeled Censavudine

Journal of labelled compounds & radiopharmaceuticals, 2022-04, Vol.65 (4), p.112-122

2022

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Synthesis of tritium labeled 30‐KDa PEG and conjugation to form [3H]Pegbelfermin

Journal of labelled compounds & radiopharmaceuticals, 2021-10, Vol.64 (12), p.477-481

2021

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The synthesis and analysis of [phenyl-14C(U)]BMS-770767 and [13C6]BMS-770767 for use in discovery biotransformation, human ADME and bioanalytical studies

Journal of labelled compounds & radiopharmaceuticals, 2016-12, Vol.59 (14), p.657-664

2016

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The syntheses of isotopically labelled CB-1 antagonists for the treatment of obesity

Journal of labelled compounds & radiopharmaceuticals, 2016-12, Vol.59 (14), p.665-672

2016

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Synthesis of isotopically labeled daclatasvir for use in human clinical studies

Journal of labelled compounds & radiopharmaceuticals, 2016-04, Vol.59 (4), p.164-170

2016

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The syntheses of [14C]BMS-823778 for use in a human ADME clinical study and of [13CD3 13CD2]BMT-094817, a stable-isotope labeled standard of a newly detected human metabolite

Journal of labelled compounds & radiopharmaceuticals, 2016-05, Vol.59 (6), p.255-259

2016

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Synthesis of stable isotope-labeled epothilone D using a degradation-reconstruction approach

Journal of labelled compounds & radiopharmaceuticals, 2015-07, Vol.58 (9), p.361-369

2015

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Synthesis of a stable isotopically labeled universal surrogate peptide for use as an internal standard in LC-MS/MS bioanalysis of human IgG and Fc-fusion protein drug candidates

Journal of labelled compounds & radiopharmaceuticals, 2014-07, Vol.57 (9), p.579-583

2014

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Synthesis of unlabelled and stable‐isotope–labelled glucuronide metabolites of dapagliflozin and synthesis of stable‐isotope–labelled dapagliflozin

Journal of labelled compounds & radiopharmaceuticals, 2017-03, Vol.60 (3), p.150-159

2017

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Distinguishing a phosphate ester prodrug from its isobaric sulfate metabolite by mass spectrometry without the metabolite standard

Rapid communications in mass spectrometry, 2009-10, Vol.23 (19), p.3107-3113

2009

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An alternative and robust synthesis of [13C4]Baraclude® (entecavir)

Journal of labelled compounds & radiopharmaceuticals, 2013-10, Vol.56 (12), p.632-636

2013

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An improved synthesis of [2-14C]2, 5-dichloropyrimidine

Journal of labelled compounds & radiopharmaceuticals, 2012-06, Vol.55 (8), p.300-302

2012

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Carbon-14 labeled methyl 2-chloro-2-oxoacetate: a convenient carbon-14 labeled oxalyl chloride equivalent

Journal of labelled compounds & radiopharmaceuticals, 2009-11, Vol.52 (13), p.549-552

2009

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A novel synthesis of [2-14C]2,5-dichloropyrimidine

Journal of labelled compounds & radiopharmaceuticals, 2011-11, Vol.54 (13), p.813-815

2011

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LC-MS/MS bioanalysis of plasma 1, 14-tetradecanedioic acid and 1, 16-hexadecanedioic acid as candidate biomarkers for organic anion-transporting polypeptide mediated drug-drug interactions

Bioanalysis, 2018-09, Vol.10 (18), p.1473-1485

2018

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Synthesis and stability of a carbon-14-labeled 3-hydroxy-3-methylglutaryl coenzyme-A reductase inhibitor

Journal of labelled compounds & radiopharmaceuticals, 2011-02, Vol.54 (2), p.72-79

2011

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The syntheses and in vitro biotransformation studies of [14C]apixaban, a highly potent, selective, efficacious and orally bioavailable inhibitor of blood coagulation Factor Xa

Journal of labelled compounds & radiopharmaceuticals, 2011-06, Vol.54 (8), p.418-425

2011

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Synthesis of [3α-3H] 17α-Hydroxy pregnenolone and [3α-3H] Pregnenolone

Journal of labelled compounds & radiopharmaceuticals, 2014-01, Vol.57 (1), p.1-11

2014

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Synthesis of multi-labeled [14C]Aripiprazole

Journal of labelled compounds & radiopharmaceuticals, 2006-01, Vol.49 (1), p.1-9

2006

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Carbon-14 labeling of Saxagliptin (BMS-477118)

Journal of labelled compounds & radiopharmaceuticals, 2007-11, Vol.50 (13), p.1224-1229

2007

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Synthesis of carbon-14 and stable isotope labeled Avagacestat: a novel gamma secretase inhibitor for the treatment of Alzheimer's disease

Journal of labelled compounds & radiopharmaceuticals, 2014-08, Vol.57 (10), p.600-605

2014

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Synthesis of [1,2-3H]ethylamine hydrochloride and [3H]-labeled apadenoson for a human ADME study

Journal of labelled compounds & radiopharmaceuticals, 2008-02, Vol.51 (2), p.113-117

2008

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Overcoming bioanalytical challenges in an Onglyza(®) intravenous [(14)C]microdose absolute bioavailability study with accelerator MS

Bioanalysis, 2012-08, Vol.4 (15), p.1855-1870

2012

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Nucleophilic (Radio)Fluorination of Redox-Active Esters via Radical-Polar Crossover Enabled by Photoredox Catalysis

Synthesis of a dual carbon‐14‐labeled calcitonin gene‐related peptide receptor antagonist for use in a human absorption–distribution–metabolism–elimination study

Synthesis of carbon‐14 and stable isotope labeled Censavudine

Synthesis of tritium labeled 30‐KDa PEG and conjugation to form [3H]Pegbelfermin

The synthesis and analysis of [phenyl-14C(U)]BMS-770767 and [13C6]BMS-770767 for use in discovery biotransformation, human ADME and bioanalytical studies

The syntheses of isotopically labelled CB-1 antagonists for the treatment of obesity

Synthesis of isotopically labeled daclatasvir for use in human clinical studies

The syntheses of [14C]BMS-823778 for use in a human ADME clinical study and of [13CD3 13CD2]BMT-094817, a stable-isotope labeled standard of a newly detected human metabolite

Synthesis of stable isotope-labeled epothilone D using a degradation-reconstruction approach

Synthesis of a stable isotopically labeled universal surrogate peptide for use as an internal standard in LC-MS/MS bioanalysis of human IgG and Fc-fusion protein drug candidates

Synthesis of unlabelled and stable‐isotope–labelled glucuronide metabolites of dapagliflozin and synthesis of stable‐isotope–labelled dapagliflozin

Distinguishing a phosphate ester prodrug from its isobaric sulfate metabolite by mass spectrometry without the metabolite standard

An alternative and robust synthesis of [13C4]Baraclude® (entecavir)

An improved synthesis of [2-14C]2, 5-dichloropyrimidine

Carbon-14 labeled methyl 2-chloro-2-oxoacetate: a convenient carbon-14 labeled oxalyl chloride equivalent

A novel synthesis of [2-14C]2,5-dichloropyrimidine

LC-MS/MS bioanalysis of plasma 1, 14-tetradecanedioic acid and 1, 16-hexadecanedioic acid as candidate biomarkers for organic anion-transporting polypeptide mediated drug-drug interactions

Synthesis and stability of a carbon-14-labeled 3-hydroxy-3-methylglutaryl coenzyme-A reductase inhibitor

The syntheses and in vitro biotransformation studies of [14C]apixaban, a highly potent, selective, efficacious and orally bioavailable inhibitor of blood coagulation Factor Xa

Synthesis of [3α-3H] 17α-Hydroxy pregnenolone and [3α-3H] Pregnenolone

Synthesis of multi-labeled [14C]Aripiprazole

Carbon-14 labeling of Saxagliptin (BMS-477118)

Synthesis of carbon-14 and stable isotope labeled Avagacestat: a novel gamma secretase inhibitor for the treatment of Alzheimer's disease

Synthesis of [1,2-3H]ethylamine hydrochloride and [3H]-labeled apadenoson for a human ADME study

Overcoming bioanalytical challenges in an Onglyza(®) intravenous [(14)C]microdose absolute bioavailability study with accelerator MS

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