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Lessons from crystal structures of kainate receptors

Neuropharmacology, 2017-01, Vol.112 (Pt A), p.16-28

2017

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7‑Phenoxy-Substituted 3,4-Dihydro‑2H‑1,2,4-benzothiadiazine 1,1-Dioxides as Positive Allosteric Modulators of α‑Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptors with Nanomolar Potency

Journal of medicinal chemistry, 2018-01, Vol.61 (1), p.251-264

2018

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Exploring thienothiadiazine dioxides as isosteric analogues of benzo- and pyridothiadiazine dioxides in the search of new AMPA and kainate receptor positive allosteric modulators

European journal of medicinal chemistry, 2024-01, Vol.264, p.116036-116036, Article 116036

2024

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Tyr702 Is an Important Determinant of Agonist Binding and Domain Closure of the Ligand-Binding Core of GluR2

Molecular pharmacology, 2005-03, Vol.67 (3), p.703-713

2005

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Enhancing Action of Positive Allosteric Modulators through the Design of Dimeric Compounds

Journal of medicinal chemistry, 2018-06, Vol.61 (12), p.5279-5291

2018

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Lessons from more than 80 structures of the GluA2 ligand-binding domain in complex with agonists, antagonists and allosteric modulators

Neuropharmacology, 2011, Vol.60 (1), p.135-150

2011

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Identification and Structure-Function Study of Positive Allosteric Modulators of Kainate Receptors

Molecular pharmacology, 2017-06, Vol.91 (6), p.576-585

2017

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A pharmacological profile of the high-affinity GluK5 kainate receptor

European journal of pharmacology, 2016-10, Vol.788, p.315-320

2016

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Development of Thiochroman Dioxide Analogues of Benzothiadiazine Dioxides as New Positive Allosteric Modulators of α‑Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptors

ACS chemical neuroscience, 2021-07, Vol.12 (14), p.2679-2692

2021

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(S)‑2-Amino-3-(5-methyl-3-hydroxyisoxazol-4-yl)propanoic Acid (AMPA) and Kainate Receptor Ligands: Further Exploration of Bioisosteric Replacements and Structural and Biological Investigation

Journal of medicinal chemistry, 2018-03, Vol.61 (5), p.2124-2130

2018

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Crystal Structures of Potent Dimeric Positive Allosteric Modulators at the Ligand-Binding Domain of the GluA2 Receptor

ACS medicinal chemistry letters, 2019-03, Vol.10 (3), p.243-247

2019

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The ionotropic glutamate receptor GluA2 in complex with bicyclic pyrimidinedione-based compounds: when small compound modifications have distinct effects on binding interactions

ACS chemical neuroscience, 2020-06, Vol.11 (12), p.1791-1800

2020

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Structure and Affinity of Two Bicyclic Glutamate Analogues at AMPA and Kainate Receptors

ACS chemical neuroscience, 2017-09, Vol.8 (9), p.2056-2064

2017

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Synthesis and Pharmacology of Mono‑, Di‑, and Trialkyl-Substituted 7‑Chloro-3,4-dihydro‑2H‑1,2,4-benzothiadiazine 1,1-Dioxides Combined with X‑ray Structure Analysis to Understand the Unexpected Structure–Activity Relationship at AMPA Receptors

ACS chemical neuroscience, 2016-03, Vol.7 (3), p.378-390

2016

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Lessons from crystal structures of kainate receptors

7‑Phenoxy-Substituted 3,4-Dihydro‑2H‑1,2,4-benzothiadiazine 1,1-Dioxides as Positive Allosteric Modulators of α‑Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptors with Nanomolar Potency

Exploring thienothiadiazine dioxides as isosteric analogues of benzo- and pyridothiadiazine dioxides in the search of new AMPA and kainate receptor positive allosteric modulators

Tyr702 Is an Important Determinant of Agonist Binding and Domain Closure of the Ligand-Binding Core of GluR2

Enhancing Action of Positive Allosteric Modulators through the Design of Dimeric Compounds

Lessons from more than 80 structures of the GluA2 ligand-binding domain in complex with agonists, antagonists and allosteric modulators

Identification and Structure-Function Study of Positive Allosteric Modulators of Kainate Receptors

A pharmacological profile of the high-affinity GluK5 kainate receptor

Development of Thiochroman Dioxide Analogues of Benzothiadiazine Dioxides as New Positive Allosteric Modulators of α‑Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptors

(S)‑2-Amino-3-(5-methyl-3-hydroxyisoxazol-4-yl)propanoic Acid (AMPA) and Kainate Receptor Ligands: Further Exploration of Bioisosteric Replacements and Structural and Biological Investigation

Crystal Structures of Potent Dimeric Positive Allosteric Modulators at the Ligand-Binding Domain of the GluA2 Receptor

The ionotropic glutamate receptor GluA2 in complex with bicyclic pyrimidinedione-based compounds: when small compound modifications have distinct effects on binding interactions

Structure and Affinity of Two Bicyclic Glutamate Analogues at AMPA and Kainate Receptors

Synthesis and Pharmacology of Mono‑, Di‑, and Trialkyl-Substituted 7‑Chloro-3,4-dihydro‑2H‑1,2,4-benzothiadiazine 1,1-Dioxides Combined with X‑ray Structure Analysis to Understand the Unexpected Structure–Activity Relationship at AMPA Receptors

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