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Accessing Drug Metabolites via Transition-Metal Catalyzed C−H Oxidation: The Liver as Synthetic Inspiration

Angewandte Chemie (International ed.), 2016-11, Vol.55 (46), p.14218-14238

International ed. in English, 2016

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Quaternary Charge-Transfer Complex Enables Photoenzymatic Intermolecular Hydroalkylation of Olefins

Journal of the American Chemical Society, 2021-01, Vol.143 (1), p.97-102

2021

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Intermolecular Crossed [2 + 2] Cycloaddition Promoted by Visible-Light Triplet Photosensitization: Expedient Access to Polysubstituted 2‑Oxaspiro[3.3]heptanes

Journal of the American Chemical Society, 2021-03, Vol.143 (10), p.4055-4063

2021

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Synthetic strategy: natural products on demand

Nature chemistry, 2014-06, Vol.6 (6), p.460

Hamann, Lawrence G

2014

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Expedient access to saturated nitrogen heterocycles by photoredox cyclization of imino-tethered dihydropyridines

Chemical science (Cambridge), 2019-11, Vol.1 (41), p.9591-9596

2019

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Regioselective Synthesis and Slow-Release Suzuki–Miyaura Cross-Coupling of MIDA Boronate-Functionalized Isoxazoles and Triazoles

Journal of organic chemistry, 2011-12, Vol.76 (24), p.10241-10248

2011

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Discovery of a novel indole pharmacophore for the irreversible inhibition of myeloperoxidase (MPO)

Bioorganic & medicinal chemistry, 2020-06, Vol.28 (12), p.115548-115548, Article 115548

2020

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Die Erschließung von Wirkstoffmetaboliten durch übergangsmetallkatalysierte C-H-Oxidation: die Leber als Inspiration für die Synthese

Angewandte Chemie, 2016-11, Vol.128 (46), p.14430-14451

2016

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One-Pot Reductive Amination and Suzuki–Miyaura Cross-Coupling of Formyl Aryl and Heteroaryl MIDA Boronates in Array Format

Journal of organic chemistry, 2011-06, Vol.76 (12), p.4930-4940

2011

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Inhibitors of HIV-1 attachment: The discovery and structure–activity relationships of tetrahydroisoquinolines as replacements for the piperazine benzamide in the 3-glyoxylyl 6-azaindole pharmacophore

Bioorganic & medicinal chemistry letters, 2016-01, Vol.26 (1), p.160-167

2016

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2-Alkyloxazoles as potent and selective PI4KIIIβ inhibitors demonstrating inhibition of HCV replication

Bioorganic & medicinal chemistry letters, 2014-08, Vol.24 (16), p.3714-3718

2014

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One-Pot C–N/C–C Cross-Coupling of Methyliminodiacetic Acid Boronyl Arenes Enabled by Protective Enolization

Organic letters, 2012-11, Vol.14 (21), p.5578-5581

2012

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Synthesis and SAR of azolopyrimidines as potent and selective dipeptidyl peptidase-4 (DPP4) inhibitors for type 2 diabetes

Bioorganic & medicinal chemistry letters, 2010-08, Vol.20 (15), p.4395-4398

2010

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Substituted piperidinyl glycinyl 2-cyano-4,5-methano pyrrolidines as potent and stable dipeptidyl peptidase IV inhibitors

Bioorganic & medicinal chemistry letters, 2013-03, Vol.23 (6), p.1622-1625

2013

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Discovery of pyridyl sulfonamide 11-beta-hydroxysteroid dehydrogenase type 1 (11β-HSD1) inhibitors for the treatment of metabolic disorders

Bioorganic & medicinal chemistry letters, 2014-11, Vol.24 (21), p.5045-5049

2014

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Generation of 3,8-substituted 1,2,4-triazolopyridines as potent inhibitors of human 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD-1)

Bioorganic & medicinal chemistry letters, 2011-07, Vol.21 (14), p.4146-4149

2011

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A scalable synthesis of (1R,3S,5R)-2-(tert-butoxycarbonyl)-2-azabicyclo[3.1.0]hexane-3-carboxylic acid

Tetrahedron letters, 2013-12, Vol.54 (49), p.6722-6724

2013

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7-Oxopyrrolopyridine-derived DPP4 inhibitors—mitigation of CYP and hERG liabilities via introduction of polar functionalities in the active site

Bioorganic & medicinal chemistry letters, 2011-11, Vol.21 (22), p.6646-6651

2011

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Synthesis, SAR, and atropisomerism of imidazolopyrimidine DPP4 inhibitors

Bioorganic & medicinal chemistry letters, 2010-11, Vol.20 (21), p.6273-6276

2010

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Palladium-Catalyzed Microwave-Assisted Amination of 1-Bromonaphthalenes and 5- and 8-Bromoquinolines

Organic letters, 2003-03, Vol.5 (6), p.897-900

2003

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Potent non-nitrile dipeptidic dipeptidyl peptidase IV inhibitors

Bioorganic & medicinal chemistry, 2007-12, Vol.17 (23), p.6476-6480

2007

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Synthesis and SAR of tetrahydropyrrolo[1,2-b][1,2,5]thiadiazol-2(3H)-one 1,1-dioxide analogues as highly potent selective androgen receptor modulators

Bioorganic & medicinal chemistry letters, 2007-08, Vol.17 (16), p.4487-4490

2007

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Tandem optimization of target activity and elimination of mutagenic potential in a potent series of N-aryl bicyclic hydantoin-based selective androgen receptor modulators

Bioorganic & medicinal chemistry letters, 2007-04, Vol.17 (7), p.1860-1864

2007

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Pyridine amides as potent and selective inhibitors of 11β-hydroxysteroid dehydrogenase type 1

Bioorganic & medicinal chemistry, 2008-06, Vol.18 (11), p.3168-3172

2008

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Structure–activity relationships and sub-type selectivity in an oxabicyclic estrogen receptor α/β agonist scaffold

Bioorganic & medicinal chemistry letters, 2005-03, Vol.15 (5), p.1463-1466

2005

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Accessing Drug Metabolites via Transition-Metal Catalyzed C−H Oxidation: The Liver as Synthetic Inspiration

Quaternary Charge-Transfer Complex Enables Photoenzymatic Intermolecular Hydroalkylation of Olefins

Intermolecular Crossed [2 + 2] Cycloaddition Promoted by Visible-Light Triplet Photosensitization: Expedient Access to Polysubstituted 2‑Oxaspiro[3.3]heptanes

Synthetic strategy: natural products on demand

Expedient access to saturated nitrogen heterocycles by photoredox cyclization of imino-tethered dihydropyridines

Regioselective Synthesis and Slow-Release Suzuki–Miyaura Cross-Coupling of MIDA Boronate-Functionalized Isoxazoles and Triazoles

Discovery of a novel indole pharmacophore for the irreversible inhibition of myeloperoxidase (MPO)

Die Erschließung von Wirkstoffmetaboliten durch übergangsmetallkatalysierte C-H-Oxidation: die Leber als Inspiration für die Synthese

One-Pot Reductive Amination and Suzuki–Miyaura Cross-Coupling of Formyl Aryl and Heteroaryl MIDA Boronates in Array Format

Inhibitors of HIV-1 attachment: The discovery and structure–activity relationships of tetrahydroisoquinolines as replacements for the piperazine benzamide in the 3-glyoxylyl 6-azaindole pharmacophore

2-Alkyloxazoles as potent and selective PI4KIIIβ inhibitors demonstrating inhibition of HCV replication

One-Pot C–N/C–C Cross-Coupling of Methyliminodiacetic Acid Boronyl Arenes Enabled by Protective Enolization

Synthesis and SAR of azolopyrimidines as potent and selective dipeptidyl peptidase-4 (DPP4) inhibitors for type 2 diabetes

Substituted piperidinyl glycinyl 2-cyano-4,5-methano pyrrolidines as potent and stable dipeptidyl peptidase IV inhibitors

Discovery of pyridyl sulfonamide 11-beta-hydroxysteroid dehydrogenase type 1 (11β-HSD1) inhibitors for the treatment of metabolic disorders

Generation of 3,8-substituted 1,2,4-triazolopyridines as potent inhibitors of human 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD-1)

A scalable synthesis of (1R,3S,5R)-2-(tert-butoxycarbonyl)-2-azabicyclo[3.1.0]hexane-3-carboxylic acid

7-Oxopyrrolopyridine-derived DPP4 inhibitors—mitigation of CYP and hERG liabilities via introduction of polar functionalities in the active site

Synthesis, SAR, and atropisomerism of imidazolopyrimidine DPP4 inhibitors

Palladium-Catalyzed Microwave-Assisted Amination of 1-Bromonaphthalenes and 5- and 8-Bromoquinolines

Potent non-nitrile dipeptidic dipeptidyl peptidase IV inhibitors

Synthesis and SAR of tetrahydropyrrolo[1,2-b][1,2,5]thiadiazol-2(3H)-one 1,1-dioxide analogues as highly potent selective androgen receptor modulators

Tandem optimization of target activity and elimination of mutagenic potential in a potent series of N-aryl bicyclic hydantoin-based selective androgen receptor modulators

Pyridine amides as potent and selective inhibitors of 11β-hydroxysteroid dehydrogenase type 1

Structure–activity relationships and sub-type selectivity in an oxabicyclic estrogen receptor α/β agonist scaffold

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