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Ruthenium Half-Sandwich Complexes Bound to Protein Kinase Pim-1

Angewandte Chemie (International ed.), 2006-02, Vol.45 (10), p.1580-1585

2006

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Discovery of Novel, Induced-Pocket Binding Oxazolidinones as Potent, Selective, and Orally Bioavailable Tankyrase Inhibitors

Journal of medicinal chemistry, 2013-06, Vol.56 (11), p.4320-4342

2013

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A Modular Synthesis of the Lamellarins: Total Synthesis of Lamellarin G Trimethyl Ether

Journal of organic chemistry, 2004-04, Vol.69 (7), p.2362-2366

2004

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Inhibition of Inactive States of Tetrodotoxin-Sensitive Sodium Channels Reduces Spontaneous Firing of C-Fiber Nociceptors and Produces Analgesia in Formalin and Complete Freund's Adjuvant Models of Pain

PloS one, 2015-09, Vol.10 (9), p.e0138140

2015

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Ruthenium half-sandwich complexes as protein kinase inhibitors: derivatization of the pyridocarbazole pharmacophore ligand

Organic & biomolecular chemistry, 2007-01, Vol.5 (8), p.1218-1227

2007

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Sulfonamides as Selective NaV1.7 Inhibitors: Optimizing Potency and Pharmacokinetics to Enable in Vivo Target Engagement

ACS medicinal chemistry letters, 2016-12, Vol.7 (12), p.1062-1067

2016

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Structure-Based Design of 2‑Aminopyridine Oxazolidinones as Potent and Selective Tankyrase Inhibitors

ACS medicinal chemistry letters, 2013-12, Vol.4 (12), p.1218-1223

2013

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Ruthenium Half-Sandwich Complexes as Protein Kinase Inhibitors: An N-Succinimidyl Ester for Rapid Derivatizations of the Cyclopentadienyl Moiety

Organic letters, 2006-11, Vol.8 (24), p.5465-5468

2006

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Rapid Access to Unexplored Chemical Space by Ligand Scanning around a Ruthenium Center: Discovery of Potent and Selective Protein Kinase Inhibitors

Journal of the American Chemical Society, 2006-01, Vol.128 (3), p.877-884

2006

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Sulfonamides as Selective NaV1.7 Inhibitors: Optimizing Potency and Pharmacokinetics While Mitigating Metabolic Liabilities

Journal of medicinal chemistry, 2017-07, Vol.60 (14), p.5969-5989

2017

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Exploring Chemical Space with Organometallics: Ruthenium Complexes as Protein Kinase Inhibitors

Synlett, 2007-05, Vol.2007 (8), p.1177-1189

2007

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An Organometallic Inhibitor for Glycogen Synthase Kinase 3

Journal of the American Chemical Society, 2004-10, Vol.126 (42), p.13594-13595

2004

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The discovery of benzoxazine sulfonamide inhibitors of NaV1.7: Tools that bridge efficacy and target engagement

Bioorganic & medicinal chemistry letters, 2017-08, Vol.27 (15), p.3477-3485

2017

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Pyrido[2,3-a]pyrrolo[3,4-c]carbazole-5,7(6H)-diones: Synthesis, Cyclometalation, and Protein Kinase Inhibition

Synthesis (Stuttgart), 2005-06, Vol.2005 (9), p.1521-1527

2005

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Switching on a Signaling Pathway with an Organoruthenium Complex

Angewandte Chemie (International ed.), 2005-03, Vol.44 (13), p.1984-1987

2005

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Application of a Parallel Synthetic Strategy in the Discovery of Biaryl Acyl Sulfonamides as Efficient and Selective Na V 1.7 Inhibitors

Journal of medicinal chemistry, 2016-09, Vol.59 (17), p.7818-7839

2016

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Abstract 1621: Discovery of pyridyl pyrrolopyridinones as potent and selective CK1γ inhibitors

Cancer research (Chicago, Ill.), 2014-10, Vol.74 (19_Supplement), p.1621-1621

2014

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Corrigendum to “Purinylpyridinylamino-based DFG-in/αC-helix-out B-Raf inhibitors: Applying mutant versus wild-type B-Raf selectivity indices for compound profiling” [Bioorg. Med. Chem. 24 (2016) 2215–2234]

Bioorganic & medicinal chemistry, 2016-07, Vol.24 (13), p.3093-3093

2016

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The discovery of aminopyrazines as novel, potent Na(v)1.7 antagonists: hit-to-lead identification and SAR

Bioorganic & medicinal chemistry letters, 2012-03, Vol.22 (5), p.2033-2042

2012

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An unusual dehalogenation in the Suzuki coupling of 4-bromopyrrole-2-carboxylates

Tetrahedron letters, 2003-01, Vol.44 (3), p.427-430

2003

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2-Phenylamino-6-cyano-1H-benzimidazole-based isoform selective casein kinase 1 gamma (CK1γ) inhibitors

Bioorganic & medicinal chemistry letters, 2012-09, Vol.22 (17)

2012

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Sulfonamides as Selective Na V 1.7 Inhibitors: Optimizing Potency and Pharmacokinetics to Enable in Vivo Target Engagement

ACS medicinal chemistry letters, 2016-12, Vol.7 (12), p.1062-1067

2016

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Correction to “Sulfonamides as Selective NaV1.7 Inhibitors: Optimizing Potency and Pharmacokinetics to Enable in Vivo Target Engagement”

ACS medicinal chemistry letters, 2017-03, Vol.8 (3), p.378-378

2017

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Correction to "Sulfonamides as Selective Na V 1.7 Inhibitors: Optimizing Potency and Pharmacokinetics to Enable in Vivo Target Engagement"

ACS medicinal chemistry letters, 2017-03, Vol.8 (3), p.378-378

2017

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Structure-Based Design of Potent and Selective CK1γ Inhibitors

ACS medicinal chemistry letters, 2012-12, Vol.3 (12), p.1059-1064

2012

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Ruthenium Half-Sandwich Complexes Bound to Protein Kinase Pim-1

Discovery of Novel, Induced-Pocket Binding Oxazolidinones as Potent, Selective, and Orally Bioavailable Tankyrase Inhibitors

A Modular Synthesis of the Lamellarins: Total Synthesis of Lamellarin G Trimethyl Ether

Inhibition of Inactive States of Tetrodotoxin-Sensitive Sodium Channels Reduces Spontaneous Firing of C-Fiber Nociceptors and Produces Analgesia in Formalin and Complete Freund's Adjuvant Models of Pain

Ruthenium half-sandwich complexes as protein kinase inhibitors: derivatization of the pyridocarbazole pharmacophore ligand

Sulfonamides as Selective NaV1.7 Inhibitors: Optimizing Potency and Pharmacokinetics to Enable in Vivo Target Engagement

Structure-Based Design of 2‑Aminopyridine Oxazolidinones as Potent and Selective Tankyrase Inhibitors

Ruthenium Half-Sandwich Complexes as Protein Kinase Inhibitors: An N-Succinimidyl Ester for Rapid Derivatizations of the Cyclopentadienyl Moiety

Rapid Access to Unexplored Chemical Space by Ligand Scanning around a Ruthenium Center: Discovery of Potent and Selective Protein Kinase Inhibitors

Sulfonamides as Selective NaV1.7 Inhibitors: Optimizing Potency and Pharmacokinetics While Mitigating Metabolic Liabilities

Exploring Chemical Space with Organometallics: Ruthenium Complexes as Protein Kinase Inhibitors

An Organometallic Inhibitor for Glycogen Synthase Kinase 3

The discovery of benzoxazine sulfonamide inhibitors of NaV1.7: Tools that bridge efficacy and target engagement

Pyrido[2,3-a]pyrrolo[3,4-c]carbazole-5,7(6H)-diones: Synthesis, Cyclometalation, and Protein Kinase Inhibition

Switching on a Signaling Pathway with an Organoruthenium Complex

Application of a Parallel Synthetic Strategy in the Discovery of Biaryl Acyl Sulfonamides as Efficient and Selective Na V 1.7 Inhibitors

Abstract 1621: Discovery of pyridyl pyrrolopyridinones as potent and selective CK1γ inhibitors

Corrigendum to “Purinylpyridinylamino-based DFG-in/αC-helix-out B-Raf inhibitors: Applying mutant versus wild-type B-Raf selectivity indices for compound profiling” [Bioorg. Med. Chem. 24 (2016) 2215–2234]

The discovery of aminopyrazines as novel, potent Na(v)1.7 antagonists: hit-to-lead identification and SAR

An unusual dehalogenation in the Suzuki coupling of 4-bromopyrrole-2-carboxylates

2-Phenylamino-6-cyano-1H-benzimidazole-based isoform selective casein kinase 1 gamma (CK1γ) inhibitors

Sulfonamides as Selective Na V 1.7 Inhibitors: Optimizing Potency and Pharmacokinetics to Enable in Vivo Target Engagement

Correction to “Sulfonamides as Selective NaV1.7 Inhibitors: Optimizing Potency and Pharmacokinetics to Enable in Vivo Target Engagement”

Correction to "Sulfonamides as Selective Na V 1.7 Inhibitors: Optimizing Potency and Pharmacokinetics to Enable in Vivo Target Engagement"

Structure-Based Design of Potent and Selective CK1γ Inhibitors

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