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(−)-Rhazinilam and the diphenylpyridazinone NSC 613241: Two compounds inducing the formation of morphologically similar tubulin spirals but binding apparently to two distinct sites on tubulin

Archives of biochemistry and biophysics, 2016-08, Vol.604, p.63-73

2016

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Insight on [1,3]thiazolo[4,5-e]isoindoles as tubulin polymerization inhibitors

European journal of medicinal chemistry, 2021-02, Vol.212, p.113122, Article 113122

2021

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12,13-Aziridinyl Epothilones. Stereoselective Synthesis of Trisubstituted Olefinic Bonds from Methyl Ketones and Heteroaromatic Phosphonates and Design, Synthesis, and Biological Evaluation of Potent Antitumor Agents

Journal of the American Chemical Society, 2017-05, Vol.139 (21), p.7318-7334

2017

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Total Synthesis of Potent Antitumor Macrolide (-)-Zampanolide: An Oxidative Intramolecular Cyclization-Based Strategy

European journal of organic chemistry, 2012-08, Vol.2012 (22), p.4130-4139

2012

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New Arylthioindoles and Related Bioisosteres at the Sulfur Bridging Group. 4. Synthesis, Tubulin Polymerization, Cell Growth Inhibition, and Molecular Modeling Studies

Journal of medicinal chemistry, 2009-12, Vol.52 (23), p.7512-7527

2009

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Interactions of Halichondrin B and Eribulin with Tubulin

Journal of chemical information and modeling, 2011-06, Vol.51 (6), p.1393-1404

2011

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Enantioselective Synthesis of (+)-Chamaecypanone C: A Novel Microtubule Inhibitor

Angewandte Chemie (International ed.), 2009-01, Vol.48 (8), p.1494-1497

2009

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Comparison of the Activities of the Truncated Halichondrin B Analog NSC 707389 (E7389) with Those of the Parent Compound and a Proposed Binding Site on Tubulin

Molecular pharmacology, 2006-12, Vol.70 (6), p.1866-1875

2006

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Deciphering the key heterocyclic scaffolds in targeting microtubules, kinases and carbonic anhydrases for cancer drug development

Pharmacology & therapeutics (Oxford), 2021-09, Vol.225, p.107860, Article 107860

2021

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Laulimalide and Paclitaxel: A Comparison of Their Effects on Tubulin Assembly and Their Synergistic Action When Present Simultaneously

Molecular pharmacology, 2004-07, Vol.66 (1), p.113-121

2004

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Actin is the primary cellular receptor of bistramide A

Nature chemical biology, 2005-12, Vol.1 (7), p.383-388

2005

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(−)-RHAZINILAM AND THE DIPHENYLPYRIDAZINONE NSC 613241: TWO COMPOUNDS INDUCING THE FORMATION OF MORPHOLOGICALLY SIMILAR TUBULIN SPIRALS BUT BINDING APPARENTLY TO TWO DISTINCT SITES ON TUBULIN1,2

Archives of biochemistry and biophysics, 2016-06, Vol.604, p.63-73

2016

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Intracellular Activation and Deactivation of Tasidotin, an Analog of Dolastatin 15: Correlation with Cytotoxicity

Molecular pharmacology, 2009-01, Vol.75 (1), p.218-226

2009

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Corrigendum to “The interaction of spongistatin 1 with tubulin” [Arch. Biochem. Biophys. 727 (2022) 109296 (7 pages)]

Archives of biochemistry and biophysics, 2022-11, Vol.730, p.109412-109412, Article 109412

2022

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Drug-Linker Constructs Bearing Unique Dual-Mechanism Tubulin Binding Payloads Tethered through Cleavable and Non-Cleavable Linkers

Tetrahedron, 2024-11, p.134350, Article 134350

2024

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Interaction of a Cyclostreptin Analogue with the Microtubule Taxoid Site: The Covalent Reaction Rapidly Follows Binding

Journal of natural products (Washington, D.C.), 2008-03, Vol.71 (3), p.370-374

2008

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The interaction of spongistatin 1 with tubulin

Archives of biochemistry and biophysics, 2022-09, Vol.727, p.109296-109296, Article 109296

2022

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Design, synthesis and biological evaluation of 2-phenyl indole analogues of OXi8006 as colchicine site inhibitors of tubulin polymerization and vascular disrupting agents

Bioorganic & medicinal chemistry, 2024-11, p.117981, Article 117981

2024

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Interaction of diazonamide A with tubulin

Archives of biochemistry and biophysics, 2020-02, Vol.680, p.108217-108217, Article 108217

2020

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Development of [1,2]oxazoloisoindoles tubulin polymerization inhibitors: Further chemical modifications and potential therapeutic effects against lymphomas

European journal of medicinal chemistry, 2022-12, Vol.243, p.114744-114744, Article 114744

2022

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Novel pyrazolo[4,3-d]pyrimidine microtubule targeting agents (MTAs): Synthesis, structure–activity relationship, in vitro and in vivo evaluation as antitumor agents

Bioorganic & medicinal chemistry letters, 2021-06, Vol.41, p.127923-127923, Article 127923

2021

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(â)-Doliculide, a New Macrocyclic Depsipeptide Enhancer of Actin Assembly

The Journal of biological chemistry, 2002-08, Vol.277 (35), p.32165-32171

2002

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Abstract 6244: Design, synthesis, and structure-activity relationships of substituted pyrido[3,2- d ]pyrimidines as microtubule targeting agents and anti-cancer agents

Cancer research (Chicago, Ill.), 2023-04, Vol.83 (7_Supplement), p.6244-6244

2023

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Induction of Ferroptosis in Glioblastoma and Ovarian Cancers by a New Pyrrole Tubulin Assembly Inhibitor

Journal of medicinal chemistry, 2022-12, Vol.65 (23), p.15805-15818

2022

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Novel pyrazolo4,3-dpyrimidine microtubule targeting agents (MTAs): Synthesis, structure-activity relationship, in vitro and in vivo evaluation as antitumor agents

Bioorganic & medicinal chemistry letters, 2021-06, Vol.41, p.127923

2021

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(−)-Rhazinilam and the diphenylpyridazinone NSC 613241: Two compounds inducing the formation of morphologically similar tubulin spirals but binding apparently to two distinct sites on tubulin

Insight on [1,3]thiazolo[4,5-e]isoindoles as tubulin polymerization inhibitors

12,13-Aziridinyl Epothilones. Stereoselective Synthesis of Trisubstituted Olefinic Bonds from Methyl Ketones and Heteroaromatic Phosphonates and Design, Synthesis, and Biological Evaluation of Potent Antitumor Agents

Total Synthesis of Potent Antitumor Macrolide (-)-Zampanolide: An Oxidative Intramolecular Cyclization-Based Strategy

New Arylthioindoles and Related Bioisosteres at the Sulfur Bridging Group. 4. Synthesis, Tubulin Polymerization, Cell Growth Inhibition, and Molecular Modeling Studies

Interactions of Halichondrin B and Eribulin with Tubulin

Enantioselective Synthesis of (+)-Chamaecypanone C: A Novel Microtubule Inhibitor

Comparison of the Activities of the Truncated Halichondrin B Analog NSC 707389 (E7389) with Those of the Parent Compound and a Proposed Binding Site on Tubulin

Deciphering the key heterocyclic scaffolds in targeting microtubules, kinases and carbonic anhydrases for cancer drug development

Laulimalide and Paclitaxel: A Comparison of Their Effects on Tubulin Assembly and Their Synergistic Action When Present Simultaneously

Actin is the primary cellular receptor of bistramide A

(−)-RHAZINILAM AND THE DIPHENYLPYRIDAZINONE NSC 613241: TWO COMPOUNDS INDUCING THE FORMATION OF MORPHOLOGICALLY SIMILAR TUBULIN SPIRALS BUT BINDING APPARENTLY TO TWO DISTINCT SITES ON TUBULIN1,2

Intracellular Activation and Deactivation of Tasidotin, an Analog of Dolastatin 15: Correlation with Cytotoxicity

Corrigendum to “The interaction of spongistatin 1 with tubulin” [Arch. Biochem. Biophys. 727 (2022) 109296 (7 pages)]

Drug-Linker Constructs Bearing Unique Dual-Mechanism Tubulin Binding Payloads Tethered through Cleavable and Non-Cleavable Linkers

Interaction of a Cyclostreptin Analogue with the Microtubule Taxoid Site: The Covalent Reaction Rapidly Follows Binding

The interaction of spongistatin 1 with tubulin

Design, synthesis and biological evaluation of 2-phenyl indole analogues of OXi8006 as colchicine site inhibitors of tubulin polymerization and vascular disrupting agents

Interaction of diazonamide A with tubulin

Development of [1,2]oxazoloisoindoles tubulin polymerization inhibitors: Further chemical modifications and potential therapeutic effects against lymphomas

Novel pyrazolo[4,3-d]pyrimidine microtubule targeting agents (MTAs): Synthesis, structure–activity relationship, in vitro and in vivo evaluation as antitumor agents

(â)-Doliculide, a New Macrocyclic Depsipeptide Enhancer of Actin Assembly

Abstract 6244: Design, synthesis, and structure-activity relationships of substituted pyrido[3,2- d ]pyrimidines as microtubule targeting agents and anti-cancer agents

Induction of Ferroptosis in Glioblastoma and Ovarian Cancers by a New Pyrrole Tubulin Assembly Inhibitor

Novel pyrazolo4,3-dpyrimidine microtubule targeting agents (MTAs): Synthesis, structure-activity relationship, in vitro and in vivo evaluation as antitumor agents

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