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Thiazole in the targeted anticancer drug discovery

Future medicinal chemistry, 2019-08, Vol.11 (16), p.1929-1952

2019

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Identification of a novel antifungal backbone of naphthalimide thiazoles with synergistic potential for chemical and dynamic treatment

Future medicinal chemistry, 2021-12, Vol.13 (23), p.2047-2067

2021

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Synthesis and biological evaluation of aminomethyl and alkoxymethyl derivatives as carbonic anhydrase, acetylcholinesterase and butyrylcholinesterase inhibitors

Journal of enzyme inhibition and medicinal chemistry, 2017-01, Vol.32 (1), p.1174-1182

2017

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4-Adamantyl-(2-(arylidene)hydrazinyl)thiazoles as potential antidiabetic agents: experimental and docking studies

Future medicinal chemistry, 2023-04, Vol.15 (7), p.599-613

2023

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Novel N -bridged pyrazole-1-carbothioamides with potential antiproliferative activity: design, synthesis, in vitro and in silico studies

Future medicinal chemistry, 2021-10, Vol.13 (20), p.1743-1766

2021

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Chemical modification of Arthrobacter sarcosine oxidase by N-methylisothiazolinone reduces reactivity toward oxygen

Bioscience, biotechnology, and biochemistry, 2024-05, Vol.88 (6), p.630-636

2024

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Synthesis of 4-benzyl-1,3-thiazole derivatives as potential anti-inflammatory agents: An analogue-based drug design approach

Journal of enzyme inhibition and medicinal chemistry, 2009-06, Vol.24 (3), p.890-897

2009

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Efficacy and safety evaluation of avatrombopag in immune thrombocytopenia: analyses of a phase III study and long-term extension

Platelets (Edinburgh), 2022-02, Vol.33 (2), p.257-264

2022

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Novel xylenyl-spaced bis-thiazoles/thiazines: synthesis, biological profile as herpes simplex virus type 1 inhibitors and in silico simulations

Future medicinal chemistry, 2024-01, Vol.16 (1), p.27-41

2024

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Discovery of new thymol-3,4-disubstituted thiazole hybrids as dual COX-2/5-LOX inhibitors with in vivo proof

Journal of enzyme inhibition and medicinal chemistry, 2024-12, Vol.39 (1), p.2309171-2309171

2024

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Synthesis of new 1,3-thiazol derivatives of maleopimaric acid as anticancer, antibacterial and antifungal agents

Natural product research, 2021-04, Vol.35 (8), p.1340-1348

2021

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Synthesis of hydrazinyl-thiazole ester derivatives, in vitro trypanocidal and leishmanicidal activities

Future medicinal chemistry, 2024-02, Vol.16 (3), p.221-238

2024

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Synthesis and biological evaluation of thiazole derivatives as LbSOD inhibitors

Journal of enzyme inhibition and medicinal chemistry, 2019-01, Vol.34 (1), p.333-342

2019

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Masitinib for the treatment of mild to moderate Alzheimer's disease

Expert review of neurotherapeutics, 2015-06, Vol.15 (6), p.587-596

2015

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Imidazothiazole-based potent inhibitors of V600E-B-RAF kinase with promising anti-melanoma activity: biological and computational studies

Journal of enzyme inhibition and medicinal chemistry, 2020-01, Vol.35 (1), p.1712-1726

2020

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Benzo[ d ]thiazole-2-carboxamides as new antituberculosis chemotypes inhibiting mycobacterial ATP phosphoribosyl transferase

Future medicinal chemistry, 2022-12, Vol.14 (24), p.1847-1864

2022

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New pyrazolyl-thiazolidinone/thiazole derivatives as celecoxib/dasatinib analogues with selective COX-2, HER-2 and EGFR inhibitory effects: design, synthesis, anti-inflammatory/anti-proliferative activities, apoptosis, molecular modelling and ADME studies

Journal of enzyme inhibition and medicinal chemistry, 2023-12, Vol.38 (1), p.2281262-2281262

2023

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Inhibition studies on a panel of human carbonic anhydrases with N1-substituted secondary sulfonamides incorporating thiazolinone or imidazolone-indole tails

Journal of enzyme inhibition and medicinal chemistry, 2018-01, Vol.33 (1), p.629-638

2018

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Selective CDK9 degradation using a proteolysis-targeting chimera (PROTAC) strategy

Future medicinal chemistry, 2022-01, Vol.14 (3), p.131-134

2022

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Synthesis, antiviral activity, preliminary pharmacokinetics and structural parameters of thiazolide amine salts

Future medicinal chemistry, 2021-10, Vol.13 (20), p.1731-1741

2021

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Isatin thiazoline hybrids as dual inhibitors of HIV-1 reverse transcriptase

Journal of enzyme inhibition and medicinal chemistry, 2017-01, Vol.32 (1), p.130-136

2017

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Triad pyrazole-thiazole-coumarin heterocyclic core effectively inhibit HSP and drive cancer cells to apoptosis

Journal of biomolecular structure & dynamics, 2023, Vol.41 (23), p.14382-14397

2023

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Synthesis, antimicrobial and anticonvulsant screening of small library of tetrahydro-2H-thiopyran-4-yl based thiazoles and selenazoles

Journal of enzyme inhibition and medicinal chemistry, 2016-11, Vol.31 (sup2), p.24-39

2016

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Design, synthesis and cytotoxic evaluation of novel bis-thiazole derivatives as preferential Pim1 kinase inhibitors with in vivo and in silico study

Journal of enzyme inhibition and medicinal chemistry, 2023-12, Vol.38 (1), p.2166936-2166936

2023

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A new thiodiketopiperzaine from the marine sponge Tedania sp

Natural product research, 2020-04, Vol.34 (8), p.1113-1117

2020

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Thiazole in the targeted anticancer drug discovery

Identification of a novel antifungal backbone of naphthalimide thiazoles with synergistic potential for chemical and dynamic treatment

Synthesis and biological evaluation of aminomethyl and alkoxymethyl derivatives as carbonic anhydrase, acetylcholinesterase and butyrylcholinesterase inhibitors

4-Adamantyl-(2-(arylidene)hydrazinyl)thiazoles as potential antidiabetic agents: experimental and docking studies

Novel N -bridged pyrazole-1-carbothioamides with potential antiproliferative activity: design, synthesis, in vitro and in silico studies

Chemical modification of Arthrobacter sarcosine oxidase by N-methylisothiazolinone reduces reactivity toward oxygen

Synthesis of 4-benzyl-1,3-thiazole derivatives as potential anti-inflammatory agents: An analogue-based drug design approach

Efficacy and safety evaluation of avatrombopag in immune thrombocytopenia: analyses of a phase III study and long-term extension

Novel xylenyl-spaced bis-thiazoles/thiazines: synthesis, biological profile as herpes simplex virus type 1 inhibitors and in silico simulations

Discovery of new thymol-3,4-disubstituted thiazole hybrids as dual COX-2/5-LOX inhibitors with in vivo proof

Synthesis of new 1,3-thiazol derivatives of maleopimaric acid as anticancer, antibacterial and antifungal agents

Synthesis of hydrazinyl-thiazole ester derivatives, in vitro trypanocidal and leishmanicidal activities

Synthesis and biological evaluation of thiazole derivatives as LbSOD inhibitors

Masitinib for the treatment of mild to moderate Alzheimer's disease

Imidazothiazole-based potent inhibitors of V600E-B-RAF kinase with promising anti-melanoma activity: biological and computational studies

Benzo[ d ]thiazole-2-carboxamides as new antituberculosis chemotypes inhibiting mycobacterial ATP phosphoribosyl transferase

New pyrazolyl-thiazolidinone/thiazole derivatives as celecoxib/dasatinib analogues with selective COX-2, HER-2 and EGFR inhibitory effects: design, synthesis, anti-inflammatory/anti-proliferative activities, apoptosis, molecular modelling and ADME studies

Inhibition studies on a panel of human carbonic anhydrases with N1-substituted secondary sulfonamides incorporating thiazolinone or imidazolone-indole tails

Selective CDK9 degradation using a proteolysis-targeting chimera (PROTAC) strategy

Synthesis, antiviral activity, preliminary pharmacokinetics and structural parameters of thiazolide amine salts

Isatin thiazoline hybrids as dual inhibitors of HIV-1 reverse transcriptase

Triad pyrazole-thiazole-coumarin heterocyclic core effectively inhibit HSP and drive cancer cells to apoptosis

Synthesis, antimicrobial and anticonvulsant screening of small library of tetrahydro-2H-thiopyran-4-yl based thiazoles and selenazoles

Design, synthesis and cytotoxic evaluation of novel bis-thiazole derivatives as preferential Pim1 kinase inhibitors with in vivo and in silico study

A new thiodiketopiperzaine from the marine sponge Tedania sp

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