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Preliminary Structure–Activity Relationships and Biological Evaluation of Novel Antitubercular Indolecarboxamide Derivatives Against Drug-Susceptible and Drug-Resistant Mycobacterium tuberculosis Strains

Journal of medicinal chemistry, 2013-05, Vol.56 (10), p.4093-4103

2013

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Inhibitors of the sulfur assimilation pathway in bacterial pathogens as enhancers of antibiotic therapy

Current medicinal chemistry, 2015-01, Vol.22 (2), p.187-213

2015

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Nitric oxide-releasing cyclodextrins as biodegradable antibacterial scaffolds: a patent evaluation of US2019343869(A1)

Expert opinion on therapeutic patents, 2020-12, Vol.30 (12), p.901-905

Pieroni, Marco

2020

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Inhibitors of O-Acetylserine Sulfhydrylase with a Cyclopropane-Carboxylic Acid Scaffold Are Effective Colistin Adjuvants in Gram Negative Bacteria

Pharmaceuticals (Basel, Switzerland), 2022-06, Vol.15 (6), p.766

2022

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Refining the structure−activity relationships of 2-phenylcyclopropane carboxylic acids as inhibitors of O-acetylserine sulfhydrylase isoforms

Journal of enzyme inhibition and medicinal chemistry, 2019-01, Vol.34 (1), p.31-43

2019

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Discovery of Substituted (2-Aminooxazol-4-yl)Isoxazole-3-carboxylic Acids as Inhibitors of Bacterial Serine Acetyltransferase in the Quest for Novel Potential Antibacterial Adjuvants

Pharmaceuticals (Basel, Switzerland), 2021-02, Vol.14 (2), p.174

2021

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Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand-based drug design

Journal of enzyme inhibition and medicinal chemistry, 2018-01, Vol.33 (1), p.1444-1452

2018

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Discovering a new class of antifungal agents that selectively inhibits microbial carbonic anhydrases

Journal of enzyme inhibition and medicinal chemistry, 2018-01, Vol.33 (1), p.1537-1544

2018

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Pyrido[1,2-a]benzimidazole-Based Agents Active Against Tuberculosis (TB), Multidrug-Resistant (MDR) TB and Extensively Drug-Resistant (XDR) TB

ChemMedChem, 2011-02, Vol.6 (2), p.334-342

2011

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Derivatives of 3-isoxazolecarboxylic acid esters: a potent and selective compound class against replicating and nonreplicating Mycobacterium tuberculosis

Current topics in medicinal chemistry, 2012-04, Vol.12 (7), p.729-734

2012

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Identification of Human Alanine–Glyoxylate Aminotransferase Ligands as Pharmacological Chaperones for Variants Associated with Primary Hyperoxaluria Type 1

Journal of medicinal chemistry, 2022-07, Vol.65 (14), p.9718-9734

2022

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Substituted N‑Phenyl-5-(2-(phenylamino)thiazol-4-yl)isoxazole-3-carboxamides Are Valuable Antitubercular Candidates that Evade Innate Efflux Machinery

Journal of medicinal chemistry, 2017-08, Vol.60 (16), p.7108-7122

2017

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Design, synthesis and investigation on the structure–activity relationships of N-substituted 2-aminothiazole derivatives as antitubercular agents

European journal of medicinal chemistry, 2014-01, Vol.72, p.26-34

2014

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Rational Design and Synthesis of Thioridazine Analogues as Enhancers of the Antituberculosis Therapy

Journal of medicinal chemistry, 2015-08, Vol.58 (15), p.5842-5853

2015

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Integration of Enhanced Sampling Methods with Saturation Transfer Difference Experiments to Identify Protein Druggable Pockets

Journal of chemical information and modeling, 2018-03, Vol.58 (3), p.710-723

2018

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2‑Aminooxazole as a Novel Privileged Scaffold in Antitubercular Medicinal Chemistry

ACS medicinal chemistry letters, 2020-07, Vol.11 (7), p.1435-1441

2020

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Chemical Probes to Investigate Central Nervous System Disorders: Design, Synthesis and Mechanism of Action of a Potent Human Serine Racemase Inhibitor

ACS medicinal chemistry letters, 2024-08, Vol.15 (8), p.1298-1305

2024

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Rational Design, Synthesis, and Preliminary Structure–Activity Relationships of α‑Substituted-2-Phenylcyclopropane Carboxylic Acids as Inhibitors of Salmonella typhimurium O‑Acetylserine Sulfhydrylase

Journal of medicinal chemistry, 2016-03, Vol.59 (6), p.2567-2578

2016

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Discovery of antitubercular 2,4-diphenyl-1H-imidazoles from chemical library repositioning and rational design

European journal of medicinal chemistry, 2015-07, Vol.100, p.44-49

2015

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Expanding the knowledge around antitubercular 5-(2-aminothiazol-4-yl)isoxazole-3-carboxamides: Hit–to–lead optimization and release of a novel antitubercular chemotype via scaffold derivatization

European journal of medicinal chemistry, 2023-01, Vol.245 (Pt 2), p.114916-114916, Article 114916

2023

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Discovery of New Potential Anti-Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target-Focused Repurposing Approaches

ChemMedChem, 2016-09, Vol.11 (17), p.1904-1914

2016

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Further insights into the SAR of α-substituted cyclopropylamine derivatives as inhibitors of histone demethylase KDM1A

European journal of medicinal chemistry, 2015-03, Vol.92, p.377-386

2015

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Preliminary structure−activity relationships analysis on N-(3,5-dichlorophenyl)-4,5-dihydronaphtho[1,2-d]thiazol-2-amine, a disruptor of mycobacterial energetics

Medicinal chemistry research, 2024-03, Vol.33 (3), p.518-531

2024

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Rational Design of 5-Phenyl-3-isoxazolecarboxylic Acid Ethyl Esters as Growth Inhibitors of Mycobacterium tuberculosis. A Potent and Selective Series for Further Drug Development

Journal of medicinal chemistry, 2010-01, Vol.53 (2), p.678-688

2010

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Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O‑Acetyltransferase Inhibitor

ACS medicinal chemistry letters, 2020-05, Vol.11 (5), p.790-797

2020

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Preliminary Structure–Activity Relationships and Biological Evaluation of Novel Antitubercular Indolecarboxamide Derivatives Against Drug-Susceptible and Drug-Resistant Mycobacterium tuberculosis Strains

Inhibitors of the sulfur assimilation pathway in bacterial pathogens as enhancers of antibiotic therapy

Nitric oxide-releasing cyclodextrins as biodegradable antibacterial scaffolds: a patent evaluation of US2019343869(A1)

Inhibitors of O-Acetylserine Sulfhydrylase with a Cyclopropane-Carboxylic Acid Scaffold Are Effective Colistin Adjuvants in Gram Negative Bacteria

Refining the structure−activity relationships of 2-phenylcyclopropane carboxylic acids as inhibitors of O-acetylserine sulfhydrylase isoforms

Discovery of Substituted (2-Aminooxazol-4-yl)Isoxazole-3-carboxylic Acids as Inhibitors of Bacterial Serine Acetyltransferase in the Quest for Novel Potential Antibacterial Adjuvants

Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand-based drug design

Discovering a new class of antifungal agents that selectively inhibits microbial carbonic anhydrases

Pyrido[1,2-a]benzimidazole-Based Agents Active Against Tuberculosis (TB), Multidrug-Resistant (MDR) TB and Extensively Drug-Resistant (XDR) TB

Derivatives of 3-isoxazolecarboxylic acid esters: a potent and selective compound class against replicating and nonreplicating Mycobacterium tuberculosis

Identification of Human Alanine–Glyoxylate Aminotransferase Ligands as Pharmacological Chaperones for Variants Associated with Primary Hyperoxaluria Type 1

Substituted N‑Phenyl-5-(2-(phenylamino)thiazol-4-yl)isoxazole-3-carboxamides Are Valuable Antitubercular Candidates that Evade Innate Efflux Machinery

Design, synthesis and investigation on the structure–activity relationships of N-substituted 2-aminothiazole derivatives as antitubercular agents

Rational Design and Synthesis of Thioridazine Analogues as Enhancers of the Antituberculosis Therapy

Integration of Enhanced Sampling Methods with Saturation Transfer Difference Experiments to Identify Protein Druggable Pockets

2‑Aminooxazole as a Novel Privileged Scaffold in Antitubercular Medicinal Chemistry

Chemical Probes to Investigate Central Nervous System Disorders: Design, Synthesis and Mechanism of Action of a Potent Human Serine Racemase Inhibitor

Rational Design, Synthesis, and Preliminary Structure–Activity Relationships of α‑Substituted-2-Phenylcyclopropane Carboxylic Acids as Inhibitors of Salmonella typhimurium O‑Acetylserine Sulfhydrylase

Discovery of antitubercular 2,4-diphenyl-1H-imidazoles from chemical library repositioning and rational design

Expanding the knowledge around antitubercular 5-(2-aminothiazol-4-yl)isoxazole-3-carboxamides: Hit–to–lead optimization and release of a novel antitubercular chemotype via scaffold derivatization

Discovery of New Potential Anti-Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target-Focused Repurposing Approaches

Further insights into the SAR of α-substituted cyclopropylamine derivatives as inhibitors of histone demethylase KDM1A

Preliminary structure−activity relationships analysis on N-(3,5-dichlorophenyl)-4,5-dihydronaphtho[1,2-d]thiazol-2-amine, a disruptor of mycobacterial energetics

Rational Design of 5-Phenyl-3-isoxazolecarboxylic Acid Ethyl Esters as Growth Inhibitors of Mycobacterium tuberculosis. A Potent and Selective Series for Further Drug Development

Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O‑Acetyltransferase Inhibitor

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