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Challenging the Drug-Likeness Dogma for New Drug Discovery in Tuberculosis

Frontiers in microbiology, 2018-07, Vol.9, p.1367-1367

2018

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Indoleamides are active against drug-resistant Mycobacterium tuberculosis

Nature communications, 2013-12, Vol.4 (1), Article 2907

2013

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Cycloserine enantiomers are reversible inhibitors of human alanine:glyoxylate aminotransferase: implications for Primary Hyperoxaluria type 1

Biochemical journal, 2019-12, Vol.476 (24), p.3751-3768

2019

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Sodium Hyaluronate Nanocomposite Respirable Microparticles to Tackle Antibiotic Resistance with Potential Application in Treatment of Mycobacterial Pulmonary Infections

Pharmaceutics, 2019-05, Vol.11 (5), p.203

2019

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Inhibitors of O-Acetylserine Sulfhydrylase with a Cyclopropane-Carboxylic Acid Scaffold Are Effective Colistin Adjuvants in Gram Negative Bacteria

Pharmaceuticals (Basel, Switzerland), 2022-06, Vol.15 (6), p.766

2022

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Refining the structure−activity relationships of 2-phenylcyclopropane carboxylic acids as inhibitors of O-acetylserine sulfhydrylase isoforms

Journal of enzyme inhibition and medicinal chemistry, 2019-01, Vol.34 (1), p.31-43

2019

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Discovery of Substituted (2-Aminooxazol-4-yl)Isoxazole-3-carboxylic Acids as Inhibitors of Bacterial Serine Acetyltransferase in the Quest for Novel Potential Antibacterial Adjuvants

Pharmaceuticals (Basel, Switzerland), 2021-02, Vol.14 (2), p.174

2021

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Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand-based drug design

Journal of enzyme inhibition and medicinal chemistry, 2018-01, Vol.33 (1), p.1444-1452

2018

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A Competitive O-Acetylserine Sulfhydrylase Inhibitor Modulates the Formation of Cysteine Synthase Complex

Catalysts, 2021-06, Vol.11 (6), p.700

2021

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Efflux Activity Differentially Modulates the Levels of Isoniazid and Rifampicin Resistance among Multidrug Resistant and Monoresistant Mycobacterium tuberculosis Strains

Antibiotics (Basel), 2018-03, Vol.7 (1), p.18

2018

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Synthesis of 7-Desmethyl Analogs of (+)- and (−)-Huperzine A

Heterocycles, 2015, Vol.91 (12), p.2285

2015

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Biochemical Characterization of Aspergillus fumigatus AroH, a Putative Aromatic Amino Acid Aminotransferase

Frontiers in molecular biosciences, 2018-11, Vol.5, p.104-104

2018

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Identification of Human Alanine–Glyoxylate Aminotransferase Ligands as Pharmacological Chaperones for Variants Associated with Primary Hyperoxaluria Type 1

Journal of medicinal chemistry, 2022-07, Vol.65 (14), p.9718-9734

2022

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2‑Aminooxazole as a Novel Privileged Scaffold in Antitubercular Medicinal Chemistry

ACS medicinal chemistry letters, 2020-07, Vol.11 (7), p.1435-1441

2020

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Chemical Probes to Investigate Central Nervous System Disorders: Design, Synthesis and Mechanism of Action of a Potent Human Serine Racemase Inhibitor

ACS medicinal chemistry letters, 2024-07

2024

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Preliminary structure−activity relationships analysis on N-(3,5-dichlorophenyl)-4,5-dihydronaphtho[1,2-d]thiazol-2-amine, a disruptor of mycobacterial energetics

Medicinal chemistry research, 2024-03, Vol.33 (3), p.518-531

2024

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Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O‑Acetyltransferase Inhibitor

ACS medicinal chemistry letters, 2020-05, Vol.11 (5), p.790-797

2020

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Adjuvant therapies against tuberculosis: discovery of a 2-aminothiazole targeting

Future microbiology, 2018-09, Vol.13 (12), p.1383-1402

2018

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Cover Picture: Discovery of New Potential Anti-Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target-Focused Repurposing Approaches (ChemMedChem 17/2016)

ChemMedChem, 2016-09, Vol.11 (17), p.1876-1876

2016

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In vitro Digestion of Zingiber officinale Extract and Evaluation of Stability as a First Step to Determine its Bioaccesibility

Natural product communications, 2018-09, Vol.13 (9), p.1934578

2018

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Searching for innovative quinolone-like scaffolds: synthesis and biological evaluation of 2,1-benzothiazine 2,2-dioxide derivatives

MedChemComm, 2012-09, Vol.3 (9), p.1092

2012

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Correction to From 6-Aminoquinolone Antibacterials to 6-Amino-7-thiopyranopyridinylquinolone Ethyl Esters as Inhibitors of Staphylococcus aureus Multidrug Efflux Pumps

Journal of medicinal chemistry, 2011-03, Vol.54 (5), p.1537-1537

2011

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Searching for innovative quinolone-like scaffolds: synthesis and biological evaluation of 2,1-benzothiazine 2,2-dioxide derivativesElectronic supplementary information (ESI) available: Microbiologic procedures, EtBr Efflux inhibition assay, full experimental part, spectral data, elemental analyses and LC-MS analyses. See DOI: 10.1039/c2md20101a

2012-08

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Causes and consequences of oil price shocks on the UK economy

Economic modelling, 2018-06, Vol.72, p.223-236

2018

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The effects of military and non-military government expenditures on private consumption

Journal of peace research, 2017-05, Vol.54 (3), p.442-456

2017

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Challenging the Drug-Likeness Dogma for New Drug Discovery in Tuberculosis

Indoleamides are active against drug-resistant Mycobacterium tuberculosis

Cycloserine enantiomers are reversible inhibitors of human alanine:glyoxylate aminotransferase: implications for Primary Hyperoxaluria type 1

Sodium Hyaluronate Nanocomposite Respirable Microparticles to Tackle Antibiotic Resistance with Potential Application in Treatment of Mycobacterial Pulmonary Infections

Inhibitors of O-Acetylserine Sulfhydrylase with a Cyclopropane-Carboxylic Acid Scaffold Are Effective Colistin Adjuvants in Gram Negative Bacteria

Refining the structure−activity relationships of 2-phenylcyclopropane carboxylic acids as inhibitors of O-acetylserine sulfhydrylase isoforms

Discovery of Substituted (2-Aminooxazol-4-yl)Isoxazole-3-carboxylic Acids as Inhibitors of Bacterial Serine Acetyltransferase in the Quest for Novel Potential Antibacterial Adjuvants

Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand-based drug design

A Competitive O-Acetylserine Sulfhydrylase Inhibitor Modulates the Formation of Cysteine Synthase Complex

Efflux Activity Differentially Modulates the Levels of Isoniazid and Rifampicin Resistance among Multidrug Resistant and Monoresistant Mycobacterium tuberculosis Strains

Synthesis of 7-Desmethyl Analogs of (+)- and (−)-Huperzine A

Biochemical Characterization of Aspergillus fumigatus AroH, a Putative Aromatic Amino Acid Aminotransferase

Identification of Human Alanine–Glyoxylate Aminotransferase Ligands as Pharmacological Chaperones for Variants Associated with Primary Hyperoxaluria Type 1

2‑Aminooxazole as a Novel Privileged Scaffold in Antitubercular Medicinal Chemistry

Chemical Probes to Investigate Central Nervous System Disorders: Design, Synthesis and Mechanism of Action of a Potent Human Serine Racemase Inhibitor

Preliminary structure−activity relationships analysis on N-(3,5-dichlorophenyl)-4,5-dihydronaphtho[1,2-d]thiazol-2-amine, a disruptor of mycobacterial energetics

Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O‑Acetyltransferase Inhibitor

Adjuvant therapies against tuberculosis: discovery of a 2-aminothiazole targeting

Cover Picture: Discovery of New Potential Anti-Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target-Focused Repurposing Approaches (ChemMedChem 17/2016)

In vitro Digestion of Zingiber officinale Extract and Evaluation of Stability as a First Step to Determine its Bioaccesibility

Searching for innovative quinolone-like scaffolds: synthesis and biological evaluation of 2,1-benzothiazine 2,2-dioxide derivatives

Correction to From 6-Aminoquinolone Antibacterials to 6-Amino-7-thiopyranopyridinylquinolone Ethyl Esters as Inhibitors of Staphylococcus aureus Multidrug Efflux Pumps

Causes and consequences of oil price shocks on the UK economy

The effects of military and non-military government expenditures on private consumption

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