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4-(2-[2-(2(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl)benzonitrile and Related 2-Aminoethylbenzofuran H3 Receptor Antagonists Potently Enhance Cognition and Attention

Journal of medicinal chemistry, 2005-01, Vol.48 (1), p.38-55

2005

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Perspectives on cognitive domains, H3 receptor ligands and neurological disease

Expert opinion on investigational drugs, 2004-10, Vol.13 (10), p.1237-1248

2004

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Two novel and selective nonimidazole H3 receptor antagonists A-304121 and A-317920: II. In vivo behavioral and neurophysiological characterization

The Journal of pharmacology and experimental therapeutics, 2003-06, Vol.305 (3), p.897

2003

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An 80-amino acid deletion in the third intracellular loop of a naturally occurring human histamine H3 isoform confers pharmacological differences and constitutive activity

The Journal of pharmacology and experimental therapeutics, 2007-12, Vol.323 (3), p.888

2007

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Two novel and selective nonimidazole histamine H3 receptor antagonists A-304121 and A-317920: I. In vitro pharmacological effects

The Journal of pharmacology and experimental therapeutics, 2003-06, Vol.305 (3), p.887

2003

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G protein-dependent pharmacology of histamine H3 receptor ligands: evidence for heterogeneous active state receptor conformations

The Journal of pharmacology and experimental therapeutics, 2005-07, Vol.314 (1), p.271

2005

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Design of a New Histamine H3 Receptor Antagonist Chemotype: (3aR,6aR)-5-Alkyl-1-aryl-octahydropyrrolo[3,4-b]pyrroles, Synthesis, and Structure−Activity Relationships

Journal of medicinal chemistry, 2009-08, Vol.52 (15), p.4640-4649

2009

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An Efficient Multigram Synthesis of the Potent Histamine H3 Antagonist GT-2331 and the Reassessment of the Absolute Configuration

Journal of organic chemistry, 2004-01, Vol.69 (1), p.192-194

2004

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Pharmacological properties and procognitive effects of ABT-288, a potent and selective histamine H3 receptor antagonist

The Journal of pharmacology and experimental therapeutics, 2012-10, Vol.343 (1), p.233

2012

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Use of a fluorescent imaging plate reader--based calcium assay to assess pharmacological differences between the human and rat vanilloid receptor

Journal of biomolecular screening, 2002-10, Vol.7 (5), p.466-475

2002

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Assessment of pharmacology and potential anti-obesity properties of H3 receptor antagonists/inverse agonists

Expert opinion on investigational drugs, 2005-03, Vol.14 (3), p.223-241

2005

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Structure−Activity Studies on a Series of a 2-Aminopyrimidine-Containing Histamine H4 Receptor Ligands

Journal of medicinal chemistry, 2008-10, Vol.51 (20), p.6571-6580

2008

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The Alkaloid Conessine and Analogues as Potent Histamine H3 Receptor Antagonists

Journal of medicinal chemistry, 2008-09, Vol.51 (17), p.5423-5430

2008

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Medicinal chemistry and biological properties of non-imidazole histamine H3 antagonists

Mini reviews in medicinal chemistry, 2004-11, Vol.4 (9), p.979

2004

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Synthesis and SAR of 5-Amino- and 5-(Aminomethyl)benzofuran Histamine H3 Receptor Antagonists with Improved Potency

Journal of medicinal chemistry, 2005-10, Vol.48 (20), p.6482-6490

2005

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Detection of multiple H 3 receptor affinity states utilizing [ 3 H]A‐349821, a novel, selective, non‐imidazole histamine H 3 receptor inverse agonist radioligand

British journal of pharmacology, 2009-01, Vol.148 (5), p.657-670

2009

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Synthesis, Potency, and In Vivo Profiles of Quinoline Containing Histamine H3 Receptor Inverse Agonists

Journal of medicinal chemistry, 2007-11, Vol.50 (22), p.5439-5448

2007

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H3 receptor antagonists/inverse agonists as anti-obesity agents

Current opinion in investigational drugs (London, England : 2000), 2003-10, Vol.4 (10), p.1190

Hancock, Arthur A

2003

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Analysis of Apparent Noncompetitive Responses to Competitive H1-Histamine Receptor Antagonists in Fluorescent Imaging Plate Reader-Based Calcium Assays

SLAS discovery, 1999-10, Vol.4 (5), p.249-258

1999

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Structure−Activity Studies for a Novel Series of Tricyclic Substituted Hexahydrobenz[e]isoindole α1A Adrenoceptor Antagonists as Potential Agents for the Symptomatic Treatment of Benign Prostatic Hyperplasia (BPH)

Journal of medicinal chemistry, 2000-04, Vol.43 (8), p.1586-1603

2000

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In vitro Optimization of Structure Activity Relationships of Analogues of A‐331440 Combining Radioligand Receptor Binding Assays and Micronucleus Assays of Potential Antiobesity Histamine H3 Receptor Antagonists

Basic & clinical pharmacology & toxicology, 2004-09, Vol.95 (3), p.144-152

2004

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Detection of multiple H3 receptor affinity states utilizing [3H]A‐349821, a novel, selective, non‐imidazole histamine H3 receptor inverse agonist radioligand

British journal of pharmacology, 2006-07, Vol.148 (5), p.657-670

2006

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COMPARISON OF α1-ADRENOCEPTOR AGONISTS IN CANINE URETHRAL PRESSURE PROFILOMETRY AND ABDOMINAL LEAK POINT PRESSURE MODELS

The Journal of urology, 2001, Vol.166 (4), p.1555-1559

2001

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H3 receptor blockade by thioperamide enhances cognition in rats without inducing locomotor sensitization

Psychopharmacologia, 2003-06, Vol.167 (4), p.363-372

2003

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4-(2-[2-(2(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl)benzonitrile and Related 2-Aminoethylbenzofuran H3 Receptor Antagonists Potently Enhance Cognition and Attention

Perspectives on cognitive domains, H3 receptor ligands and neurological disease

Two novel and selective nonimidazole H3 receptor antagonists A-304121 and A-317920: II. In vivo behavioral and neurophysiological characterization

An 80-amino acid deletion in the third intracellular loop of a naturally occurring human histamine H3 isoform confers pharmacological differences and constitutive activity

Two novel and selective nonimidazole histamine H3 receptor antagonists A-304121 and A-317920: I. In vitro pharmacological effects

G protein-dependent pharmacology of histamine H3 receptor ligands: evidence for heterogeneous active state receptor conformations

Design of a New Histamine H3 Receptor Antagonist Chemotype: (3aR,6aR)-5-Alkyl-1-aryl-octahydropyrrolo[3,4-b]pyrroles, Synthesis, and Structure−Activity Relationships

An Efficient Multigram Synthesis of the Potent Histamine H3 Antagonist GT-2331 and the Reassessment of the Absolute Configuration

Pharmacological properties and procognitive effects of ABT-288, a potent and selective histamine H3 receptor antagonist

Pharmacological properties of ABT-239 [4-(2-{2-[(2R)-2-Methylpyrrolidinyl]ethyl}-benzofuran-5-yl)benzonitrile]: II. Neurophysiological characterization and broad preclinical efficacy in cognition and schizophrenia of a potent and selective histamine H3 receptor antagonist

Use of a fluorescent imaging plate reader--based calcium assay to assess pharmacological differences between the human and rat vanilloid receptor

Assessment of pharmacology and potential anti-obesity properties of H3 receptor antagonists/inverse agonists

Structure−Activity Studies on a Series of a 2-Aminopyrimidine-Containing Histamine H4 Receptor Ligands

The Alkaloid Conessine and Analogues as Potent Histamine H3 Receptor Antagonists

Medicinal chemistry and biological properties of non-imidazole histamine H3 antagonists

Synthesis and SAR of 5-Amino- and 5-(Aminomethyl)benzofuran Histamine H3 Receptor Antagonists with Improved Potency

Detection of multiple H 3 receptor affinity states utilizing [ 3 H]A‐349821, a novel, selective, non‐imidazole histamine H 3 receptor inverse agonist radioligand

Synthesis, Potency, and In Vivo Profiles of Quinoline Containing Histamine H3 Receptor Inverse Agonists

H3 receptor antagonists/inverse agonists as anti-obesity agents

Analysis of Apparent Noncompetitive Responses to Competitive H1-Histamine Receptor Antagonists in Fluorescent Imaging Plate Reader-Based Calcium Assays

Structure−Activity Studies for a Novel Series of Tricyclic Substituted Hexahydrobenz[e]isoindole α1A Adrenoceptor Antagonists as Potential Agents for the Symptomatic Treatment of Benign Prostatic Hyperplasia (BPH)

In vitro Optimization of Structure Activity Relationships of Analogues of A‐331440 Combining Radioligand Receptor Binding Assays and Micronucleus Assays of Potential Antiobesity Histamine H3 Receptor Antagonists

Detection of multiple H3 receptor affinity states utilizing [3H]A‐349821, a novel, selective, non‐imidazole histamine H3 receptor inverse agonist radioligand

COMPARISON OF α1-ADRENOCEPTOR AGONISTS IN CANINE URETHRAL PRESSURE PROFILOMETRY AND ABDOMINAL LEAK POINT PRESSURE MODELS

H3 receptor blockade by thioperamide enhances cognition in rats without inducing locomotor sensitization

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