Details

Autor(en) / Beteiligte

• Wang, Xiao-Jian
• Tian, Yu-Lin
• Zhang, Qing-Yang
• Qi, Jian-Guo
• Yin, Da-Li

Titel

An efficient synthesis of substituted 1,4-diazepines by a Pd catalyzed amination and sequential hydrogenation condensation

Ist Teil von

• Chinese chemical letters, 2013-08, Vol.24 (8), p.743-746

Ort / Verlag

Elsevier B.V

Erscheinungsjahr

2013

Quelle

Alma/SFX Local Collection

Beschreibungen/Notizen

• An efficient synthesis of substituted 1,4-diazepines is developed.The accessible intermediates have been obtained via Pd-catalyzed amination.The subsequent hydrogenation and intramolecular condensation sequences could be conducted successively in one pot without special operation.The mild and general strategy enables the synthesis of various substituted 1,4-diazepines in high yields.