Details

Autor(en) / Beteiligte

• Saito, Akio
• Kasai, Jun
• Odaira, Yu
• Fukaya, Haruhiko
• Hanzawa, Yuji

Titel

Synthesis of 2,3-Dihydroquinolin-4(1H)-ones through Catalytic Metathesis of o-Alkynylanilines and Aldehydes

Ist Teil von

• Journal of organic chemistry, 2009-08, Vol.74 (15), p.5644-5647

Ort / Verlag

United States: American Chemical Society

Erscheinungsjahr

2009

Quelle

MEDLINE

Beschreibungen/Notizen

• SbF5−MeOH catalytic system efficiently promotes the alkyne−carbonyl metathesis of o-alkynylaniline derivatives and aldehydes to afford 2,3-disubstituted dihydroquinolinones in moderate to high yields with high trans-selectivity.